CN116171273B - 化合物的制造方法 - Google Patents
化合物的制造方法 Download PDFInfo
- Publication number
- CN116171273B CN116171273B CN202180060304.5A CN202180060304A CN116171273B CN 116171273 B CN116171273 B CN 116171273B CN 202180060304 A CN202180060304 A CN 202180060304A CN 116171273 B CN116171273 B CN 116171273B
- Authority
- CN
- China
- Prior art keywords
- general formula
- compound represented
- group
- formula
- added
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D301/00—Preparation of oxiranes
- C07D301/02—Synthesis of the oxirane ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/48—Compounds containing oxirane rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/27—Preparation of carboxylic acid esters from ortho-esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/39—Preparation of carboxylic acid esters by oxidation of groups which are precursors for the acid moiety of the ester
- C07C67/42—Preparation of carboxylic acid esters by oxidation of groups which are precursors for the acid moiety of the ester by oxidation of secondary alcohols or ketones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020134138 | 2020-08-06 | ||
| JP2020-134138 | 2020-08-06 | ||
| PCT/JP2021/029343 WO2022030622A1 (ja) | 2020-08-06 | 2021-08-06 | 化合物の製造方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN116171273A CN116171273A (zh) | 2023-05-26 |
| CN116171273B true CN116171273B (zh) | 2024-05-14 |
Family
ID=80118171
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202180060304.5A Active CN116171273B (zh) | 2020-08-06 | 2021-08-06 | 化合物的制造方法 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US12428387B2 (https=) |
| EP (1) | EP4194445B1 (https=) |
| JP (1) | JP7427096B2 (https=) |
| CN (1) | CN116171273B (https=) |
| WO (1) | WO2022030622A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2978668T3 (es) | 2019-04-19 | 2024-09-17 | Kureha Corp | Agente fungicida para uso agrícola u hortícola, método de control de enfermedades de las plantas, y producto para el uso en el control de enfermedades de las plantas |
Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012530110A (ja) * | 2009-06-18 | 2012-11-29 | ビーエーエスエフ ソシエタス・ヨーロピア | 抗菌性1,2,4−トリアゾリル誘導体 |
| CN103059004A (zh) * | 2012-12-21 | 2013-04-24 | 泰州职业技术学院 | 一种制备1-[α-(2,4-二氟苯基)-2,3-环氧丙基]-1H-1,2,4-三氮唑方法 |
| CN103930417A (zh) * | 2011-11-11 | 2014-07-16 | 株式会社吴羽 | 4-苄基-1-甲基-6-氧杂二环[3,2,0]庚烷衍生物的制造方法 |
| CN104540818A (zh) * | 2012-10-11 | 2015-04-22 | 株式会社吴羽 | 环烷醇衍生物制备方法及唑衍生物制备方法 |
| WO2016005211A1 (en) * | 2014-07-08 | 2016-01-14 | Basf Se | Process for the preparation of substituted oxiranes and triazoles |
| WO2019093522A1 (ja) * | 2017-11-13 | 2019-05-16 | 株式会社クレハ | アゾール誘導体、中間体化合物、及びアゾール誘導体の製造方法、ならびに農園芸用薬剤及び工業用材料保護剤 |
Family Cites Families (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0099165A1 (en) | 1982-03-23 | 1984-01-25 | Imperial Chemical Industries Plc | Triazole and imidazole compounds, process for their preparation and their use as fungicides and plant growth regulators, and intermediates for their synthesis |
| ZA831466B (en) | 1982-03-23 | 1984-10-31 | Ici Plc | Heterocyclic compounds |
| US4533659A (en) | 1982-06-09 | 1985-08-06 | Ciba-Geigy Corporation | Microbicidal 2-(1H-1,2,4-triazolylmethyl-1'-yl)-2-siloxy-2-phenyl-acetates |
| DE3315619A1 (de) | 1983-04-29 | 1984-10-31 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von oxiranen |
| GB9125791D0 (en) | 1991-12-04 | 1992-02-05 | Schering Agrochemicals Ltd | Herbicides |
| DE10349503A1 (de) | 2003-10-23 | 2005-05-25 | Bayer Cropscience Ag | Fungizide Wirkstoffkombinationen |
| DE102004045242A1 (de) | 2004-09-17 | 2006-03-23 | Bayer Cropscience Ag | Synergistische fungizide Wirkstoffkombinationen |
| US20120108422A1 (en) | 2009-06-18 | 2012-05-03 | Basf Se | Antifungal 1,2,4-triazolyl Derivatives |
| JP5852562B2 (ja) | 2010-04-28 | 2016-02-03 | 塩野義製薬株式会社 | 新規なセフェム誘導体 |
| US20150051231A1 (en) | 2010-09-29 | 2015-02-19 | Fmc Quimica Do Brasil Ltda. | Synergistic combinations of triazoles, strobilurins and benzimidazoles, uses, formulations, production processes and applications using the same |
| US20140142185A1 (en) | 2011-03-14 | 2014-05-22 | Shalini Sharma | 3-Benzyloxyphenyloxoacetic Acid Compounds for Reducing Uric Acid |
| DK2731935T3 (en) | 2011-07-13 | 2016-06-06 | Basf Agro Bv | FUNGICIDE SUBSTITUTED 2- [2-HALOGENALKYL-4- (PHENOXY) -PHENYL] -1- [1,2,4] TRIAZOL-1-YLETHANOL COMPOUNDS |
| CN102491959B (zh) | 2011-12-19 | 2015-03-25 | 江苏澄扬作物科技有限公司 | 一种环氧乙烷衍生物的制备方法 |
| WO2013144105A1 (en) | 2012-03-31 | 2013-10-03 | Novozymes A/S | Epoxidation using peroxygenase |
| US20160029630A1 (en) | 2012-11-27 | 2016-02-04 | Basf Se | Substituted 2-[phenoxy-phenyl]-1-[1,2,4]triazol-1-yl-ethanol compounds and their use as fungicides |
| US20150307459A1 (en) | 2012-11-27 | 2015-10-29 | Basf Se | Substituted 2-[phenoxy-phenyl]-1-[1,2,4]triazol-1-yl-ethanol Compounds and Their Use as Fungicides |
| WO2014095672A1 (en) | 2012-12-19 | 2014-06-26 | Basf Se | Substituted [1,2,4]triazole compounds and their use as fungicides |
| CN105164111B (zh) | 2012-12-19 | 2018-11-20 | 巴斯夫欧洲公司 | 取代[1,2,4]三唑及其作为杀真菌剂的用途 |
| EA030875B1 (ru) | 2012-12-20 | 2018-10-31 | Басф Агро Б.В. | Композиции, содержащие триазольное соединение |
| BR112015007183A2 (pt) | 2012-12-20 | 2017-07-04 | Basf Se | composições, uso de uma composição, método para o combate dos fungos e semente |
| WO2015055755A1 (en) | 2013-10-18 | 2015-04-23 | Basf Se | Agricultural mixtures comprising carboxamide compound |
| AR100743A1 (es) | 2014-06-06 | 2016-10-26 | Basf Se | Compuestos de [1,2,4]triazol sustituido |
| MX2018001885A (es) | 2015-08-14 | 2018-08-16 | Bayer Cropscience Ag | Derivados de triazol, sus intermediarios y su utilizacion como fungicidas. |
| CA3052898A1 (en) | 2017-02-10 | 2018-08-16 | Bayer Aktiengesellschaft | Composition for controlling harmful microorganisms comprising 1 -(phenoxy-pyridinyl)-2-(1,2,4-triazol-1 -yl)-ethanol derivatives |
| JP2019206375A (ja) | 2018-05-30 | 2019-12-05 | Toto株式会社 | 梱包箱 |
| JP2019048845A (ja) | 2018-11-07 | 2019-03-28 | 住友化学株式会社 | 複素環化合物を含有する組成物 |
| ES2978668T3 (es) | 2019-04-19 | 2024-09-17 | Kureha Corp | Agente fungicida para uso agrícola u hortícola, método de control de enfermedades de las plantas, y producto para el uso en el control de enfermedades de las plantas |
| CN115209737B (zh) | 2020-02-27 | 2025-08-15 | 先正达农作物保护股份公司 | 杀真菌组合物 |
-
2021
- 2021-08-06 CN CN202180060304.5A patent/CN116171273B/zh active Active
- 2021-08-06 EP EP21853755.3A patent/EP4194445B1/en active Active
- 2021-08-06 WO PCT/JP2021/029343 patent/WO2022030622A1/ja not_active Ceased
- 2021-08-06 US US18/040,365 patent/US12428387B2/en active Active
- 2021-08-06 JP JP2022541750A patent/JP7427096B2/ja active Active
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012530110A (ja) * | 2009-06-18 | 2012-11-29 | ビーエーエスエフ ソシエタス・ヨーロピア | 抗菌性1,2,4−トリアゾリル誘導体 |
| CN103930417A (zh) * | 2011-11-11 | 2014-07-16 | 株式会社吴羽 | 4-苄基-1-甲基-6-氧杂二环[3,2,0]庚烷衍生物的制造方法 |
| CN104540818A (zh) * | 2012-10-11 | 2015-04-22 | 株式会社吴羽 | 环烷醇衍生物制备方法及唑衍生物制备方法 |
| CN103059004A (zh) * | 2012-12-21 | 2013-04-24 | 泰州职业技术学院 | 一种制备1-[α-(2,4-二氟苯基)-2,3-环氧丙基]-1H-1,2,4-三氮唑方法 |
| WO2016005211A1 (en) * | 2014-07-08 | 2016-01-14 | Basf Se | Process for the preparation of substituted oxiranes and triazoles |
| WO2019093522A1 (ja) * | 2017-11-13 | 2019-05-16 | 株式会社クレハ | アゾール誘導体、中間体化合物、及びアゾール誘導体の製造方法、ならびに農園芸用薬剤及び工業用材料保護剤 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20230271929A1 (en) | 2023-08-31 |
| JPWO2022030622A1 (https=) | 2022-02-10 |
| US12428387B2 (en) | 2025-09-30 |
| CN116171273A (zh) | 2023-05-26 |
| WO2022030622A1 (ja) | 2022-02-10 |
| EP4194445A1 (en) | 2023-06-14 |
| JP7427096B2 (ja) | 2024-02-02 |
| EP4194445B1 (en) | 2025-04-16 |
| EP4194445A4 (en) | 2024-08-14 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| SG176212A1 (en) | Process for the production of dronedarone intermediates | |
| JP2015532309A (ja) | オスペミフェンの製造方法 | |
| CN116171273B (zh) | 化合物的制造方法 | |
| JP2002173492A (ja) | 軸不斉を有する光学活性な4級アンモニウム塩とそれを用いたβ−ヒドロキシケトンの立体選択的合成 | |
| US9656947B2 (en) | Process for creating carbon-carbon bonds using carbonyl compounds | |
| AU2012269895A1 (en) | Hybrid molecules containing pharmacophores of fluconazole as antifungal agents and their preparation | |
| WO2019208043A1 (ja) | 窒素上無保護イミン化合物の製造方法 | |
| US9738607B2 (en) | Scalable process for the preparation of Sorafenib tosylate ethanol solvate and Sorafenib tosylate form III | |
| JPS60260555A (ja) | 2‐置換‐5‐メチルピリジン類及びその合成方法 | |
| CN107954960B (zh) | 一种1,3-二氢异苯并呋喃类化合物的合成方法 | |
| Ahmad et al. | Borontribromide-mediated C–C bond formation in cyclic ketones: a transition metal free approach | |
| CN1557808A (zh) | 3-取代哌嗪三氮唑醇类抗真菌化合物及其盐类 | |
| JP7515684B2 (ja) | アゾール誘導体の製造方法 | |
| KR900007628B1 (ko) | 이미다졸 유도체의 제조방법 | |
| JPH04230678A (ja) | 新規の2,3−ジヒドロベンゾフランおよびその製造法 | |
| CN107746388B (zh) | 一种伏立康唑中间体的制备方法 | |
| Lee et al. | Facile Synthesis of Vinyl Sulfones from β-Bromo Alcohols | |
| CN110028437B (zh) | 一种微波促进制备2-苯基-3-醛基吲哚类化合物的方法 | |
| KR100209246B1 (ko) | 트리아졸 유도체의 제조방법 | |
| JP4194984B2 (ja) | フェニルナフチルイミダゾール化合物 | |
| KR101354175B1 (ko) | 2-(3,3-디메톡시)프로파노에이트기로부터 메틸 (e)-2-(3-메톡시)아크릴레이트기의 제조방법 | |
| JP5142241B2 (ja) | ニコチン酸エステル化合物の製造方法 | |
| TW200932730A (en) | Method for preparing 1-methallyl -2-(2'-hydroxyl-5'-methylphenyl) benzotriazole compound and derivatives thereof | |
| KR20120058314A (ko) | 스타틴 화합물의 제조방법 및 이에 사용되는 중간체 화합물 | |
| CN107793392A (zh) | 一种2‑取代‑1‑(2‑噻吩)‑1‑戊酮的合成方法 |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PB01 | Publication | ||
| PB01 | Publication | ||
| SE01 | Entry into force of request for substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| GR01 | Patent grant | ||
| GR01 | Patent grant |