CN87104582A - 制备酰化的杂环化合物的方法 - Google Patents

制备酰化的杂环化合物的方法 Download PDF

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Publication number
CN87104582A
CN87104582A CN198787104582A CN87104582A CN87104582A CN 87104582 A CN87104582 A CN 87104582A CN 198787104582 A CN198787104582 A CN 198787104582A CN 87104582 A CN87104582 A CN 87104582A CN 87104582 A CN87104582 A CN 87104582A
Authority
CN
China
Prior art keywords
bromo
formula
tetramethyleneimine
product
monohydrate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN198787104582A
Other languages
English (en)
Chinese (zh)
Inventor
雅诺斯·汤普
雅诺斯·弗舍尔
拉兹罗·多贝
拉兹罗·孔兹
米哈里·马约
伊瓦·培特伊
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Egis Pharmaceuticals PLC
Original Assignee
Egis Pharmaceuticals PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egis Pharmaceuticals PLC filed Critical Egis Pharmaceuticals PLC
Publication of CN87104582A publication Critical patent/CN87104582A/zh
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/12—Oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C22—METALLURGY; FERROUS OR NON-FERROUS ALLOYS; TREATMENT OF ALLOYS OR NON-FERROUS METALS
    • C22B—PRODUCTION AND REFINING OF METALS; PRETREATMENT OF RAW MATERIALS
    • C22B9/00—General processes of refining or remelting of metals; Apparatus for electroslag or arc remelting of metals
    • C22B9/02—Refining by liquating, filtering, centrifuging, distilling, or supersonic wave action including acoustic waves

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Acoustics & Sound (AREA)
  • Manufacturing & Machinery (AREA)
  • Physics & Mathematics (AREA)
  • Mechanical Engineering (AREA)
  • Metallurgy (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CN198787104582A 1986-07-04 1987-07-03 制备酰化的杂环化合物的方法 Pending CN87104582A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU862811A HU196368B (en) 1986-07-04 1986-07-04 Process for production of 1-/3-brom-/25/-methil-prophionil/-pirrolidin-/25/-carbonic acid
HU2811/86 1986-07-04

Publications (1)

Publication Number Publication Date
CN87104582A true CN87104582A (zh) 1988-01-20

Family

ID=10961203

Family Applications (1)

Application Number Title Priority Date Filing Date
CN198787104582A Pending CN87104582A (zh) 1986-07-04 1987-07-03 制备酰化的杂环化合物的方法

Country Status (19)

Country Link
JP (1) JPS6322557A (it)
KR (1) KR880001589A (it)
CN (1) CN87104582A (it)
AT (1) AT387382B (it)
CH (1) CH672786A5 (it)
CS (1) CS262693B2 (it)
DD (1) DD263984A5 (it)
DE (1) DE3722278A1 (it)
DK (1) DK343587A (it)
ES (1) ES2004443A6 (it)
FI (1) FI872966A (it)
GR (1) GR871051B (it)
HU (1) HU196368B (it)
IT (1) IT1221952B (it)
NO (1) NO872796L (it)
PL (1) PL150350B1 (it)
PT (1) PT85256B (it)
SE (1) SE8702753L (it)
YU (1) YU118087A (it)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103086939A (zh) * 2011-10-28 2013-05-08 华中药业股份有限公司 1-(3-溴-2-d-甲基丙酰基)吡咯烷-2-羧酸的重结晶方法

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8802849A (nl) * 1988-11-18 1990-06-18 Stamicarbon Werkwijze voor de enantioselectieve bereiding van d-(-)-3-hal-methylpropionzuur of derivaten daarvan en de bereiding van captopril daaruit.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU184082B (en) * 1979-12-29 1984-06-28 Egyt Gyogyszervegyeszeti Gyar Process for preparing 1-3-/3mercapto-/2s/-methyl-propinyl/-pyrrolidine-/2s/-carboxylic acid
IE50839B1 (en) * 1980-02-26 1986-07-23 Wyeth John & Brother Ltd Novel processes for preparing proline derivatives and analogous compounds

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103086939A (zh) * 2011-10-28 2013-05-08 华中药业股份有限公司 1-(3-溴-2-d-甲基丙酰基)吡咯烷-2-羧酸的重结晶方法

Also Published As

Publication number Publication date
SE8702753L (sv) 1988-01-05
FI872966A (fi) 1988-01-05
GR871051B (en) 1987-11-09
DD263984A5 (de) 1989-01-18
DE3722278A1 (de) 1988-01-07
CS505187A2 (en) 1988-08-16
ES2004443A6 (es) 1989-01-01
IT1221952B (it) 1990-08-31
PT85256A (en) 1987-08-01
PT85256B (pt) 1990-03-30
KR880001589A (ko) 1988-04-25
NO872796L (no) 1988-01-05
IT8721179A0 (it) 1987-07-03
HU196368B (en) 1988-11-28
DK343587D0 (da) 1987-07-03
HUT44491A (en) 1988-03-28
JPS6322557A (ja) 1988-01-30
DK343587A (da) 1988-01-05
CH672786A5 (it) 1989-12-29
FI872966A0 (fi) 1987-07-03
NO872796D0 (no) 1987-07-03
PL150350B1 (en) 1990-05-31
YU118087A (en) 1988-06-30
PL266620A1 (en) 1988-07-07
ATA168087A (de) 1988-06-15
AT387382B (de) 1989-01-10
SE8702753D0 (sv) 1987-07-03
CS262693B2 (en) 1989-03-14

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WD01 Invention patent application deemed withdrawn after publication