CO2018011935A2 - Derivados aromáticos de sulfonamida - Google Patents

Derivados aromáticos de sulfonamida

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Publication number
CO2018011935A2
CO2018011935A2 CONC2018/0011935A CO2018011935A CO2018011935A2 CO 2018011935 A2 CO2018011935 A2 CO 2018011935A2 CO 2018011935 A CO2018011935 A CO 2018011935A CO 2018011935 A2 CO2018011935 A2 CO 2018011935A2
Authority
CO
Colombia
Prior art keywords
aromatic derivatives
sulfonamide
sulfonamide aromatic
compounds
derivatives
Prior art date
Application number
CONC2018/0011935A
Other languages
English (en)
Inventor
Arwed Cleve
Stefan Werner
Stefanie Mesch
Nico Bräuer
Simon Anthony Herbert
Markus Koch
Henrik Dahllöf
Maren Osmers
Elizabeth Hardaker
Anton Lishchynskyi
Original Assignee
Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of CO2018011935A2 publication Critical patent/CO2018011935A2/es

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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
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    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • C07C311/15Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
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    • C07C311/17Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom to an acyclic carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
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    • C07C311/38Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring having sulfur atoms of sulfonamide groups and amino groups bound to carbon atoms of six-membered rings of the same carbon skeleton
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Abstract

Sulfonamidas aromáticas sustituidas de la fórmula (I) (I) composiciones farmacéuticas y combinaciones que comprenden dichos compuestos y el uso de dichos compuestos para elaborar una composición farmacéutica para el tratamiento o la profilaxis de una enfermedad.
CONC2018/0011935A 2016-05-03 2018-11-02 Derivados aromáticos de sulfonamida CO2018011935A2 (es)

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