CO5090902A1 - Pirroles sustituidos - Google Patents

Pirroles sustituidos

Info

Publication number
CO5090902A1
CO5090902A1 CO00096628A CO00096628A CO5090902A1 CO 5090902 A1 CO5090902 A1 CO 5090902A1 CO 00096628 A CO00096628 A CO 00096628A CO 00096628 A CO00096628 A CO 00096628A CO 5090902 A1 CO5090902 A1 CO 5090902A1
Authority
CO
Colombia
Prior art keywords
heteroaryl
pirroles
replaced
heterocycle
alkyl
Prior art date
Application number
CO00096628A
Other languages
English (en)
Spanish (es)
Inventor
Fotouchi Nader
Kong Norman
Allen John Lovey
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CO5090902A1 publication Critical patent/CO5090902A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
CO00096628A 1999-12-22 2000-12-20 Pirroles sustituidos CO5090902A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17155799P 1999-12-22 1999-12-22

Publications (1)

Publication Number Publication Date
CO5090902A1 true CO5090902A1 (es) 2001-10-30

Family

ID=22624198

Family Applications (1)

Application Number Title Priority Date Filing Date
CO00096628A CO5090902A1 (es) 1999-12-22 2000-12-20 Pirroles sustituidos

Country Status (28)

Country Link
US (1) US6281356B1 (xx)
EP (1) EP1242409A2 (xx)
JP (1) JP2003518112A (xx)
KR (1) KR100508741B1 (xx)
CN (1) CN1193027C (xx)
AR (1) AR027035A1 (xx)
AU (1) AU782920B2 (xx)
BR (1) BR0016516A (xx)
CA (1) CA2394852A1 (xx)
CO (1) CO5090902A1 (xx)
CZ (1) CZ20022492A3 (xx)
HK (1) HK1054382A1 (xx)
HR (1) HRP20020536A2 (xx)
HU (1) HUP0204572A3 (xx)
IL (1) IL150200A0 (xx)
JO (1) JO2199B1 (xx)
MA (1) MA26860A1 (xx)
MX (1) MXPA02006162A (xx)
MY (1) MY133682A (xx)
NO (1) NO20022927D0 (xx)
NZ (1) NZ519359A (xx)
PE (1) PE20011098A1 (xx)
PL (1) PL357603A1 (xx)
RU (1) RU2261862C2 (xx)
UY (1) UY26498A1 (xx)
WO (1) WO2001046178A2 (xx)
YU (1) YU46302A (xx)
ZA (1) ZA200204313B (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030139373A1 (en) * 2001-11-20 2003-07-24 Breimer Lars Holger Method for cancer therapy
TW200918046A (en) 2002-04-03 2009-05-01 Novartis Ag Indolylmaleimide derivatives
GB0303319D0 (en) 2003-02-13 2003-03-19 Novartis Ag Organic compounds
PE20151997A1 (es) 2013-03-15 2016-01-13 Plexxikon Inc Compuestos heterociclicos y usos de los mismos
US20140303121A1 (en) 2013-03-15 2014-10-09 Plexxikon Inc. Heterocyclic compounds and uses thereof
HUE045355T2 (hu) * 2016-07-21 2019-12-30 Inst Farmakologii Polskiej Akademii Nauk Az 5-HT7 szerotoninreceptort kötõ imidazolil-szubsztituált indolszármazékok és gyógyszerészeti készítményeik
CA3079029A1 (en) 2017-10-13 2019-04-18 Plexxikon Inc. Solid forms of a compound for modulating kinases

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK278989B6 (sk) 1988-02-10 1998-05-06 F. Hoffmann-La Roche Ag Substituované pyroly, ich použitie na výrobu lieči
US5380746A (en) 1989-05-05 1995-01-10 Goedecke Aktiengesellschaft Bis-(1H-indol-3-YL)-maleinimide derivatives, processes for the preparation thereof and pharmaceutical compositions containing them
PT93947B (pt) * 1989-05-05 1996-11-29 Goedecke Ag Processo para a preparacao de novos derivados de maleinimidas e de composicoes farmaceuticas que os contem
EP0630242B1 (en) * 1992-03-20 1999-01-20 The Wellcome Foundation Limited Further indole derivatives with antiviral activity
EP0630241A1 (en) 1992-03-20 1994-12-28 The Wellcome Foundation Limited Indole derivatives with antiviral activity
DE4217964A1 (de) * 1992-05-30 1993-12-02 Goedecke Ag Indolocarbazol-Imide und deren Verwendung
PE91598A1 (es) 1996-07-29 1998-12-24 Hoffmann La Roche Pirroles sustituidos
PE91698A1 (es) 1996-07-29 1998-12-24 Hoffmann La Roche Pirroles sustituidos
PE91498A1 (es) 1996-07-29 1998-12-22 Hoffmann La Roche Pirroles sustituidos
CZ299068B6 (cs) * 1998-03-17 2008-04-16 F. Hoffmann-La Roche Ag Substituovaný bisindolylmaleinimid a farmaceutický prostredek s jeho obsahem

Also Published As

Publication number Publication date
HRP20020536A2 (en) 2004-08-31
AU3726701A (en) 2001-07-03
WO2001046178A2 (en) 2001-06-28
JO2199B1 (en) 2003-12-23
NZ519359A (en) 2004-04-30
RU2002119557A (ru) 2004-01-10
IL150200A0 (en) 2002-12-01
CZ20022492A3 (cs) 2003-02-12
HK1054382A1 (en) 2003-11-28
YU46302A (sh) 2005-06-10
EP1242409A2 (en) 2002-09-25
AU782920B2 (en) 2005-09-08
KR20020062365A (ko) 2002-07-25
US6281356B1 (en) 2001-08-28
MY133682A (en) 2007-11-30
ZA200204313B (en) 2003-08-29
MXPA02006162A (es) 2002-12-05
BR0016516A (pt) 2002-09-17
UY26498A1 (es) 2001-06-29
CN1411457A (zh) 2003-04-16
PL357603A1 (en) 2004-07-26
KR100508741B1 (ko) 2005-08-17
MA26860A1 (fr) 2004-12-20
AR027035A1 (es) 2003-03-12
CA2394852A1 (en) 2001-06-28
HUP0204572A2 (en) 2003-05-28
PE20011098A1 (es) 2001-10-26
JP2003518112A (ja) 2003-06-03
HUP0204572A3 (en) 2004-07-28
NO20022927L (no) 2002-06-18
CN1193027C (zh) 2005-03-16
NO20022927D0 (no) 2002-06-18
RU2261862C2 (ru) 2005-10-10
WO2001046178A3 (en) 2001-12-06

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