CO5251420A1 - Compuestos mimeticos de peptidos de giros beta, bibliotecas de tales compuestos, y proceso para la fabricacion de los mismos - Google Patents

Compuestos mimeticos de peptidos de giros beta, bibliotecas de tales compuestos, y proceso para la fabricacion de los mismos

Info

Publication number
CO5251420A1
CO5251420A1 CO00097142A CO00097142A CO5251420A1 CO 5251420 A1 CO5251420 A1 CO 5251420A1 CO 00097142 A CO00097142 A CO 00097142A CO 00097142 A CO00097142 A CO 00097142A CO 5251420 A1 CO5251420 A1 CO 5251420A1
Authority
CO
Colombia
Prior art keywords
compounds
manufacture
aryl
libraries
geta
Prior art date
Application number
CO00097142A
Other languages
English (en)
Spanish (es)
Inventor
Adam Golebiowski
Sean Rees Klopfenstein
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of CO5251420A1 publication Critical patent/CO5251420A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/047Simultaneous synthesis of different peptide species; Peptide libraries
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0215Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing natural amino acids, forming a peptide bond via their side chain functional group, e.g. epsilon-Lys, gamma-Glu

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Health & Medical Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Indole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CO00097142A 1999-12-21 2000-12-21 Compuestos mimeticos de peptidos de giros beta, bibliotecas de tales compuestos, y proceso para la fabricacion de los mismos CO5251420A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17282399P 1999-12-21 1999-12-21

Publications (1)

Publication Number Publication Date
CO5251420A1 true CO5251420A1 (es) 2003-02-28

Family

ID=22629385

Family Applications (1)

Application Number Title Priority Date Filing Date
CO00097142A CO5251420A1 (es) 1999-12-21 2000-12-21 Compuestos mimeticos de peptidos de giros beta, bibliotecas de tales compuestos, y proceso para la fabricacion de los mismos

Country Status (16)

Country Link
EP (1) EP1240169A1 (hu)
JP (1) JP2003518124A (hu)
KR (1) KR20020062352A (hu)
CN (1) CN1413214A (hu)
AU (1) AU2286401A (hu)
BR (1) BR0016518A (hu)
CA (1) CA2393759A1 (hu)
CO (1) CO5251420A1 (hu)
CZ (1) CZ20022110A3 (hu)
HU (1) HUP0300100A2 (hu)
IL (1) IL149834A0 (hu)
MX (1) MXPA02006330A (hu)
NO (1) NO20022953D0 (hu)
PE (1) PE20010955A1 (hu)
PL (1) PL355971A1 (hu)
WO (1) WO2001046197A1 (hu)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20220064171A1 (en) * 2018-12-27 2022-03-03 Holosmedic Novel compound and pharmaceutical composition comprising same for enhancing anticancer activity
WO2020139044A1 (ko) * 2018-12-27 2020-07-02 홀로스메딕 주식회사 신규한 화합물 및 이를 포함하는 항암 활성 증진용 약학 조성물
CA3159791A1 (en) * 2019-10-31 2021-05-06 Holosmedic Hexahydro-2h-pyrazino[1,2-a]pyrazine-6,9-dione derivatives and pharmaceutical compositions for prevention or treatment of cancer comprising same

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5929237A (en) * 1995-10-27 1999-07-27 Molecumetics Ltd. Reverse-turn mimetics and methods relating thereto
US6013458A (en) * 1995-10-27 2000-01-11 Molecumetics, Ltd. Reverse-turn mimetics and methods relating thereto

Also Published As

Publication number Publication date
MXPA02006330A (es) 2002-12-13
EP1240169A1 (en) 2002-09-18
IL149834A0 (en) 2002-11-10
AU2286401A (en) 2001-07-03
WO2001046197A1 (en) 2001-06-28
JP2003518124A (ja) 2003-06-03
BR0016518A (pt) 2002-09-24
NO20022953L (no) 2002-06-19
PL355971A1 (en) 2004-05-31
CA2393759A1 (en) 2001-06-28
PE20010955A1 (es) 2001-10-11
HUP0300100A2 (en) 2003-05-28
CN1413214A (zh) 2003-04-23
NO20022953D0 (no) 2002-06-19
KR20020062352A (ko) 2002-07-25
CZ20022110A3 (cs) 2002-11-13

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Legal Events

Date Code Title Description
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