CN109069529B - 用于治疗性化合物的靶向配体 - Google Patents

用于治疗性化合物的靶向配体 Download PDF

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CN109069529B
CN109069529B CN201780016137.8A CN201780016137A CN109069529B CN 109069529 B CN109069529 B CN 109069529B CN 201780016137 A CN201780016137 A CN 201780016137A CN 109069529 B CN109069529 B CN 109069529B
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targeting ligand
expression
linked
compound
oligomeric compound
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CN109069529A (zh
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D·B·罗泽玛
D·H·维基菲尔德
A·V·布罗金
J·D·本森
李
裴涛
F·弗雷兹
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Arrowhead Pharmaceuticals Inc
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    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
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    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
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CN201780016137.8A 2016-03-07 2017-03-07 用于治疗性化合物的靶向配体 Active CN109069529B (zh)

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US201662304652P 2016-03-07 2016-03-07
US62/304,652 2016-03-07
US201662370754P 2016-08-04 2016-08-04
US62/370,754 2016-08-04
US201662426916P 2016-11-28 2016-11-28
US62/426,916 2016-11-28
PCT/US2017/021175 WO2017156012A1 (en) 2016-03-07 2017-03-07 Targeting ligands for therapeutic compounds

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US (4) US10246709B2 (OSRAM)
EP (1) EP3426261A4 (OSRAM)
JP (4) JP6983797B2 (OSRAM)
KR (3) KR102515329B1 (OSRAM)
CN (2) CN113797348A (OSRAM)
AU (3) AU2017229469B2 (OSRAM)
BR (1) BR112018068230B1 (OSRAM)
CA (1) CA3011946A1 (OSRAM)
IL (3) IL296377A (OSRAM)
JO (2) JOP20170057B1 (OSRAM)
MX (3) MX2018009854A (OSRAM)
NZ (2) NZ744357A (OSRAM)
TW (3) TWI783434B (OSRAM)
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WO (1) WO2017156012A1 (OSRAM)

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