CN106608867A - 艾氟康唑及其中间体的制备方法、其中间体 - Google Patents
艾氟康唑及其中间体的制备方法、其中间体 Download PDFInfo
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- CN106608867A CN106608867A CN201510696284.7A CN201510696284A CN106608867A CN 106608867 A CN106608867 A CN 106608867A CN 201510696284 A CN201510696284 A CN 201510696284A CN 106608867 A CN106608867 A CN 106608867A
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- 0 *C*(C(*)=O)c(c(F)c1)ccc1F Chemical compound *C*(C(*)=O)c(c(F)c1)ccc1F 0.000 description 3
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Abstract
Description
Claims (10)
Priority Applications (1)
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CN201510696284.7A CN106608867B (zh) | 2015-10-23 | 2015-10-23 | 艾氟康唑及其中间体的制备方法、其中间体 |
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CN201510696284.7A CN106608867B (zh) | 2015-10-23 | 2015-10-23 | 艾氟康唑及其中间体的制备方法、其中间体 |
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CN106608867A true CN106608867A (zh) | 2017-05-03 |
CN106608867B CN106608867B (zh) | 2019-09-13 |
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Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2020133411A1 (zh) | 2018-12-29 | 2020-07-02 | 山东威智医药工业有限公司 | 一种艾氟康唑的制备方法 |
US10829475B2 (en) | 2017-05-19 | 2020-11-10 | Kaken Pharmaceutical Co., Ltd. | Production and purification methods for efinaconazole |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1906146A (zh) * | 2003-11-27 | 2007-01-31 | 住友化学株式会社 | 环氧基三唑化合物的制备方法及其中间体 |
CN104557746A (zh) * | 2015-01-19 | 2015-04-29 | 苏州信恩医药科技有限公司 | 一种艾氟康唑中间体的合成方法 |
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2015
- 2015-10-23 CN CN201510696284.7A patent/CN106608867B/zh active Active
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1906146A (zh) * | 2003-11-27 | 2007-01-31 | 住友化学株式会社 | 环氧基三唑化合物的制备方法及其中间体 |
CN104557746A (zh) * | 2015-01-19 | 2015-04-29 | 苏州信恩医药科技有限公司 | 一种艾氟康唑中间体的合成方法 |
Non-Patent Citations (2)
Title |
---|
VITO CAPRIATI等: "Oxiranyl Anion-Mediated Synthesis of Highly Enantiomerically Enriched Styrene Oxide Derivatives", 《ORGANIC LETTERS》 * |
王积涛: "《有机化学第三版上册》", 31 December 2009 * |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US10829475B2 (en) | 2017-05-19 | 2020-11-10 | Kaken Pharmaceutical Co., Ltd. | Production and purification methods for efinaconazole |
WO2020133411A1 (zh) | 2018-12-29 | 2020-07-02 | 山东威智医药工业有限公司 | 一种艾氟康唑的制备方法 |
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CN106608867B (zh) | 2019-09-13 |
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Address after: 277514 No.88, Weizhi Avenue, Tengzhou biomedical industrial park, Zaozhuang City, Shandong Province Co-patentee after: SHANGHAI VIWIT PHARMACEUTICAL Co.,Ltd. Patentee after: Weizhi Pharmaceutical Co.,Ltd. Address before: 88 No. 277514 Shandong city of Zaozhuang province Tengzhou biological medicine industry base wise Avenue Co-patentee before: SHANGHAI VIWIT PHARMACEUTICAL Co.,Ltd. Patentee before: VIWIT PHARMACEUTICAL Co.,Ltd. |
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Address after: 88 No. 277514 Shandong city of Zaozhuang province Tengzhou biological medicine industry base wise Avenue Co-patentee after: SHANGHAI VIWIT PHARMACEUTICAL Co.,Ltd. Patentee after: Weizhi Pharmaceutical Co.,Ltd. Address before: 277514 No.88, Weizhi Avenue, Tengzhou biomedical industrial park, Zaozhuang City, Shandong Province Co-patentee before: SHANGHAI VIWIT PHARMACEUTICAL Co.,Ltd. Patentee before: Weizhi Pharmaceutical Co.,Ltd. |
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CP02 | Change in the address of a patent holder | ||
CP03 | Change of name, title or address |
Address after: No. 88, Weizhi Avenue, biomedical industrial park, Tengzhou City, Zaozhuang City, Shandong Province, 277500 Patentee after: Weizhi Pharmaceutical Co.,Ltd. Patentee after: SHANGHAI VIWIT PHARMACEUTICAL Co.,Ltd. Address before: 277514 No. 88 Weizhi Avenue, Tengzhou Biomedical Industry Base, Zaozhuang City, Shandong Province Patentee before: Weizhi Pharmaceutical Co.,Ltd. Patentee before: SHANGHAI VIWIT PHARMACEUTICAL Co.,Ltd. |
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