CR10782A - Compuestos para inhibir la progresion mitotica - Google Patents

Compuestos para inhibir la progresion mitotica

Info

Publication number
CR10782A
CR10782A CR10782A CR10782A CR10782A CR 10782 A CR10782 A CR 10782A CR 10782 A CR10782 A CR 10782A CR 10782 A CR10782 A CR 10782A CR 10782 A CR10782 A CR 10782A
Authority
CR
Costa Rica
Prior art keywords
compounds
mythical
progression
inhibit
cancer
Prior art date
Application number
CR10782A
Other languages
English (en)
Spanish (es)
Inventor
Christopher F Claiborne
Todd B Sells
Stephen G Stroud
Original Assignee
Millenium Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39315133&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR10782(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Millenium Pharmaceuticals Inc filed Critical Millenium Pharmaceuticals Inc
Publication of CR10782A publication Critical patent/CR10782A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CR10782A 2006-11-16 2009-05-08 Compuestos para inhibir la progresion mitotica CR10782A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US85934006P 2006-11-16 2006-11-16

Publications (1)

Publication Number Publication Date
CR10782A true CR10782A (es) 2009-06-24

Family

ID=39315133

Family Applications (3)

Application Number Title Priority Date Filing Date
CR10782A CR10782A (es) 2006-11-16 2009-05-08 Compuestos para inhibir la progresion mitotica
CR20140154A CR20140154A (es) 2006-11-16 2014-04-04 Compuestos para inhibir la progresión mitotica
CR20140544A CR20140544A (es) 2006-11-16 2014-11-27 Compuestos para inhibir la progresión mitotica

Family Applications After (2)

Application Number Title Priority Date Filing Date
CR20140154A CR20140154A (es) 2006-11-16 2014-04-04 Compuestos para inhibir la progresión mitotica
CR20140544A CR20140544A (es) 2006-11-16 2014-11-27 Compuestos para inhibir la progresión mitotica

Country Status (34)

Country Link
US (7) US8026246B2 (https=)
EP (4) EP2086981B1 (https=)
JP (3) JP5102839B2 (https=)
KR (2) KR101342014B1 (https=)
CN (2) CN103483343B (https=)
AR (1) AR064246A1 (https=)
AT (1) ATE556076T1 (https=)
AU (1) AU2007322046B2 (https=)
BR (1) BRPI0718803B8 (https=)
CA (1) CA2669680C (https=)
CL (1) CL2007003244A1 (https=)
CR (3) CR10782A (https=)
CY (1) CY1112828T1 (https=)
DK (2) DK2497772T3 (https=)
EA (1) EA015779B1 (https=)
ES (3) ES2528793T3 (https=)
GE (1) GEP20125459B (https=)
HR (2) HRP20120490T1 (https=)
IL (1) IL198690A0 (https=)
MA (1) MA30988B1 (https=)
MX (3) MX343391B (https=)
MY (1) MY153243A (https=)
NO (1) NO343338B1 (https=)
NZ (3) NZ577042A (https=)
PH (1) PH12012502057B1 (https=)
PL (2) PL2086981T3 (https=)
PT (2) PT2086981E (https=)
RS (2) RS52313B (https=)
SG (2) SG176443A1 (https=)
SI (2) SI2497772T1 (https=)
TW (1) TWI401255B (https=)
UA (1) UA94129C2 (https=)
WO (1) WO2008063525A1 (https=)
ZA (1) ZA200903279B (https=)

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JO3434B1 (ar) 2009-07-31 2019-10-20 Millennium Pharm Inc مركبات صيدلانية لمعالجة السرطان وامراض واضطرابات اخري
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US20120107304A1 (en) 2010-04-27 2012-05-03 Boehringer Ingelheim International Gmbh Combination therapy in treatment of oncological and fibrotic diseases
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AR086656A1 (es) 2011-06-03 2014-01-15 Millennium Pharm Inc Combinacion de inhibidores de mek e inhibidores selectivos de la quinasa aurora a
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CN103772391A (zh) * 2012-10-23 2014-05-07 杨子娇 一类治疗房角狭窄的化合物及其用途
WO2014153509A1 (en) 2013-03-22 2014-09-25 Millennium Pharmaceuticals, Inc. Combination of catalytic mtorc 1/2 inhibitors and selective inhibitors of aurora a kinase
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WO2016106357A1 (en) * 2014-12-23 2016-06-30 Millennnium Pharmaceuticals, Inc. Combination of raf inhibitors and aurora kinase inhibitors
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CA2997769A1 (en) 2015-09-09 2017-03-16 Icahn School Of Medicine At Mount Sinai Heterocyclic constrained tricyclic sulfonamides as anti-cancer agents
CA2997784A1 (en) 2015-09-09 2017-03-16 Icahn School Of Medicine At Mount Sinai Heterocyclic constrained tricyclic sulfonamides as anti-cancer agents
JP6591036B2 (ja) 2016-02-26 2019-10-16 公益財団法人がん研究会 Ｈｐ１の機能に着目した抗癌剤のスクリーニング方法及び評価系
ES3057783T3 (en) 2016-03-15 2026-03-04 Oryzon Genomics Sa Combinations of lsd1 inhibitors for use in the treatment of neoplastic diseases
JP6188986B1 (ja) * 2017-03-23 2017-08-30 株式会社ノエビア 時計遺伝子発現量調整剤及びエラスチン産生促進剤
US11874276B2 (en) 2018-04-05 2024-01-16 Dana-Farber Cancer Institute, Inc. STING levels as a biomarker for cancer immunotherapy
WO2020049208A1 (es) 2018-09-09 2020-03-12 Fundacio Privada Institut De Recerca De La Sida - Caixa Aurora cinasa como diana para tratar, prevenir o curar una infección por vih o sida
US20220305048A1 (en) 2019-08-26 2022-09-29 Dana-Farber Cancer Institute, Inc. Use of heparin to promote type 1 interferon signaling
JP2025511697A (ja) 2022-04-07 2025-04-16 イーライ リリー アンド カンパニー Ｋｒａｓ ｇ１２ｃ阻害剤を作製するための方法
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Also Published As

Publication number Publication date
US20110312942A1 (en) 2011-12-22
PH12012502057B1 (en) 2018-10-24
BRPI0718803B8 (pt) 2021-05-25
NZ611898A (en) 2015-01-30
CR20140154A (es) 2014-07-23
PH12012502057A1 (en) 2015-09-14
JP2012006965A (ja) 2012-01-12
CN103483343A (zh) 2014-01-01
US8026246B2 (en) 2011-09-27
MX2009004670A (es) 2009-05-15
PT2086981E (pt) 2012-06-20
MY153243A (en) 2015-01-29
US20150166545A1 (en) 2015-06-18
CY1112828T1 (el) 2016-02-10
JP5452811B2 (ja) 2014-03-26
CA2669680A1 (en) 2008-05-29
EP2086981B1 (en) 2012-05-02
EP2497773B1 (en) 2015-02-25
UA94129C2 (ru) 2011-04-11
MX343391B (es) 2016-11-04
WO2008063525A1 (en) 2008-05-29
SG176443A1 (en) 2011-12-29
KR101342014B1 (ko) 2013-12-19
PL2497772T3 (pl) 2015-05-29
US20110312943A1 (en) 2011-12-22
JP5102839B2 (ja) 2012-12-19
HK1175777A1 (en) 2013-07-12
US9765076B2 (en) 2017-09-19
KR20090091173A (ko) 2009-08-26
CA2669680C (en) 2012-04-10
PL2086981T3 (pl) 2012-09-28
CN101547924A (zh) 2009-09-30
ES2384123T3 (es) 2012-06-29
AU2007322046B2 (en) 2012-04-05
SG10201503350TA (en) 2015-06-29
CN101547924B (zh) 2013-09-25
NZ597252A (en) 2013-06-28
KR20110113210A (ko) 2011-10-14
EA015779B1 (ru) 2011-12-30
KR101110458B1 (ko) 2012-03-13
HK1217699A1 (en) 2017-01-20
EP2497772B1 (en) 2014-10-29
JP2010510215A (ja) 2010-04-02
ES2528793T3 (es) 2015-02-12
NO343338B1 (no) 2019-02-04
US10836766B2 (en) 2020-11-17
PT2497772E (pt) 2015-02-05
CL2007003244A1 (es) 2008-04-04
HK1134672A1 (en) 2010-05-07
US20210214361A1 (en) 2021-07-15
EP2086981A1 (en) 2009-08-12
EP2497773A1 (en) 2012-09-12
US9988384B2 (en) 2018-06-05
US20080167292A1 (en) 2008-07-10
AR064246A1 (es) 2009-03-25
HRP20120490T1 (hr) 2012-07-31
RS53788B1 (sr) 2015-06-30
DK2086981T3 (da) 2012-08-06
CN103483343B (zh) 2016-06-01
TW200829589A (en) 2008-07-16
JP2014055166A (ja) 2014-03-27
US20190031662A1 (en) 2019-01-31
SI2497772T1 (sl) 2015-03-31
ATE556076T1 (de) 2012-05-15
AU2007322046A1 (en) 2008-05-29
SI2086981T1 (sl) 2012-12-31
US20240400567A1 (en) 2024-12-05
GEP20125459B (en) 2012-03-26
HRP20150047T1 (en) 2015-03-13
TWI401255B (zh) 2013-07-11
CR20140544A (es) 2015-01-12
NZ577042A (en) 2012-03-30
BRPI0718803B1 (pt) 2020-11-17
HK1175778A1 (en) 2013-07-12
MA30988B1 (fr) 2009-12-01
ES2537451T3 (es) 2015-06-08
US11958855B2 (en) 2024-04-16
EP2944639A1 (en) 2015-11-18
ZA200903279B (en) 2010-07-28
EP2944639B1 (en) 2017-01-04
MX348568B (es) 2017-06-20
NO20091864L (no) 2009-06-15
BRPI0718803A2 (pt) 2013-12-03
RS52313B (sr) 2012-12-31
DK2497772T3 (en) 2015-01-19
IL198690A0 (en) 2010-02-17
EA200970486A1 (ru) 2009-10-30
EP2497772A1 (en) 2012-09-12

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