CN106414420B - 制备1-茚满醇和1-茚满胺的方法 - Google Patents
制备1-茚满醇和1-茚满胺的方法 Download PDFInfo
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- CN106414420B CN106414420B CN201580005701.7A CN201580005701A CN106414420B CN 106414420 B CN106414420 B CN 106414420B CN 201580005701 A CN201580005701 A CN 201580005701A CN 106414420 B CN106414420 B CN 106414420B
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- XDBBXXBHCWLVLU-UHFFFAOYSA-N CC(C)(C1)C(c(cccc2)c2[Br]=C)OC1=O Chemical compound CC(C)(C1)C(c(cccc2)c2[Br]=C)OC1=O XDBBXXBHCWLVLU-UHFFFAOYSA-N 0.000 description 1
- 0 CC1(C)C([*+]*)c2cc(F)ccc2C1 Chemical compound CC1(C)C([*+]*)c2cc(F)ccc2C1 0.000 description 1
- WNUMETVZOQJKKN-QRIDDKLISA-N O=C1O[C@@H]2c3cc(F)ccc3CC2C1 Chemical compound O=C1O[C@@H]2c3cc(F)ccc3CC2C1 WNUMETVZOQJKKN-QRIDDKLISA-N 0.000 description 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
- C07F7/1872—Preparation; Treatments not provided for in C07F7/20
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J23/00—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00
- B01J23/38—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals
- B01J23/40—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals of the platinum group metals
- B01J23/44—Palladium
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
- C07C209/54—Preparation of compounds containing amino groups bound to a carbon skeleton by rearrangement reactions
- C07C209/58—Preparation of compounds containing amino groups bound to a carbon skeleton by rearrangement reactions from or via amides
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
- C07C211/39—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton
- C07C211/41—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing condensed ring systems
- C07C211/42—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of an unsaturated carbon skeleton containing condensed ring systems with six-membered aromatic rings being part of the condensed ring systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/28—Preparation of carboxylic acid esters by modifying the hydroxylic moiety of the ester, such modification not being an introduction of an ester group
- C07C67/297—Preparation of carboxylic acid esters by modifying the hydroxylic moiety of the ester, such modification not being an introduction of an ester group by splitting-off hydrogen or functional groups; by hydrogenolysis of functional groups
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/02—Esters of acyclic saturated monocarboxylic acids having the carboxyl group bound to an acyclic carbon atom or to hydrogen
- C07C69/22—Esters of acyclic saturated monocarboxylic acids having the carboxyl group bound to an acyclic carbon atom or to hydrogen having three or more carbon atoms in the acid moiety
- C07C69/24—Esters of acyclic saturated monocarboxylic acids having the carboxyl group bound to an acyclic carbon atom or to hydrogen having three or more carbon atoms in the acid moiety esterified with monohydroxylic compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/62—Halogen-containing esters
- C07C69/63—Halogen-containing esters of saturated acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2523/00—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group C07C2521/00
- C07C2523/38—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group C07C2521/00 of noble metals
- C07C2523/40—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group C07C2521/00 of noble metals of the platinum group metals
- C07C2523/44—Palladium
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Catalysts (AREA)
- Indole Compounds (AREA)
- Furan Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP14152790 | 2014-01-28 | ||
| EP14152790.3 | 2014-01-28 | ||
| PCT/EP2015/051344 WO2015113903A1 (de) | 2014-01-28 | 2015-01-23 | Verfahren zur herstellung von 1-indanolen und 1-indanaminen |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN106414420A CN106414420A (zh) | 2017-02-15 |
| CN106414420B true CN106414420B (zh) | 2018-12-14 |
Family
ID=49999830
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN201580005701.7A Active CN106414420B (zh) | 2014-01-28 | 2015-01-23 | 制备1-茚满醇和1-茚满胺的方法 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US9796737B2 (enExample) |
| EP (1) | EP3099671B1 (enExample) |
| JP (1) | JP6475265B2 (enExample) |
| KR (1) | KR102362143B1 (enExample) |
| CN (1) | CN106414420B (enExample) |
| BR (1) | BR112016017513B1 (enExample) |
| DK (1) | DK3099671T3 (enExample) |
| ES (1) | ES2657797T3 (enExample) |
| IL (1) | IL246831B (enExample) |
| MX (1) | MX362690B (enExample) |
| TW (1) | TWI668201B (enExample) |
| WO (1) | WO2015113903A1 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112020023820A2 (pt) * | 2018-05-23 | 2021-04-13 | Bayer Aktiengesellschaft | Processo para produzir derivados de 4-aminoindano substituídos a partir de 2-(hidroxialquil)-anilinas |
| CN109438253B (zh) * | 2018-10-08 | 2021-04-23 | 苏利制药科技江阴有限公司 | 一种合成2-氨基茚的方法 |
| CA3153003C (en) | 2018-11-29 | 2023-10-17 | Bayer Cropscience Lp | Herbicidal compositions for animal grazelands and methods for applying the same |
| CN113797978B (zh) * | 2021-10-12 | 2023-11-07 | 青岛科技大学 | 一类聚三芳基氧膦负载钯/铜双金属催化剂的制备方法及应用 |
| CN121175287A (zh) | 2023-03-29 | 2025-12-19 | 安道麦阿甘有限公司 | 用于制备胺中间体的方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| OA13024A (en) | 2003-02-05 | 2006-11-10 | Bayer Cropscience Gmbh | Amino 1, 3, 5-triazines N-substituted with chiral bicyclic radicals, process for their preparation, compositions thereof and their use as herbicides and plant growth regulators. |
| US7804803B2 (en) * | 2005-07-25 | 2010-09-28 | Honeywell International Inc. | Neighbor based TDMA slot assignment |
| PT2001296E (pt) | 2006-03-29 | 2015-03-02 | Bayer Cropscience Ag | Agentes herbicidas como dispersões que contêm diflufenicano e flurtamona |
| WO2007114213A1 (ja) * | 2006-03-30 | 2007-10-11 | Asahi Kasei Pharma Corporation | 置換二環式環状誘導体及びその用途 |
| KR100929437B1 (ko) * | 2007-08-02 | 2009-12-03 | 포항공과대학교 산학협력단 | 광학 활성을 갖는 아민의 제조방법 |
-
2015
- 2015-01-23 EP EP15701198.2A patent/EP3099671B1/de active Active
- 2015-01-23 MX MX2016009839A patent/MX362690B/es active IP Right Grant
- 2015-01-23 KR KR1020167022941A patent/KR102362143B1/ko active Active
- 2015-01-23 ES ES15701198.2T patent/ES2657797T3/es active Active
- 2015-01-23 CN CN201580005701.7A patent/CN106414420B/zh active Active
- 2015-01-23 WO PCT/EP2015/051344 patent/WO2015113903A1/de not_active Ceased
- 2015-01-23 US US15/114,385 patent/US9796737B2/en active Active
- 2015-01-23 BR BR112016017513-1A patent/BR112016017513B1/pt active IP Right Grant
- 2015-01-23 DK DK15701198.2T patent/DK3099671T3/da active
- 2015-01-23 JP JP2016565561A patent/JP6475265B2/ja active Active
- 2015-01-26 TW TW104102456A patent/TWI668201B/zh active
-
2016
- 2016-07-19 IL IL246831A patent/IL246831B/en active IP Right Grant
Non-Patent Citations (5)
| Title |
|---|
| A catalytic asymmetric approach to C1-chiral 3-methylene-indan-1-ols;Roya Mirabdolbaghi et al.;《Tetrahedron》;20111221;第68卷;1988-1991 * |
| Rapid Catalyst Screening by a Continuous-Flow Microreactor Interfaced with Ultra-High-Pressure Liquid Chromatography;Hui Fang et al.;《J. Org. Chem.》;20100728;第75卷;5619-5626 * |
| Synthesis of 1-Indanols and 1-Indanamines by Intramolecular Palladium(0)-Catalyzed C(sp3)-H Arylation: Impact of Conformational Effects;Simon Janody et al.;《Chem. Eur. J.》;20140728;第20卷;11084-11090 * |
| Synthesis of 3-methyleneindan-1-ol scaffold from modified Baylis–Hillman adduct: tandem Pd-catalyzed 5-exo-trig cyclization and iodide ion-assisted formal d-carbon elimination/decarboxylation;Ko Hoon Kim et al.;《Tetrahedron Letters》;20110826;第52卷;5605-5609 * |
| Synthesis of Polycyclic Molecules by Double C(sp2)-H/C(sp3)-H Arylations with a Single Palladium Catalyst;Cathleen Pierre et al.;《Organic Letters》;20110307;第13卷(第7期);1816-1819 * |
Also Published As
| Publication number | Publication date |
|---|---|
| MX362690B (es) | 2019-02-01 |
| BR112016017513A2 (enExample) | 2017-08-08 |
| EP3099671A1 (de) | 2016-12-07 |
| US20160340370A1 (en) | 2016-11-24 |
| JP6475265B2 (ja) | 2019-02-27 |
| BR112016017513B1 (pt) | 2022-03-03 |
| KR20160113643A (ko) | 2016-09-30 |
| TW201613843A (en) | 2016-04-16 |
| WO2015113903A1 (de) | 2015-08-06 |
| ES2657797T3 (es) | 2018-03-06 |
| IL246831B (en) | 2018-11-29 |
| EP3099671B1 (de) | 2017-12-27 |
| US9796737B2 (en) | 2017-10-24 |
| DK3099671T3 (da) | 2018-01-29 |
| JP2017508783A (ja) | 2017-03-30 |
| KR102362143B1 (ko) | 2022-02-10 |
| MX2016009839A (es) | 2016-10-31 |
| CN106414420A (zh) | 2017-02-15 |
| TWI668201B (zh) | 2019-08-11 |
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