MX2015011720A - Proceso para la preparcion de monoacido de (2s,5r)-{[(4-aminopiper idin-4-il)carbonil]-7-oxo-1,6-diaza-biciclo[3.2.1 oct-6-il} ester sulfurico. - Google Patents

Proceso para la preparcion de monoacido de (2s,5r)-{[(4-aminopiper idin-4-il)carbonil]-7-oxo-1,6-diaza-biciclo[3.2.1 oct-6-il} ester sulfurico.

Info

Publication number
MX2015011720A
MX2015011720A MX2015011720A MX2015011720A MX2015011720A MX 2015011720 A MX2015011720 A MX 2015011720A MX 2015011720 A MX2015011720 A MX 2015011720A MX 2015011720 A MX2015011720 A MX 2015011720A MX 2015011720 A MX2015011720 A MX 2015011720A
Authority
MX
Mexico
Prior art keywords
aminopiperidin
diaza
bicyclo
oxo
carbonyl
Prior art date
Application number
MX2015011720A
Other languages
English (en)
Inventor
Mahesh Vithalbhai Patel
Prasad Keshav Deshpande
Karuna Suresh Wankhede
Mahesh Manikrao Surwase
Satish Bhawsar
Ravindra Dattatraya Yeole
Original Assignee
Wockhardt Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wockhardt Ltd filed Critical Wockhardt Ltd
Publication of MX2015011720A publication Critical patent/MX2015011720A/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems

Abstract

Se describe un procedimiento para la preparación de monoácido de (2S, 5R) -{[(4-aminopiperidin-4-il)carbonil] -7-oxo-1,6-diaza-bici clo [3.2.1] -Oct-6-il} éster sulfúrico.
MX2015011720A 2013-03-08 2013-10-12 Proceso para la preparcion de monoacido de (2s,5r)-{[(4-aminopiper idin-4-il)carbonil]-7-oxo-1,6-diaza-biciclo[3.2.1 oct-6-il} ester sulfurico. MX2015011720A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN716MU2013 2013-03-08
PCT/IB2013/059329 WO2015033191A1 (en) 2013-03-08 2013-10-12 A process for preparation of (2s, 5r)- sulfuric acid mono-{[(4-aminopiperidin-4-yl) carbonyl]-7-oxo-1,6-diaza-bicyclo[3.2.1]-oct-6-yl} ester

Publications (1)

Publication Number Publication Date
MX2015011720A true MX2015011720A (es) 2015-12-01

Family

ID=54250568

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015011720A MX2015011720A (es) 2013-03-08 2013-10-12 Proceso para la preparcion de monoacido de (2s,5r)-{[(4-aminopiper idin-4-il)carbonil]-7-oxo-1,6-diaza-biciclo[3.2.1 oct-6-il} ester sulfurico.

Country Status (11)

Country Link
US (1) US9556174B2 (es)
JP (1) JP6182621B2 (es)
KR (1) KR101780577B1 (es)
CN (1) CN105143224A (es)
AU (1) AU2013399862B2 (es)
BR (1) BR112015021151A2 (es)
CA (1) CA2904084C (es)
MX (1) MX2015011720A (es)
NZ (1) NZ711329A (es)
RU (1) RU2621051C2 (es)
WO (1) WO2015033191A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2015011723A (es) * 2013-03-08 2016-06-06 Wockhardt Ltd Proceso para la preparacion de una sal de sodio de (2s, 5r) -2-carboxamido-7-oxo-6-sulfooxi-1,6-diaza-biciclo[3.2.1]-octano.
CN111072660B (zh) * 2018-10-22 2021-05-18 新发药业有限公司 一种瑞来巴坦的简便制备方法
CN111943950B (zh) * 2020-09-10 2022-03-29 山东安信制药有限公司 一种瑞来巴坦的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69416869T2 (de) * 1993-12-29 1999-07-01 Pfizer Diazabicyclische neurokinin antagonisten
US8152507B2 (en) * 2007-06-27 2012-04-10 Sekisui Chemical Co., Ltd. Apparatus and method for manufacturing multiplex interlayer for safety glass
KR101800610B1 (ko) * 2008-01-18 2017-11-23 머크 샤프 앤드 돔 코포레이션 베타­락타마제 억제제
WO2010126820A2 (en) * 2009-04-30 2010-11-04 Merck Sharp & Dohme Corp. Preparation of alkyl esters of n-protected oxo-azacycloalkylcarboxylic acids
SG191320A1 (en) * 2010-12-22 2013-07-31 Meiji Seika Pharma Co Ltd Optically-active diazabicyclooctane derivative and method for manufacturing same
BR112014003476A2 (pt) * 2011-09-13 2017-03-01 Wockhardt Ltd compostos contendo nitrogênio e seu uso
BR112015021186A2 (pt) * 2013-03-08 2017-07-18 Wockhardt Ltd processo para a preparação de (2s,5r)-7-oxo-6-sulfóxi-2-[((3r)-pirrolidina-3-carbonil)-hidrazino carbonil]-1,6-diaza-biciclo[3.2.1]octano
BR112015021332B1 (pt) * 2013-03-08 2020-06-30 Wockhardt Limited sal de sódio de ácido (2s, 5r)-6-benzilóxi-7-oxo-1,6-diaza-biciclo [3.2.1] octano-2-carboxílico e sua preparação
MX2015011723A (es) * 2013-03-08 2016-06-06 Wockhardt Ltd Proceso para la preparacion de una sal de sodio de (2s, 5r) -2-carboxamido-7-oxo-6-sulfooxi-1,6-diaza-biciclo[3.2.1]-octano.
NZ711327A (en) * 2013-03-08 2016-06-24 Wockhardt Ltd A process for preparation of (2s, 5r)-7-oxo-6-sulphooxy-2-[((3r)-piperidine-3-carbonyl)-hydrazino carbonyl]-1,6-diaza-bicyclo [3.2.1]- octane

Also Published As

Publication number Publication date
RU2015142581A (ru) 2017-04-20
WO2015033191A1 (en) 2015-03-12
CN105143224A (zh) 2015-12-09
RU2621051C2 (ru) 2017-05-31
JP6182621B2 (ja) 2017-08-16
US20160002233A1 (en) 2016-01-07
JP2016510063A (ja) 2016-04-04
NZ711329A (en) 2016-06-24
CA2904084C (en) 2017-03-28
KR101780577B1 (ko) 2017-09-21
CA2904084A1 (en) 2015-03-12
US9556174B2 (en) 2017-01-31
KR20150125998A (ko) 2015-11-10
AU2013399862A1 (en) 2015-09-10
BR112015021151A2 (pt) 2017-07-18
AU2013399862B2 (en) 2016-07-14

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