CO6751253A2 - Proceso para preparar una amida de un ácido carboxílico pirazólico - Google Patents

Proceso para preparar una amida de un ácido carboxílico pirazólico

Info

Publication number
CO6751253A2
CO6751253A2 CO13173578A CO13173578A CO6751253A2 CO 6751253 A2 CO6751253 A2 CO 6751253A2 CO 13173578 A CO13173578 A CO 13173578A CO 13173578 A CO13173578 A CO 13173578A CO 6751253 A2 CO6751253 A2 CO 6751253A2
Authority
CO
Colombia
Prior art keywords
formula
compound
res
oxygen
amide
Prior art date
Application number
CO13173578A
Other languages
English (en)
Inventor
Miroslav Terinek
Dominik Faber
Stefan Koening
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of CO6751253A2 publication Critical patent/CO6751253A2/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/14—Preparation of carboxylic acid amides by formation of carboxamide groups together with reactions not involving the carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/50—Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals
    • C07C251/56—Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals of hydrocarbon radicals substituted by doubly-bound oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/62—Oximes having oxygen atoms of oxyimino groups esterified
    • C07C251/64—Oximes having oxygen atoms of oxyimino groups esterified by carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C329/00—Thiocarbonic acids; Halides, esters or anhydrides thereof
    • C07C329/02—Monothiocarbonic acids; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C329/00—Thiocarbonic acids; Halides, esters or anhydrides thereof
    • C07C329/02—Monothiocarbonic acids; Derivatives thereof
    • C07C329/04—Esters of monothiocarbonic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

La invención se refiere a un proceso para preparar la (9-diclorometilen-1, 2, 3, 4-tetrahidro-1,4-metanonaftalen-5-il)amida del ácido 3-difluorometil-1-metil-1H-pirazol-4-carboxílico que comprende acilar el oxígeno de la oxima del compuesto de fórmula VIIIen presencia de un disolvente y un agente acilante de fórmula XI R-C(X)-Cl (XI); donde X es oxígeno o azufre; Res cloro si X es oxígeno o azufre; o Res alcoxi C-C, CH-C(=CH)-O-, fenoxi o triclorometoxi si X es oxígeno; y a) si Res cloro y el compuesto de fórmula XI se añadió al compuesto de fórmula VIII; hacer reaccionar el producto obtenido de este modo de fórmula XIIadonde X es oxígeno o azufre; con el compuesto de fórmula IXb) si Res cloro y el compuesto de fórmula VIII se añadió al compuesto de fórmula XI; o Res alxoxi C-C, CH-C(=CH)-O-, fenoxi o triclorometoxi si X es oxígeno; hacer reaccionar el producto obtenido de este modo de fórmula XII
CO13173578A 2011-01-25 2013-07-23 Proceso para preparar una amida de un ácido carboxílico pirazólico CO6751253A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP11151965 2011-01-25

Publications (1)

Publication Number Publication Date
CO6751253A2 true CO6751253A2 (es) 2013-09-16

Family

ID=45524566

Family Applications (1)

Application Number Title Priority Date Filing Date
CO13173578A CO6751253A2 (es) 2011-01-25 2013-07-23 Proceso para preparar una amida de un ácido carboxílico pirazólico

Country Status (19)

Country Link
US (1) US8895757B2 (es)
EP (1) EP2668166B1 (es)
JP (2) JP6133788B2 (es)
KR (1) KR101851781B1 (es)
CN (1) CN103339113B (es)
AR (1) AR084915A1 (es)
AU (1) AU2012210547B2 (es)
BR (1) BR112013018533A2 (es)
CA (1) CA2824730C (es)
CO (1) CO6751253A2 (es)
ES (1) ES2540211T3 (es)
HR (1) HRP20150658T1 (es)
IL (1) IL227317A (es)
MX (1) MX352697B (es)
PL (1) PL2668166T3 (es)
PT (1) PT2668166E (es)
TW (1) TWI534126B (es)
UY (1) UY33879A (es)
WO (1) WO2012101139A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI534126B (zh) * 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法
TWI510472B (zh) 2012-02-15 2015-12-01 Syngenta Participations Ag 立體選擇性製備吡唑羧醯胺之方法
WO2018179632A1 (ja) 2017-03-31 2018-10-04 日本精工株式会社 レーザ溶接装置、レーザ加工装置、レーザ溶接方法、軸受の製造方法、機械の製造方法、車両の製造方法、軸受、機械、及び車両
WO2024017788A1 (en) 2022-07-22 2024-01-25 Syngenta Crop Protection Ag Solid form of a heterocyclic amide derivative

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58194853A (ja) * 1982-05-11 1983-11-12 Showa Denko Kk シクロヘキセン−アセチルオキシム誘導体
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
GT200600468A (es) * 2005-10-25 2007-06-08 Nuevos microbiocidas
MX2010011790A (es) * 2008-05-14 2010-11-25 Syngenta Ltd Proceso para la preparacion de amidas.
CN102264705A (zh) * 2008-12-24 2011-11-30 辛根塔有限公司 制备芳基酰胺的方法
EP2462108B1 (en) 2009-08-06 2013-04-17 Syngenta Participations AG Process for the preparation of pyrazole carboxylic acid amides
US8524915B2 (en) * 2010-04-20 2013-09-03 Syngenta Crop Protection Llc Process for the preparation of pyrazole carboxylic acid amides
ES2513540T3 (es) * 2010-04-20 2014-10-27 Syngenta Participations Ag Proceso para preparar amidas de ácidos carboxílicos pirazólicos
CN102844306B (zh) * 2010-04-20 2015-01-14 先正达参股股份有限公司 吡唑羧酸酰胺的制备方法
TWI534126B (zh) * 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法

Also Published As

Publication number Publication date
TWI534126B (zh) 2016-05-21
PT2668166E (pt) 2015-08-27
PL2668166T3 (pl) 2015-09-30
JP6133788B2 (ja) 2017-05-24
ES2540211T3 (es) 2015-07-09
TW201245114A (en) 2012-11-16
AU2012210547A1 (en) 2013-08-01
IL227317A (en) 2014-11-30
MX2013007914A (es) 2013-08-29
KR101851781B1 (ko) 2018-04-24
HRP20150658T1 (hr) 2015-07-31
JP2017071614A (ja) 2017-04-13
IL227317A0 (en) 2013-09-30
AU2012210547B2 (en) 2016-04-14
UY33879A (es) 2012-08-31
EP2668166A1 (en) 2013-12-04
BR112013018533A2 (pt) 2016-07-12
US20130310592A1 (en) 2013-11-21
CA2824730A1 (en) 2012-08-02
JP6419131B2 (ja) 2018-11-07
WO2012101139A1 (en) 2012-08-02
MX352697B (es) 2017-12-05
JP2014504596A (ja) 2014-02-24
CN103339113A (zh) 2013-10-02
CA2824730C (en) 2018-10-23
EP2668166B1 (en) 2015-05-13
US8895757B2 (en) 2014-11-25
CN103339113B (zh) 2015-07-22
AR084915A1 (es) 2013-07-10
KR20140019333A (ko) 2014-02-14

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