CS200538B2 - Method of producing derivatives of oleandomycin - Google Patents

Method of producing derivatives of oleandomycin Download PDF

Info

Publication number
CS200538B2
CS200538B2 CS787694A CS769478A CS200538B2 CS 200538 B2 CS200538 B2 CS 200538B2 CS 787694 A CS787694 A CS 787694A CS 769478 A CS769478 A CS 769478A CS 200538 B2 CS200538 B2 CS 200538B2
Authority
CS
Czechoslovakia
Prior art keywords
deoxy
singlet
oxooleandomycin
added
acetyl
Prior art date
Application number
CS787694A
Other languages
Czech (cs)
English (en)
Inventor
Frank Ch Sciavolino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of CS200538B2 publication Critical patent/CS200538B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CS787694A 1977-02-04 1978-01-16 Method of producing derivatives of oleandomycin CS200538B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/765,486 US4125705A (en) 1977-02-04 1977-02-04 Semi-synthetic 4-amino-oleandomycin derivatives

Publications (1)

Publication Number Publication Date
CS200538B2 true CS200538B2 (en) 1980-09-15

Family

ID=25073683

Family Applications (3)

Application Number Title Priority Date Filing Date
CS787693A CS200537B2 (en) 1977-02-04 1978-01-16 Method of producing epimeric 4-amino oleandomycin derivatives
CS78291A CS200536B2 (en) 1977-02-04 1978-01-16 Method of producing epimeric 4-amino oleandomycin derivatives
CS787694A CS200538B2 (en) 1977-02-04 1978-01-16 Method of producing derivatives of oleandomycin

Family Applications Before (2)

Application Number Title Priority Date Filing Date
CS787693A CS200537B2 (en) 1977-02-04 1978-01-16 Method of producing epimeric 4-amino oleandomycin derivatives
CS78291A CS200536B2 (en) 1977-02-04 1978-01-16 Method of producing epimeric 4-amino oleandomycin derivatives

Country Status (34)

Country Link
US (1) US4125705A (de)
JP (2) JPS5398981A (de)
AR (1) AR215666A1 (de)
AT (1) AT358169B (de)
AU (1) AU502293B1 (de)
BE (1) BE863618A (de)
BG (2) BG32116A3 (de)
CA (1) CA1106366A (de)
CH (1) CH629821A5 (de)
CS (3) CS200537B2 (de)
DD (1) DD134523A5 (de)
DE (1) DE2804509C2 (de)
DK (1) DK149628C (de)
ES (1) ES465322A1 (de)
FI (1) FI65262C (de)
FR (2) FR2383964A1 (de)
GB (1) GB1583921A (de)
GR (1) GR68692B (de)
HU (2) HU181395B (de)
IE (1) IE46395B1 (de)
IL (2) IL53959A0 (de)
IT (1) IT1094211B (de)
LU (1) LU79007A1 (de)
NL (1) NL175997C (de)
NO (2) NO145955C (de)
NZ (1) NZ186384A (de)
PH (2) PH14836A (de)
PL (3) PL113163B1 (de)
PT (1) PT67569B (de)
RO (3) RO79264A (de)
SE (2) SE445222B (de)
SU (3) SU805949A3 (de)
YU (3) YU39504B (de)
ZA (1) ZA78646B (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4133950A (en) * 1978-01-03 1979-01-09 Pfizer Inc. 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4413119A (en) * 1982-03-01 1983-11-01 Pfizer Inc. Semi-synthetic macrolides
US4363803A (en) * 1982-03-01 1982-12-14 Pfizer Inc. 3",4"-Oxyallylene erythromycin and oleandomycin, composition and method of use
JPH0240447U (de) * 1988-09-14 1990-03-19
US5141926A (en) * 1990-04-18 1992-08-25 Abbott Laboratories Erythromycin derivatives
JPH05155896A (ja) * 1991-01-18 1993-06-22 Yamanouchi Pharmaceut Co Ltd 新規マクロライド化合物及びその製造法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3022219A (en) * 1958-03-07 1962-02-20 Pfizer & Co C Acyl esters of oleandomycin
US3179652A (en) * 1961-09-05 1965-04-20 Pfizer & Co C Antibiotic recovery process and salts produced thereby
US3836519A (en) * 1973-05-04 1974-09-17 Abbott Lab Sulfonyl derivatives of erythromycin
US3842069A (en) * 1973-06-21 1974-10-15 Abbott Lab 4"-deoxy-4"-oxoerythromycin b derivatives
US4036853A (en) * 1976-08-06 1977-07-19 Pfizer Inc. Semi-synthetic oleandomycin derivatives-C8 modifications

Also Published As

Publication number Publication date
IE46395B1 (en) 1983-06-01
SE8300869D0 (sv) 1983-02-16
AR215666A1 (es) 1979-10-31
NO150439B (no) 1984-07-09
DK149628C (da) 1987-02-02
DE2804509A1 (de) 1978-08-10
JPS56135497A (en) 1981-10-22
IL61606A0 (en) 1981-01-30
SE7800269L (sv) 1978-08-05
GR68692B (de) 1982-02-01
IT7820006A0 (it) 1978-02-03
IT1094211B (it) 1985-07-26
IL53959A0 (en) 1978-04-30
YU39504B (en) 1984-12-31
FR2383964A1 (fr) 1978-10-13
JPS5827799B2 (ja) 1983-06-11
JPS5652036B2 (de) 1981-12-09
PH16491A (en) 1983-10-28
AT358169B (de) 1980-08-25
NO150439C (no) 1984-10-17
YU300377A (en) 1982-10-31
ZA78646B (en) 1978-12-27
YU39518B (en) 1984-12-31
NL175997C (nl) 1985-02-01
GB1583921A (en) 1981-02-04
YU39517B (en) 1984-12-31
IE780240L (en) 1978-08-04
AU502293B1 (en) 1979-07-19
CA1106366A (en) 1981-08-04
NO145955C (no) 1982-06-30
SU805949A3 (ru) 1981-02-15
DK149628B (da) 1986-08-18
FI780355A (fi) 1978-08-05
BG32116A3 (en) 1982-05-14
YU151782A (en) 1982-10-31
DD134523A5 (de) 1979-03-07
SE445222B (sv) 1986-06-09
HU179744B (en) 1982-12-28
BE863618A (fr) 1978-08-03
US4125705A (en) 1978-11-14
FR2396022A1 (fr) 1979-01-26
PT67569A (en) 1978-02-01
JPS5398981A (en) 1978-08-29
FR2383964B1 (de) 1981-11-27
RO79258A (ro) 1982-06-25
ES465322A1 (es) 1978-09-16
YU151882A (en) 1982-10-31
NL175997B (nl) 1984-09-03
FI65262C (fi) 1984-04-10
BG32117A4 (en) 1982-05-14
DE2804509C2 (de) 1982-12-02
PL113163B1 (en) 1980-11-29
NO780390L (no) 1978-08-07
ATA72078A (de) 1980-01-15
FI65262B (fi) 1983-12-30
FR2396022B1 (de) 1980-06-13
CS200537B2 (en) 1980-09-15
SE457085B (sv) 1988-11-28
CS200536B2 (en) 1980-09-15
NZ186384A (en) 1980-08-26
PH14836A (en) 1981-12-16
PL204041A1 (pl) 1979-06-04
PL111160B1 (en) 1980-08-30
SU888824A3 (ru) 1981-12-07
LU79007A1 (fr) 1979-09-06
PL110793B1 (en) 1980-07-31
HU181395B (en) 1983-07-28
CH629821A5 (fr) 1982-05-14
NO811914L (no) 1978-08-07
RO79264A (ro) 1982-06-25
PT67569B (en) 1979-06-18
NO145955B (no) 1982-03-22
SU1020004A3 (ru) 1983-05-23
DK51778A (da) 1978-08-05
RO75387A (ro) 1980-11-30
NL7801259A (nl) 1978-08-08

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