CN1649848A - 作为促肾上腺皮质激素释放因子(crf)拮抗剂的稠合嘧啶衍生物 - Google Patents

作为促肾上腺皮质激素释放因子(crf)拮抗剂的稠合嘧啶衍生物 Download PDF

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Publication number
CN1649848A
CN1649848A CNA028107462A CN02810746A CN1649848A CN 1649848 A CN1649848 A CN 1649848A CN A028107462 A CNA028107462 A CN A028107462A CN 02810746 A CN02810746 A CN 02810746A CN 1649848 A CN1649848 A CN 1649848A
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China
Prior art keywords
methyl
pyrimidine
dihydro
pyrrolo
compound
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Pending
Application number
CNA028107462A
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Chinese (zh)
Inventor
罗马诺·迪法比奥
安娜·M·卡佩利
恰拉·马奇奥尼
法布里齐奥·米歇利
亚历山德拉·帕斯奎里洛
贝尼德塔·佩里尼
伊维斯·圣丹尼斯
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Glaxo Group Ltd
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Glaxo Group Ltd
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Priority claimed from GB0110570A external-priority patent/GB0110570D0/en
Priority claimed from GB0110569A external-priority patent/GB0110569D0/en
Priority claimed from GB0110567A external-priority patent/GB0110567D0/en
Priority claimed from GB0117401A external-priority patent/GB0117401D0/en
Priority claimed from GB0117420A external-priority patent/GB0117420D0/en
Priority claimed from GB0117399A external-priority patent/GB0117399D0/en
Priority claimed from GB0203201A external-priority patent/GB0203201D0/en
Priority claimed from GB0206834A external-priority patent/GB0206834D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of CN1649848A publication Critical patent/CN1649848A/zh
Pending legal-status Critical Current

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CNA028107462A 2001-04-30 2002-04-30 作为促肾上腺皮质激素释放因子(crf)拮抗剂的稠合嘧啶衍生物 Pending CN1649848A (zh)

Applications Claiming Priority (16)

Application Number Priority Date Filing Date Title
GB0110569.1 2001-04-30
GB0110570A GB0110570D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110569A GB0110569D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110570.9 2001-04-30
GB0110567.5 2001-04-30
GB0110567A GB0110567D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0117401.0 2001-07-17
GB0117401A GB0117401D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117420A GB0117420D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117399.6 2001-07-17
GB0117399A GB0117399D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117420.0 2001-07-17
GB0203201.9 2002-02-11
GB0203201A GB0203201D0 (en) 2002-02-11 2002-02-11 Chemical compounds
GB0206834.4 2002-03-22
GB0206834A GB0206834D0 (en) 2002-03-22 2002-03-22 Chemical compounds

Publications (1)

Publication Number Publication Date
CN1649848A true CN1649848A (zh) 2005-08-03

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CNA028107462A Pending CN1649848A (zh) 2001-04-30 2002-04-30 作为促肾上腺皮质激素释放因子(crf)拮抗剂的稠合嘧啶衍生物

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Cited By (1)

* Cited by examiner, † Cited by third party
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CN104193745A (zh) * 2014-07-30 2014-12-10 天津市斯芬克司药物研发有限公司 一种咪唑并嘧啶羧酸类化合物及其制备方法

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WO2002100863A1 (en) * 2001-06-12 2002-12-19 Glaxo Group Limited Corticotropin releasing factor antagonists
GB0117396D0 (en) * 2001-07-17 2001-09-05 Glaxo Group Ltd Chemical compounds
EP1583531B1 (en) * 2003-01-16 2007-04-18 SB Pharmco Puerto Rico Inc Heteroaryl-substituted pyrrolo[2, 3- b]pyridine derivatives as crf receptor antagonists
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
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