CN115028617A - Cbp/ep300的杂环抑制剂及其在治疗癌症中的用途 - Google Patents

Cbp/ep300的杂环抑制剂及其在治疗癌症中的用途 Download PDF

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CN115028617A
CN115028617A CN202210701205.7A CN202210701205A CN115028617A CN 115028617 A CN115028617 A CN 115028617A CN 202210701205 A CN202210701205 A CN 202210701205A CN 115028617 A CN115028617 A CN 115028617A
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methyl
formula
independently selected
compound
membered
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Chinese (zh)
Inventor
P·西尔
S·布朗纳
F·A·罗梅罗
S·马格努森
V·H-W·徐
J·瓦伊
K·W·赖
F·王
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Genentech Inc
Constellation Pharmaceuticals Inc
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Genentech Inc
Constellation Pharmaceuticals Inc
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  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Transplantation (AREA)
  • Hematology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Peptides Or Proteins (AREA)
CN202210701205.7A 2016-05-24 2017-05-24 Cbp/ep300的杂环抑制剂及其在治疗癌症中的用途 Pending CN115028617A (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CNPCT/CN2016/083124 2016-05-24
CN2016083124 2016-05-24
PCT/US2017/034320 WO2017205536A2 (en) 2016-05-24 2017-05-24 Therapeutic compounds and uses thereof
CN201780045651.4A CN109476641B (zh) 2016-05-24 2017-05-24 Cbp/ep300的杂环抑制剂及其在治疗癌症中的用途

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CN201780045651.4A Active CN109476641B (zh) 2016-05-24 2017-05-24 Cbp/ep300的杂环抑制剂及其在治疗癌症中的用途

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US (2) US10696655B2 (https=)
EP (2) EP3464270B1 (https=)
JP (2) JP7160688B2 (https=)
CN (2) CN115028617A (https=)
MA (1) MA45122A (https=)
WO (1) WO2017205536A2 (https=)

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