BR112013004066A2 - processo para a preparação de 3-haloalquilapirazóis. - Google Patents

processo para a preparação de 3-haloalquilapirazóis.

Info

Publication number
BR112013004066A2
BR112013004066A2 BR112013004066A BR112013004066A BR112013004066A2 BR 112013004066 A2 BR112013004066 A2 BR 112013004066A2 BR 112013004066 A BR112013004066 A BR 112013004066A BR 112013004066 A BR112013004066 A BR 112013004066A BR 112013004066 A2 BR112013004066 A2 BR 112013004066A2
Authority
BR
Brazil
Prior art keywords
preparation
haloalkylpyrazoles
compound
formula
optionally substituted
Prior art date
Application number
BR112013004066A
Other languages
English (en)
Inventor
Wang Linhua
Bharat Sheth Ritesh
Original Assignee
Syngenta Particpations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Particpations Ag filed Critical Syngenta Particpations Ag
Publication of BR112013004066A2 publication Critical patent/BR112013004066A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

processo para a preparação de 3-haloalquilapirazóis. a presente invenção provê um processo para a preparação de um composto de fórmula i: caracterizado pelo fato de r¹ ser c<sym> - c<sym> haloalquila; r² ser alquila opcionalmente substituída, arila opcionalmente substituída ou heteroarila opcionalmente substituída; e r³ ser metila ou etila; compreendendo a reação de um composto de fórmula iv: em que r,r² e r³ são como definido para composto de formula i; com um agente alquilante na presença de um amido.
BR112013004066A 2010-08-10 2011-08-03 processo para a preparação de 3-haloalquilapirazóis. BR112013004066A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US37212210P 2010-08-10 2010-08-10
PCT/EP2011/063360 WO2012019950A1 (en) 2010-08-10 2011-08-03 Process for the preparation of 3-haloalkylpyrazoles

Publications (1)

Publication Number Publication Date
BR112013004066A2 true BR112013004066A2 (pt) 2017-11-14

Family

ID=44503820

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112013004066A BR112013004066A2 (pt) 2010-08-10 2011-08-03 processo para a preparação de 3-haloalquilapirazóis.

Country Status (19)

Country Link
US (3) US9359304B2 (pt)
EP (1) EP2603494B1 (pt)
JP (1) JP5869570B2 (pt)
KR (1) KR101788794B1 (pt)
CN (1) CN103052625B (pt)
AR (1) AR082593A1 (pt)
AU (1) AU2011288601B2 (pt)
BR (1) BR112013004066A2 (pt)
CA (2) CA2806436C (pt)
CO (1) CO6700822A2 (pt)
ES (1) ES2615729T3 (pt)
HU (1) HUE031724T2 (pt)
IL (1) IL224303A (pt)
MX (1) MX342390B (pt)
PL (1) PL2603494T3 (pt)
PT (1) PT2603494T (pt)
TW (1) TWI589563B (pt)
WO (1) WO2012019950A1 (pt)
ZA (1) ZA201300546B (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8871947B2 (en) 2013-02-04 2014-10-28 KingChem LLC Preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid ester
US9139507B2 (en) 2013-12-09 2015-09-22 KingChem LLC. Process for the preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylate and its analogs
WO2019002042A1 (en) * 2017-06-27 2019-01-03 Bayer Aktiengesellschaft PROCESS FOR THE PREPARATION OF SUBSTITUTED 4-AMINOINDANE DERIVATIVES

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5719201A (en) * 1995-03-30 1998-02-17 Woodbridge Foam Corporation Superabsorbent hydrophilic isocyanate-based foam and process for production thereof
JP2000044541A (ja) 1998-08-03 2000-02-15 Mitsui Chemicals Inc １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法
JP4568404B2 (ja) 2000-05-17 2010-10-27 三井化学アグロ株式会社 ピラゾールカルボン酸エステル誘導体の製造法
GB0224316D0 (en) 2002-10-18 2002-11-27 Syngenta Participations Ag Chemical compounds
DE10349500A1 (de) * 2003-10-23 2005-06-02 Bayer Cropscience Ag Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern
EP1761498A1 (de) * 2004-06-18 2007-03-14 Basf Aktiengesellschaft 1-methyl-3-difluormethyl-pyrazol-4-carbonsäure-(ortho-phenyl)-anilide und ihre verwendung als fungizid
JP4971170B2 (ja) * 2004-10-21 2012-07-11 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト ピラゾールの調製のための方法
EP1854788B8 (en) * 2005-02-25 2012-12-26 Sagami Chemical Research Institute Method for producing 1-substituted-3-fluoroalkyl pyrazole-4-carboxylate
PL1940813T3 (pl) 2005-10-25 2011-04-29 Syngenta Participations Ag Pochodne amidowe heterocykli użyteczne jako środki mikrobiobójcze
TW200817385A (en) * 2006-07-04 2008-04-16 Organon Nv Heterocyclic derivatives
WO2008053044A2 (de) 2006-11-03 2008-05-08 Basf Se Hetarylcarbonsäure-n-(biphen-2-yl)amid-verbindungen
MX2009012126A (es) * 2007-05-11 2009-11-23 Lilly Co Eli 2-[4-(pirazol-4-ilalquil)piperazin-1-il]-3-fenil-pirazinas y piridinas y 3-[4-(pirazol-4-ilalquil)piperazin-1-il]-2-fenil piridinas como antagonistas del receptor 5-ht7.
KR20100017431A (ko) 2007-05-31 2010-02-16 신젠타 파티서페이션즈 아게 피라졸의 제조 방법
JP2009215194A (ja) * 2008-03-10 2009-09-24 Mitsui Chemicals Agro Inc 含フッ素ピラゾールカルボニトリル誘導体の製造方法、及び該含フッ素ピラゾールカルボニトリル誘導体を利用した含フッ素ピラゾールカルボン酸誘導体の製造方法。
US8344156B2 (en) * 2008-03-18 2013-01-01 Mitsui Chemicals Agro, Inc. Method for producing fluorine-containing acylacetic acid derivative, method for producing fluorine-containing pyrazolecarboxylic acid ester derivative, and method for producing fluorine-containing pyrazolecarboxylic acid derivative
JP2009227643A (ja) * 2008-03-25 2009-10-08 Mitsui Chemicals Agro Inc 含フッ素アルキルカルボン酸誘導体を利用した含フッ素ピラゾール誘導体の製造方法
PL2300417T3 (pl) * 2008-05-02 2015-12-31 Basf Se Sposób wytwarzania estrów kwasu 2-(aminometylideno)-4,4-difluoro-3-oksomasłowego
AU2009245791B2 (en) 2008-05-08 2013-05-16 Basf Se Method for manufacturing aryl carboxamides
TW201012803A (en) 2008-06-06 2010-04-01 Organon Nv Heterocyclic derivatives
GB0812028D0 (en) 2008-07-01 2008-08-06 Syngenta Participations Ag Fungicidal compositions
MX2012001067A (es) * 2009-07-31 2012-03-16 Syngenta Participations Ag Procesos para la alquilacion de pirazoles.

Also Published As

Publication number Publication date
CN103052625A (zh) 2013-04-17
KR101788794B1 (ko) 2017-10-20
US9359304B2 (en) 2016-06-07
CA2806436A1 (en) 2012-02-16
PL2603494T3 (pl) 2017-08-31
MX342390B (es) 2016-09-28
AU2011288601A1 (en) 2013-01-31
ZA201300546B (en) 2018-12-19
US9926279B2 (en) 2018-03-27
TWI589563B (zh) 2017-07-01
EP2603494A1 (en) 2013-06-19
PT2603494T (pt) 2017-02-03
AU2011288601B2 (en) 2014-08-07
TW201211008A (en) 2012-03-16
CA3004565A1 (en) 2012-02-16
HUE031724T2 (en) 2017-07-28
AR082593A1 (es) 2012-12-19
KR20130091740A (ko) 2013-08-19
IL224303A (en) 2017-01-31
ES2615729T3 (es) 2017-06-08
MX2013001520A (es) 2013-02-27
CA3004565C (en) 2020-03-24
WO2012019950A1 (en) 2012-02-16
CO6700822A2 (es) 2013-06-28
JP2013535493A (ja) 2013-09-12
US20130274481A1 (en) 2013-10-17
US20160244413A1 (en) 2016-08-25
CN103052625B (zh) 2016-04-13
US20180208559A1 (en) 2018-07-26
JP5869570B2 (ja) 2016-02-24
EP2603494B1 (en) 2016-12-07
CA2806436C (en) 2019-09-10

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B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07A Technical examination (opinion): publication of technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B12B Appeal: appeal against refusal
B350 Update of information on the portal [chapter 15.35 patent gazette]