CO6700822A2 - Proceso para preparar 3-haloalquilporazoles - Google Patents

Proceso para preparar 3-haloalquilporazoles

Info

Publication number
CO6700822A2
CO6700822A2 CO13024312A CO13024312A CO6700822A2 CO 6700822 A2 CO6700822 A2 CO 6700822A2 CO 13024312 A CO13024312 A CO 13024312A CO 13024312 A CO13024312 A CO 13024312A CO 6700822 A2 CO6700822 A2 CO 6700822A2
Authority
CO
Colombia
Prior art keywords
compound
formula
optionally substituted
haloalkylporazoles
prepare
Prior art date
Application number
CO13024312A
Other languages
English (en)
Inventor
Linhua Wang
Ritesh Bharat Sheth
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of CO6700822A2 publication Critical patent/CO6700822A2/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

La presente invención proporciona un proceso para preparar un compuesto de fórmula I:donde R1 es haloalquilo C1-C4;R2 es alquilo opcionalmente sustituido, arilo opcionalmente sustitu1do o heteroarilo opcionalmente sustituido; yR3 es metilo o etilo;que comprende hacer reaccionar un compuesto de fórmula IV:donde R1, R2 y R3 son como se definen para el compuesto de fórmula I; con un agente alquilante en presencia de una amida.
CO13024312A 2010-08-10 2013-02-06 Proceso para preparar 3-haloalquilporazoles CO6700822A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US37212210P 2010-08-10 2010-08-10

Publications (1)

Publication Number Publication Date
CO6700822A2 true CO6700822A2 (es) 2013-06-28

Family

ID=44503820

Family Applications (1)

Application Number Title Priority Date Filing Date
CO13024312A CO6700822A2 (es) 2010-08-10 2013-02-06 Proceso para preparar 3-haloalquilporazoles

Country Status (19)

Country Link
US (3) US9359304B2 (es)
EP (1) EP2603494B1 (es)
JP (1) JP5869570B2 (es)
KR (1) KR101788794B1 (es)
CN (1) CN103052625B (es)
AR (1) AR082593A1 (es)
AU (1) AU2011288601B2 (es)
BR (1) BR112013004066A2 (es)
CA (2) CA3004565C (es)
CO (1) CO6700822A2 (es)
ES (1) ES2615729T3 (es)
HU (1) HUE031724T2 (es)
IL (1) IL224303A (es)
MX (1) MX342390B (es)
PL (1) PL2603494T3 (es)
PT (1) PT2603494T (es)
TW (1) TWI589563B (es)
WO (1) WO2012019950A1 (es)
ZA (1) ZA201300546B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8871947B2 (en) 2013-02-04 2014-10-28 KingChem LLC Preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid ester
US9139507B2 (en) 2013-12-09 2015-09-22 KingChem LLC. Process for the preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylate and its analogs
DK3645509T3 (da) * 2017-06-27 2021-06-14 Bayer Ag Fremgangsmåde til fremstilling af substituerede 4-aminoindanderivater

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5719201A (en) * 1995-03-30 1998-02-17 Woodbridge Foam Corporation Superabsorbent hydrophilic isocyanate-based foam and process for production thereof
JP2000044541A (ja) * 1998-08-03 2000-02-15 Mitsui Chemicals Inc １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法
JP4568404B2 (ja) 2000-05-17 2010-10-27 三井化学アグロ株式会社 ピラゾールカルボン酸エステル誘導体の製造法
GB0224316D0 (en) 2002-10-18 2002-11-27 Syngenta Participations Ag Chemical compounds
DE10349500A1 (de) * 2003-10-23 2005-06-02 Bayer Cropscience Ag Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern
WO2005123690A1 (de) * 2004-06-18 2005-12-29 Basf Aktiengesellschaft 1-methyl-3-difluormethyl-pyrazol-4-carbonsäure-(ortho-phenyl)-anilide und ihre verwendung als fungizid
JP4971170B2 (ja) * 2004-10-21 2012-07-11 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト ピラゾールの調製のための方法
WO2006090778A1 (ja) * 2005-02-25 2006-08-31 Sagami Chemical Research Center １－置換－３－フルオロアルキルピラゾール－４－カルボン酸エステルの製造方法
PT1940813E (pt) 2005-10-25 2011-01-20 Syngenta Participations Ag Derivados de amidas heterocíclicas úteis como microbicidas
TW200817385A (en) 2006-07-04 2008-04-16 Organon Nv Heterocyclic derivatives
WO2008053044A2 (de) 2006-11-03 2008-05-08 Basf Se Hetarylcarbonsäure-n-(biphen-2-yl)amid-verbindungen
ES2395872T3 (es) * 2007-05-11 2013-02-15 Eli Lilly And Company 2-[4-(Pirazol-4-ilalquil)piperazin-1-il]-3-fenil pirazinas y piridinas y 3-[4-(pirazol-4-ilalquil)piperazin-1-il]-2-fenil piridinas como antagonistas del receptor de 5-HT7
MX2009012602A (es) * 2007-05-31 2009-12-07 Syngenta Participations Ag Proceso para la produccion de pirazoles.
JP2009215194A (ja) * 2008-03-10 2009-09-24 Mitsui Chemicals Agro Inc 含フッ素ピラゾールカルボニトリル誘導体の製造方法、及び該含フッ素ピラゾールカルボニトリル誘導体を利用した含フッ素ピラゾールカルボン酸誘導体の製造方法。
KR101211264B1 (ko) * 2008-03-18 2012-12-18 미쓰이가가쿠 아그로 가부시키가이샤 함불소 아실아세트산 유도체의 제조방법, 함불소 피라졸카르복실산에스테르 유도체의 제조방법 및 함불소 피라졸카르복실산 유도체의 제조방법
JP2009227643A (ja) * 2008-03-25 2009-10-08 Mitsui Chemicals Agro Inc 含フッ素アルキルカルボン酸誘導体を利用した含フッ素ピラゾール誘導体の製造方法
WO2009133178A1 (de) * 2008-05-02 2009-11-05 Basf Se Verfahren zur herstellung von 2-(aminomethyliden)-4,4-difluor-3-oxobuttersäureestern
PT2285779E (pt) 2008-05-08 2013-05-22 Basf Se Processo para a produção de arilcarboxamidas
TW201012803A (en) * 2008-06-06 2010-04-01 Organon Nv Heterocyclic derivatives
GB0812028D0 (en) 2008-07-01 2008-08-06 Syngenta Participations Ag Fungicidal compositions
DK2459538T3 (en) * 2009-07-31 2015-01-05 Syngenta Participations Ag METHODS FOR ALKYLIZING PYRAZOLES

Also Published As

Publication number Publication date
US20160244413A1 (en) 2016-08-25
JP5869570B2 (ja) 2016-02-24
MX2013001520A (es) 2013-02-27
EP2603494A1 (en) 2013-06-19
US20130274481A1 (en) 2013-10-17
AR082593A1 (es) 2012-12-19
CA2806436A1 (en) 2012-02-16
JP2013535493A (ja) 2013-09-12
ZA201300546B (en) 2018-12-19
CN103052625B (zh) 2016-04-13
BR112013004066A2 (pt) 2017-11-14
ES2615729T3 (es) 2017-06-08
TWI589563B (zh) 2017-07-01
CA3004565A1 (en) 2012-02-16
AU2011288601A1 (en) 2013-01-31
KR20130091740A (ko) 2013-08-19
HUE031724T2 (en) 2017-07-28
EP2603494B1 (en) 2016-12-07
CA2806436C (en) 2019-09-10
US9926279B2 (en) 2018-03-27
PT2603494T (pt) 2017-02-03
MX342390B (es) 2016-09-28
PL2603494T3 (pl) 2017-08-31
AU2011288601B2 (en) 2014-08-07
WO2012019950A1 (en) 2012-02-16
US9359304B2 (en) 2016-06-07
TW201211008A (en) 2012-03-16
IL224303A (en) 2017-01-31
US20180208559A1 (en) 2018-07-26
CA3004565C (en) 2020-03-24
CN103052625A (zh) 2013-04-17
KR101788794B1 (ko) 2017-10-20

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