CN1714076A - 芳基脲基衍生物及其医药用途 - Google Patents

芳基脲基衍生物及其医药用途 Download PDF

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Publication number
CN1714076A
CN1714076A CNA200380103761XA CN200380103761A CN1714076A CN 1714076 A CN1714076 A CN 1714076A CN A200380103761X A CNA200380103761X A CN A200380103761XA CN 200380103761 A CN200380103761 A CN 200380103761A CN 1714076 A CN1714076 A CN 1714076A
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alkyl
cycloalkyl
halogen
phenyl
chloro
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Chinese (zh)
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J·瓦尔盖尔森
E·O·尼尔森
D·彼得斯
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NTG Nordic Transport Group AS
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Neurosearch AS
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  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Addiction (AREA)
  • Ophthalmology & Optometry (AREA)
  • Otolaryngology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Materials For Medical Uses (AREA)
CNA200380103761XA 2002-11-21 2003-11-10 芳基脲基衍生物及其医药用途 Pending CN1714076A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200201803 2002-11-21
DKPA200201803 2002-11-21

Publications (1)

Publication Number Publication Date
CN1714076A true CN1714076A (zh) 2005-12-28

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Country Status (13)

Country Link
US (1) US7521480B2 (https=)
EP (1) EP1565429B1 (https=)
JP (1) JP2006507329A (https=)
CN (1) CN1714076A (https=)
AT (1) ATE431335T1 (https=)
AU (1) AU2003280308A1 (https=)
CA (1) CA2502705A1 (https=)
DE (1) DE60327652D1 (https=)
ES (1) ES2327834T3 (https=)
MX (1) MXPA05005409A (https=)
NZ (1) NZ539499A (https=)
PT (1) PT1565429E (https=)
WO (1) WO2004046090A2 (https=)

Cited By (5)

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Publication number Priority date Publication date Assignee Title
CN106008371A (zh) * 2016-06-24 2016-10-12 谢阳 1-芳基脲基环烷基-1-甲酰胺类化合物及其药物组合物和应用
CN106946786A (zh) * 2017-04-11 2017-07-14 白银澐新生物科技有限公司 一种1‑苄基‑3‑羟基‑1h‑3‑吲唑钠盐的制备方法
WO2017219935A1 (zh) * 2016-06-22 2017-12-28 复旦大学 联芳基脲类衍生物或其盐及其制备方法和用途
CN111116420A (zh) * 2019-12-31 2020-05-08 浙江工业大学 一种对称脲类化合物的制备方法
CN114539080A (zh) * 2022-03-02 2022-05-27 八叶草健康产业研究院(厦门)有限公司 一种2-(2-氨基-6-氯苯基)-乙酸钠的制备方法

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US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
AU2005304962B2 (en) * 2004-11-09 2009-11-19 Smithkline Beecham Corporation Glycogen phosphorylase inhibitor compounds and pharmaceutical compositions thereof
FR2878522B1 (fr) * 2004-12-01 2008-04-18 Merck Sante Soc Par Actions Si Nouveaux inhibiteurs specifiques de la caspas-10
MX2007007029A (es) * 2004-12-17 2007-08-08 Neurosearch As Derivados de difenilurea utiles como activadores del canal de potasio.
EP1954696B1 (en) 2005-01-19 2011-02-23 Bristol-Myers Squibb Company 2-phenoxy-n-(1,3,4-thiadizol-2-yl)pyridin-3-amine derivatives and related compounds as p2y1 receptor inhibitors for the treatment of thromboembolic disorders
AR056867A1 (es) 2005-06-27 2007-10-31 Bristol Myers Squibb Co Antagonistas heterociclicos n- enlazados del receptor de p2y1 utiles en el tratamiento de condiciones tromboticas. composiciones farmaceuticas.
DE602006020871D1 (de) 2005-06-27 2011-05-05 Bristol Myers Squibb Co Lineare harnstoffmimetika-antagonisten des p2y1-rezeptors zur behandlung von thromboseleiden
WO2007002634A1 (en) 2005-06-27 2007-01-04 Bristol-Myers Squibb Company Carbocycle and heterocycle antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
EP1899299B1 (en) 2005-06-27 2010-10-20 Bristol-Myers Squibb Company C-linked cyclic antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
US8053454B2 (en) 2005-10-06 2011-11-08 Exelixis, Inc. Pyridopyrimidinone inhibitors of PIM-1 and/or PIM-3
AU2007224457A1 (en) * 2006-03-14 2007-09-20 Neurosearch A/S Diphenylurea derivatives and their use as chloride channel blockers or BKca channel modulators
US7960569B2 (en) 2006-10-17 2011-06-14 Bristol-Myers Squibb Company Indole antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
DE102007012908A1 (de) 2007-03-19 2008-09-25 Momentive Performance Materials Gmbh Neue Polyamid-Polysiloxan-Verbindungen
KR20100087300A (ko) * 2007-09-28 2010-08-04 글락소스미스클라인 엘엘씨 글리코겐 포스포릴라아제 억제제 화합물 및 이의 약학적 조성물
EP2225214A1 (en) * 2007-11-28 2010-09-08 NeuroSearch AS Novel phenyl-acetamide and phenyl-propionamide derivatives useful as potassium channel modulators
EP2493468A1 (en) * 2009-10-30 2012-09-05 Sanofi Amino-benzoic acid derivatives for use in the treatment of dihydrogenase-related disorders
WO2016127085A1 (en) * 2015-02-07 2016-08-11 University Of Pittsburgh - Of The Commonwealth System Of Higher Education hTRPV1 CHEMICAL AGENTS

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EP1565429B1 (en) 2009-05-13
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