CN1227241C - 具有5-羟色胺1a受体活性的芳基哌嗪类化合物 - Google Patents
具有5-羟色胺1a受体活性的芳基哌嗪类化合物 Download PDFInfo
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- CN1227241C CN1227241C CNB988135191A CN98813519A CN1227241C CN 1227241 C CN1227241 C CN 1227241C CN B988135191 A CNB988135191 A CN B988135191A CN 98813519 A CN98813519 A CN 98813519A CN 1227241 C CN1227241 C CN 1227241C
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- alkyl
- phenyl
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- hydrogen
- cycloalkyl
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- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/092—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings with aromatic radicals attached to the chain
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- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/10—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms
- C07D295/104—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by doubly bound oxygen or sulphur atoms with the ring nitrogen atoms and the doubly bound oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
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- Chemical & Material Sciences (AREA)
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- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Epidemiology (AREA)
- Addiction (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6979197P | 1997-12-16 | 1997-12-16 | |
| US6972297P | 1997-12-16 | 1997-12-16 | |
| US60/069,722 | 1997-12-16 | ||
| US60/069,791 | 1997-12-16 | ||
| US8958998P | 1998-06-17 | 1998-06-17 | |
| US60/089,589 | 1998-06-17 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB2005101041777A Division CN100355714C (zh) | 1997-12-16 | 1998-12-08 | 具有5-羟色胺1a受体活性的芳基哌嗪类化合物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN1290258A CN1290258A (zh) | 2001-04-04 |
| CN1227241C true CN1227241C (zh) | 2005-11-16 |
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ID=27371593
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB988135191A Expired - Fee Related CN1227241C (zh) | 1997-12-16 | 1998-12-08 | 具有5-羟色胺1a受体活性的芳基哌嗪类化合物 |
| CNB2005101041777A Expired - Fee Related CN100355714C (zh) | 1997-12-16 | 1998-12-08 | 具有5-羟色胺1a受体活性的芳基哌嗪类化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB2005101041777A Expired - Fee Related CN100355714C (zh) | 1997-12-16 | 1998-12-08 | 具有5-羟色胺1a受体活性的芳基哌嗪类化合物 |
Country Status (32)
| Country | Link |
|---|---|
| US (9) | US6239135B1 (https=) |
| EP (2) | EP0924205B1 (https=) |
| JP (2) | JP2002508364A (https=) |
| KR (1) | KR100539651B1 (https=) |
| CN (2) | CN1227241C (https=) |
| AR (1) | AR017864A1 (https=) |
| AT (1) | ATE296296T1 (https=) |
| AU (1) | AU747040B2 (https=) |
| BR (1) | BR9814280A (https=) |
| CA (2) | CA2506802A1 (https=) |
| CO (1) | CO4980859A1 (https=) |
| DE (1) | DE69830297T2 (https=) |
| DK (1) | DK0924205T3 (https=) |
| EA (1) | EA003703B1 (https=) |
| EG (1) | EG23983A (https=) |
| ES (1) | ES2244036T3 (https=) |
| HR (1) | HRP20000406B1 (https=) |
| HU (1) | HU226409B1 (https=) |
| ID (1) | ID26930A (https=) |
| IL (3) | IL136723A0 (https=) |
| MY (1) | MY125868A (https=) |
| NO (1) | NO317098B1 (https=) |
| NZ (1) | NZ505220A (https=) |
| PE (1) | PE20000134A1 (https=) |
| PL (1) | PL193428B1 (https=) |
| PT (1) | PT924205E (https=) |
| SV (1) | SV1998000148A (https=) |
| TR (1) | TR200001727T2 (https=) |
| TW (1) | TW520366B (https=) |
| UA (1) | UA66370C2 (https=) |
| WO (1) | WO1999031077A1 (https=) |
| ZA (1) | ZA9811473B (https=) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA66370C2 (en) * | 1997-12-16 | 2004-05-17 | Lilly Co Eli | Arylpiperazines having activity to setotonin 1 receptors |
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