BR112015021151A2 - processo para a preparação de (2s,5r)-ácido sulfúrico mono-{[(4-aminopiperidin-4-il)carbonil]-7-oxo-1,6-diazabiciclo[3.2.1]-oct-6-il} éster - Google Patents

processo para a preparação de (2s,5r)-ácido sulfúrico mono-{[(4-aminopiperidin-4-il)carbonil]-7-oxo-1,6-diazabiciclo[3.2.1]-oct-6-il} éster

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Publication number
BR112015021151A2
BR112015021151A2 BR112015021151A BR112015021151A BR112015021151A2 BR 112015021151 A2 BR112015021151 A2 BR 112015021151A2 BR 112015021151 A BR112015021151 A BR 112015021151A BR 112015021151 A BR112015021151 A BR 112015021151A BR 112015021151 A2 BR112015021151 A2 BR 112015021151A2
Authority
BR
Brazil
Prior art keywords
aminopiperidin
diazabicyclo
oxo
carbonyl
oct
Prior art date
Application number
BR112015021151A
Other languages
English (en)
Inventor
Suresh Wankhede Karuna
Manikrao Surwase Mahesh
Vithalbhai Patel Mahesh
Keshav Deshpande Prasad
Dattatraya Yeole Ravindra
Bhawsar Satish
Original Assignee
Wockhardt Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wockhardt Ltd filed Critical Wockhardt Ltd
Publication of BR112015021151A2 publication Critical patent/BR112015021151A2/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

resumo patente de invenção: "processo para a preparação de (2s,5r)-ácido sulfúrico mono-{[(4-aminopiperidin-4-il)carbonil]-7-oxo-1,6-diazabiciclo[3.2.1]-oct-6-il} éster" a presente invenção refere-se a um processo para a preparação de (2s,5r)-ácido sulfúrico mono-{[(4-aminopiperidin-4-il)carbonil]-7-oxo-1,6-diazabiciclo[3.2.1]-oct-6-il} éster, processo este que compreende reagir um composto de fórmula (ii) com um composto de fórmula (iii) para obter um composto de fórmula (iv).
BR112015021151A 2013-03-08 2013-10-12 processo para a preparação de (2s,5r)-ácido sulfúrico mono-{[(4-aminopiperidin-4-il)carbonil]-7-oxo-1,6-diazabiciclo[3.2.1]-oct-6-il} éster BR112015021151A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN716MU2013 2013-03-08
PCT/IB2013/059329 WO2015033191A1 (en) 2013-03-08 2013-10-12 A process for preparation of (2s, 5r)- sulfuric acid mono-{[(4-aminopiperidin-4-yl) carbonyl]-7-oxo-1,6-diaza-bicyclo[3.2.1]-oct-6-yl} ester

Publications (1)

Publication Number Publication Date
BR112015021151A2 true BR112015021151A2 (pt) 2017-07-18

Family

ID=54250568

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015021151A BR112015021151A2 (pt) 2013-03-08 2013-10-12 processo para a preparação de (2s,5r)-ácido sulfúrico mono-{[(4-aminopiperidin-4-il)carbonil]-7-oxo-1,6-diazabiciclo[3.2.1]-oct-6-il} éster

Country Status (11)

Country Link
US (1) US9556174B2 (pt)
JP (1) JP6182621B2 (pt)
KR (1) KR101780577B1 (pt)
CN (1) CN105143224A (pt)
AU (1) AU2013399862B2 (pt)
BR (1) BR112015021151A2 (pt)
CA (1) CA2904084C (pt)
MX (1) MX2015011720A (pt)
NZ (1) NZ711329A (pt)
RU (1) RU2621051C2 (pt)
WO (1) WO2015033191A1 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014135930A1 (en) * 2013-03-08 2014-09-12 Wockhardt Limited A process for sodium salt of (2s, 5r)-2-carboxamido-7-oxo-6-sulfooxy -1,6-diaza-bicyclo[3.2.1]octane
CN111072660B (zh) * 2018-10-22 2021-05-18 新发药业有限公司 一种瑞来巴坦的简便制备方法
CN111943950B (zh) * 2020-09-10 2022-03-29 山东安信制药有限公司 一种瑞来巴坦的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2124014C1 (ru) * 1993-12-29 1998-12-27 Пфайзер Инк. Диазабициклические соединения и содержащая их фармацевтическая композиция
CN101687357B (zh) * 2007-06-27 2014-01-15 积水化学工业株式会社 安全玻璃用多层中间膜的制造装置及制造方法
ES2533826T3 (es) * 2008-01-18 2015-04-15 Merck Sharp & Dohme Corp. Inhibidores de beta-lactamasa
US20120053350A1 (en) * 2009-04-30 2012-03-01 Ian Mangion Preparation of alkyl esters of n-protected oxo-azacycloalkylcarboxylic acids
CA2822758C (en) * 2010-12-22 2018-03-20 Meiji Seika Pharma Co., Ltd. Optically active diazabicyclooctane derivative and process for preparing the same
BR112014003476A2 (pt) * 2011-09-13 2017-03-01 Wockhardt Ltd compostos contendo nitrogênio e seu uso
WO2014135932A1 (en) * 2013-03-08 2014-09-12 Wockhardt Limited A process for preparation of (2s, 5r)-7-oxo-6-sulphooxy-2-[((3r)-pyrrolidine-3-carbonyl)-hydrazino carbonyl]-1,6-diaza-bicyclo[3.2.1]octane
WO2014135930A1 (en) * 2013-03-08 2014-09-12 Wockhardt Limited A process for sodium salt of (2s, 5r)-2-carboxamido-7-oxo-6-sulfooxy -1,6-diaza-bicyclo[3.2.1]octane
US9862718B2 (en) * 2013-03-08 2018-01-09 Wockhardt Limited Sodium salt of (2S, 5R)-6-benzyloxy-7-oxo-1,6-diaza-bicyclo [3.2.1] octane-2-carboxylic acid and its preparation
JP6285969B2 (ja) * 2013-03-08 2018-02-28 ウォックハート リミテッド （２ｓ，５ｒ）−７−オキソ−６−スルホオキシ−２−［（（３ｒ）−ピペリジン−３−カルボニル）−ヒドラジノカルボニル］−１，６−ジアザ−ビシクロ［３．２．１］オクタンの調製のためのプロセス

Also Published As

Publication number Publication date
JP6182621B2 (ja) 2017-08-16
US9556174B2 (en) 2017-01-31
RU2015142581A (ru) 2017-04-20
KR20150125998A (ko) 2015-11-10
WO2015033191A1 (en) 2015-03-12
NZ711329A (en) 2016-06-24
CA2904084A1 (en) 2015-03-12
AU2013399862A1 (en) 2015-09-10
RU2621051C2 (ru) 2017-05-31
CN105143224A (zh) 2015-12-09
AU2013399862B2 (en) 2016-07-14
US20160002233A1 (en) 2016-01-07
MX2015011720A (es) 2015-12-01
CA2904084C (en) 2017-03-28
KR101780577B1 (ko) 2017-09-21
JP2016510063A (ja) 2016-04-04

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06I Publication of requirement cancelled [chapter 6.9 patent gazette]

Free format text: ANULADA A PUBLICACAO CODIGO 6.6.1 NA RPI NO 2462 DE 13/03/2018 POR TER SIDO INDEVIDA.

B06T Formal requirements before examination [chapter 6.20 patent gazette]
B11E Dismissal acc. art. 34 of ipl - requirements for examination incomplete
B11T Dismissal of application maintained [chapter 11.20 patent gazette]