CN116171273B - 化合物的制造方法 - Google Patents

化合物的制造方法 Download PDF

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Publication number
CN116171273B
CN116171273B CN202180060304.5A CN202180060304A CN116171273B CN 116171273 B CN116171273 B CN 116171273B CN 202180060304 A CN202180060304 A CN 202180060304A CN 116171273 B CN116171273 B CN 116171273B
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CN116171273A (zh
Inventor
张替僚
小岛千绘美
今野慎悟
山崎徹
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Kureha Corp
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Kureha Corp
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D301/00Preparation of oxiranes
    • C07D301/02Synthesis of the oxirane ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D303/00Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02Compounds containing oxirane rings
    • C07D303/48Compounds containing oxirane rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/63Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00Preparation of carboxylic acid esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00Preparation of carboxylic acid esters
    • C07C67/27Preparation of carboxylic acid esters from ortho-esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00Preparation of carboxylic acid esters
    • C07C67/39Preparation of carboxylic acid esters by oxidation of groups which are precursors for the acid moiety of the ester
    • C07C67/42Preparation of carboxylic acid esters by oxidation of groups which are precursors for the acid moiety of the ester by oxidation of secondary alcohols or ketones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CN202180060304.5A 2020-08-06 2021-08-06 化合物的制造方法 Active CN116171273B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2020134138 2020-08-06
JP2020-134138 2020-08-06
PCT/JP2021/029343 WO2022030622A1 (ja) 2020-08-06 2021-08-06 化合物の製造方法

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CN116171273A CN116171273A (zh) 2023-05-26
CN116171273B true CN116171273B (zh) 2024-05-14

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US (1) US12428387B2 (https=)
EP (1) EP4194445B1 (https=)
JP (1) JP7427096B2 (https=)
CN (1) CN116171273B (https=)
WO (1) WO2022030622A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2978668T3 (es) 2019-04-19 2024-09-17 Kureha Corp Agente fungicida para uso agrícola u hortícola, método de control de enfermedades de las plantas, y producto para el uso en el control de enfermedades de las plantas

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CN104540818A (zh) * 2012-10-11 2015-04-22 株式会社吴羽 环烷醇衍生物制备方法及唑衍生物制备方法
WO2016005211A1 (en) * 2014-07-08 2016-01-14 Basf Se Process for the preparation of substituted oxiranes and triazoles
WO2019093522A1 (ja) * 2017-11-13 2019-05-16 株式会社クレハ アゾール誘導体、中間体化合物、及びアゾール誘導体の製造方法、ならびに農園芸用薬剤及び工業用材料保護剤

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DE3315619A1 (de) 1983-04-29 1984-10-31 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von oxiranen
GB9125791D0 (en) 1991-12-04 1992-02-05 Schering Agrochemicals Ltd Herbicides
DE10349503A1 (de) 2003-10-23 2005-05-25 Bayer Cropscience Ag Fungizide Wirkstoffkombinationen
DE102004045242A1 (de) 2004-09-17 2006-03-23 Bayer Cropscience Ag Synergistische fungizide Wirkstoffkombinationen
US20120108422A1 (en) 2009-06-18 2012-05-03 Basf Se Antifungal 1,2,4-triazolyl Derivatives
JP5852562B2 (ja) 2010-04-28 2016-02-03 塩野義製薬株式会社 新規なセフェム誘導体
US20150051231A1 (en) 2010-09-29 2015-02-19 Fmc Quimica Do Brasil Ltda. Synergistic combinations of triazoles, strobilurins and benzimidazoles, uses, formulations, production processes and applications using the same
US20140142185A1 (en) 2011-03-14 2014-05-22 Shalini Sharma 3-Benzyloxyphenyloxoacetic Acid Compounds for Reducing Uric Acid
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EA030875B1 (ru) 2012-12-20 2018-10-31 Басф Агро Б.В. Композиции, содержащие триазольное соединение
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AR100743A1 (es) 2014-06-06 2016-10-26 Basf Se Compuestos de [1,2,4]triazol sustituido
MX2018001885A (es) 2015-08-14 2018-08-16 Bayer Cropscience Ag Derivados de triazol, sus intermediarios y su utilizacion como fungicidas.
CA3052898A1 (en) 2017-02-10 2018-08-16 Bayer Aktiengesellschaft Composition for controlling harmful microorganisms comprising 1 -(phenoxy-pyridinyl)-2-(1,2,4-triazol-1 -yl)-ethanol derivatives
JP2019206375A (ja) 2018-05-30 2019-12-05 Toto株式会社 梱包箱
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ES2978668T3 (es) 2019-04-19 2024-09-17 Kureha Corp Agente fungicida para uso agrícola u hortícola, método de control de enfermedades de las plantas, y producto para el uso en el control de enfermedades de las plantas
CN115209737B (zh) 2020-02-27 2025-08-15 先正达农作物保护股份公司 杀真菌组合物

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JP2012530110A (ja) * 2009-06-18 2012-11-29 ビーエーエスエフ ソシエタス・ヨーロピア 抗菌性1,2,4−トリアゾリル誘導体
CN103930417A (zh) * 2011-11-11 2014-07-16 株式会社吴羽 4-苄基-1-甲基-6-氧杂二环[3,2,0]庚烷衍生物的制造方法
CN104540818A (zh) * 2012-10-11 2015-04-22 株式会社吴羽 环烷醇衍生物制备方法及唑衍生物制备方法
CN103059004A (zh) * 2012-12-21 2013-04-24 泰州职业技术学院 一种制备1-[α-(2,4-二氟苯基)-2,3-环氧丙基]-1H-1,2,4-三氮唑方法
WO2016005211A1 (en) * 2014-07-08 2016-01-14 Basf Se Process for the preparation of substituted oxiranes and triazoles
WO2019093522A1 (ja) * 2017-11-13 2019-05-16 株式会社クレハ アゾール誘導体、中間体化合物、及びアゾール誘導体の製造方法、ならびに農園芸用薬剤及び工業用材料保護剤

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US20230271929A1 (en) 2023-08-31
JPWO2022030622A1 (https=) 2022-02-10
US12428387B2 (en) 2025-09-30
CN116171273A (zh) 2023-05-26
WO2022030622A1 (ja) 2022-02-10
EP4194445A1 (en) 2023-06-14
JP7427096B2 (ja) 2024-02-02
EP4194445B1 (en) 2025-04-16
EP4194445A4 (en) 2024-08-14

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