MX2015011723A - Proceso para la preparacion de una sal de sodio de (2s, 5r) -2-carboxamido-7-oxo-6-sulfooxi-1,6-diaza-biciclo[3.2.1]-octano. - Google Patents
Proceso para la preparacion de una sal de sodio de (2s, 5r) -2-carboxamido-7-oxo-6-sulfooxi-1,6-diaza-biciclo[3.2.1]-octano.Info
- Publication number
- MX2015011723A MX2015011723A MX2015011723A MX2015011723A MX2015011723A MX 2015011723 A MX2015011723 A MX 2015011723A MX 2015011723 A MX2015011723 A MX 2015011723A MX 2015011723 A MX2015011723 A MX 2015011723A MX 2015011723 A MX2015011723 A MX 2015011723A
- Authority
- MX
- Mexico
- Prior art keywords
- carboxamido
- diaza
- bicyclo
- octane
- oxo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Se describe un proceso para la preparación de una sal de sodio de (2S, 5R)-2-carboxamido-7-oxo-6-sulfooxi-1,6-diaza-biciclo [3.2. 1] octano.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN718MU2013 | 2013-03-08 | ||
PCT/IB2013/059325 WO2014135930A1 (en) | 2013-03-08 | 2013-10-12 | A process for sodium salt of (2s, 5r)-2-carboxamido-7-oxo-6-sulfooxy -1,6-diaza-bicyclo[3.2.1]octane |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2015011723A true MX2015011723A (es) | 2016-06-06 |
Family
ID=54250569
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2015011723A MX2015011723A (es) | 2013-03-08 | 2013-10-12 | Proceso para la preparacion de una sal de sodio de (2s, 5r) -2-carboxamido-7-oxo-6-sulfooxi-1,6-diaza-biciclo[3.2.1]-octano. |
Country Status (12)
Country | Link |
---|---|
US (1) | US9567335B2 (es) |
EP (1) | EP3013829A1 (es) |
JP (1) | JP6253676B2 (es) |
KR (1) | KR101763056B1 (es) |
CN (1) | CN105143226A (es) |
AU (1) | AU2013380573B2 (es) |
BR (1) | BR112015021240A2 (es) |
CA (1) | CA2904089C (es) |
MX (1) | MX2015011723A (es) |
NZ (1) | NZ711326A (es) |
RU (1) | RU2632192C2 (es) |
WO (1) | WO2014135930A1 (es) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP6182621B2 (ja) * | 2013-03-08 | 2017-08-16 | ウォックハート リミテッド | (2s,5r)−硫酸モノ−{[(4−アミノピペリジン−4−イル)カルボニル]−7−オキソ−1,6−ジアザ−ビシクロ[3.2.1]オクタ−6−イル}エステルを調製するための方法 |
CN105980385B (zh) * | 2014-02-03 | 2018-01-09 | 沃克哈特有限公司 | 制备(2s,5r)‑1,6‑二氮杂‑二环[3.2.1]辛烷‑2‑腈‑7‑氧代‑6‑(磺氧基)‑单钠盐的方法 |
WO2016120752A1 (en) * | 2015-01-28 | 2016-08-04 | Wockhardt Limited | A process for preparation of (2s, 5r)-n-(2-amino ethoxy)-6-(sulfooxy)-7-oxo-1,6- diazabicyclo [3.2.1] octane-2-carboxamide |
WO2016157057A1 (en) * | 2015-03-27 | 2016-10-06 | Wockhardt Limited | A process for preparation of sodium salt of (2s, 5r) sulfuric acid mono-(2-[1,3,4]oxadiazol-2-yl-7-oxo-1,6-diazabicyclo[3.2.1 ]oct-6-yl)ester |
EP3334734B1 (en) * | 2015-08-10 | 2020-01-01 | Sandoz AG | Form c of avibactam sodium |
CN105061425B (zh) * | 2015-08-13 | 2017-01-11 | 广州楷模生物科技有限公司 | 二氮杂双环辛酮硫酸单酯的合成方法 |
CN107325096B (zh) * | 2016-04-29 | 2020-11-03 | 正大天晴药业集团股份有限公司 | 一种阿维巴坦单钠盐的结晶 |
KR102482826B1 (ko) | 2016-08-26 | 2022-12-28 | 산도즈 아게 | 아비박탐 유리 산 |
CN107880042A (zh) * | 2016-09-30 | 2018-04-06 | 上海复星星泰医药科技有限公司 | 阿维巴坦钠及其中间体化合物的制备方法 |
CN106866668B (zh) * | 2017-01-23 | 2019-01-11 | 齐鲁天和惠世制药有限公司 | 一锅法制备阿维巴坦钠的方法 |
US10434089B2 (en) | 2017-01-25 | 2019-10-08 | The Johns Hopkins University | Avibactam and carbapenems antibacterial agents |
CN110267956B (zh) * | 2017-02-08 | 2022-07-15 | 桑多斯股份公司 | 用于制备阿维巴坦钠结晶形式c的方法 |
CN109678855B (zh) * | 2017-10-18 | 2020-07-17 | 新发药业有限公司 | 一种阿维巴坦中间体的制备方法 |
CN109678856B (zh) * | 2017-10-18 | 2020-09-25 | 新发药业有限公司 | 一种阿维巴坦中间体的制备方法 |
CN107827886B (zh) * | 2017-11-23 | 2020-06-23 | 中山奕安泰医药科技有限公司 | 一种高纯度阿维巴坦的精制制备工艺 |
CN109956941B (zh) * | 2017-12-25 | 2020-08-04 | 新发药业有限公司 | 一种阿维巴坦的简便制备方法 |
CN107936017A (zh) * | 2018-01-12 | 2018-04-20 | 上海龙翔生物医药开发有限公司 | 一种通过结晶制备晶型a或晶型d阿维巴坦产品的方法 |
CN113387950A (zh) * | 2020-03-11 | 2021-09-14 | 天津科伦药物研究有限公司 | 一种阿维巴坦钠中间体的精制方法 |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2812635B1 (fr) * | 2000-08-01 | 2002-10-11 | Aventis Pharma Sa | Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens |
BR0208956A (pt) * | 2001-04-16 | 2004-07-13 | Tanabe Seiyaku Co | Abridor de canais de k ativados por cálcio de grande condutância |
JP2008536817A (ja) * | 2005-03-24 | 2008-09-11 | グラクソ グループ リミテッド | 胃腸疾患の処置用医薬として有用なイミダゾ(1,2−a)ピリジン誘導体 |
ES2533826T3 (es) * | 2008-01-18 | 2015-04-15 | Merck Sharp & Dohme Corp. | Inhibidores de beta-lactamasa |
WO2010014939A1 (en) * | 2008-07-31 | 2010-02-04 | Genentech, Inc. | Pyrimidine compounds, compositions and methods of use |
FR2951171A1 (fr) * | 2009-10-09 | 2011-04-15 | Novexel | Nouveau sel de sodium d'un compose azabicyclique sous forme enantiomere cristallisee et nouvelles formes polymorphes et pseudopolymorphes ainsi que leur preparation |
US8772490B2 (en) * | 2010-12-22 | 2014-07-08 | Meiji Seika Pharma Co., Ltd. | Optically active diazabicyclooctane derivatives and process for preparing the same |
CA2822758C (en) * | 2010-12-22 | 2018-03-20 | Meiji Seika Pharma Co., Ltd. | Optically active diazabicyclooctane derivative and process for preparing the same |
BR112013032415B1 (pt) * | 2011-06-17 | 2021-07-27 | Pfizer Anti-Infectives Ab | Processos para preparar compostos e compostos |
US8969567B2 (en) * | 2011-09-13 | 2015-03-03 | Wockhardt Ltd. | Nitrogen containing compounds and their use |
BR112014003476A2 (pt) * | 2011-09-13 | 2017-03-01 | Wockhardt Ltd | compostos contendo nitrogênio e seu uso |
US9862718B2 (en) * | 2013-03-08 | 2018-01-09 | Wockhardt Limited | Sodium salt of (2S, 5R)-6-benzyloxy-7-oxo-1,6-diaza-bicyclo [3.2.1] octane-2-carboxylic acid and its preparation |
JP6182621B2 (ja) * | 2013-03-08 | 2017-08-16 | ウォックハート リミテッド | (2s,5r)−硫酸モノ−{[(4−アミノピペリジン−4−イル)カルボニル]−7−オキソ−1,6−ジアザ−ビシクロ[3.2.1]オクタ−6−イル}エステルを調製するための方法 |
JP6285969B2 (ja) * | 2013-03-08 | 2018-02-28 | ウォックハート リミテッド | (2s,5r)−7−オキソ−6−スルホオキシ−2−[((3r)−ピペリジン−3−カルボニル)−ヒドラジノカルボニル]−1,6−ジアザ−ビシクロ[3.2.1]オクタンの調製のためのプロセス |
WO2014135932A1 (en) * | 2013-03-08 | 2014-09-12 | Wockhardt Limited | A process for preparation of (2s, 5r)-7-oxo-6-sulphooxy-2-[((3r)-pyrrolidine-3-carbonyl)-hydrazino carbonyl]-1,6-diaza-bicyclo[3.2.1]octane |
-
2013
- 2013-10-12 WO PCT/IB2013/059325 patent/WO2014135930A1/en active Application Filing
- 2013-10-12 AU AU2013380573A patent/AU2013380573B2/en not_active Ceased
- 2013-10-12 JP JP2015560790A patent/JP6253676B2/ja not_active Expired - Fee Related
- 2013-10-12 CN CN201380074164.2A patent/CN105143226A/zh active Pending
- 2013-10-12 KR KR1020157026986A patent/KR101763056B1/ko active IP Right Grant
- 2013-10-12 MX MX2015011723A patent/MX2015011723A/es unknown
- 2013-10-12 US US14/770,231 patent/US9567335B2/en not_active Expired - Fee Related
- 2013-10-12 NZ NZ711326A patent/NZ711326A/en not_active IP Right Cessation
- 2013-10-12 CA CA2904089A patent/CA2904089C/en not_active Expired - Fee Related
- 2013-10-12 BR BR112015021240A patent/BR112015021240A2/pt not_active Application Discontinuation
- 2013-10-12 RU RU2015142826A patent/RU2632192C2/ru not_active IP Right Cessation
- 2013-10-12 EP EP13812117.3A patent/EP3013829A1/en not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
AU2013380573A1 (en) | 2015-09-10 |
BR112015021240A2 (pt) | 2017-07-18 |
JP6253676B2 (ja) | 2017-12-27 |
CA2904089C (en) | 2017-05-02 |
KR101763056B1 (ko) | 2017-07-28 |
EP3013829A1 (en) | 2016-05-04 |
JP2016510062A (ja) | 2016-04-04 |
CN105143226A (zh) | 2015-12-09 |
US20160016955A1 (en) | 2016-01-21 |
US9567335B2 (en) | 2017-02-14 |
NZ711326A (en) | 2016-06-24 |
AU2013380573A8 (en) | 2016-07-07 |
CA2904089A1 (en) | 2014-09-12 |
RU2632192C2 (ru) | 2017-10-03 |
AU2013380573B2 (en) | 2016-07-07 |
WO2014135930A1 (en) | 2014-09-12 |
RU2015142826A (ru) | 2017-04-13 |
KR20150122238A (ko) | 2015-10-30 |
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