CN103619838B - 作为s1p1受体激动剂的哌啶基单羧酸 - Google Patents
作为s1p1受体激动剂的哌啶基单羧酸 Download PDFInfo
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- CN103619838B CN103619838B CN201280022925.5A CN201280022925A CN103619838B CN 103619838 B CN103619838 B CN 103619838B CN 201280022925 A CN201280022925 A CN 201280022925A CN 103619838 B CN103619838 B CN 103619838B
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Classifications
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Landscapes
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Abstract
Description
Claims (15)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP11305433.2 | 2011-04-12 | ||
EP11305433A EP2511275A1 (en) | 2011-04-12 | 2011-04-12 | Novel piperidinyl monocarboxylic acids as S1P1 receptor agonists |
PCT/EP2012/056470 WO2012140020A1 (en) | 2011-04-12 | 2012-04-10 | Novel piperidinyl monocarboxylic acids as s1p1 receptor agonists |
Publications (2)
Publication Number | Publication Date |
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CN103619838A CN103619838A (zh) | 2014-03-05 |
CN103619838B true CN103619838B (zh) | 2016-08-24 |
Family
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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CN201280022925.5A Active CN103619838B (zh) | 2011-04-12 | 2012-04-10 | 作为s1p1受体激动剂的哌啶基单羧酸 |
Country Status (24)
Country | Link |
---|---|
US (1) | US9266867B2 (zh) |
EP (2) | EP2511275A1 (zh) |
JP (1) | JP6050315B2 (zh) |
KR (1) | KR101854152B1 (zh) |
CN (1) | CN103619838B (zh) |
AU (1) | AU2012241981B2 (zh) |
BR (1) | BR112013026434B1 (zh) |
CA (1) | CA2833180C (zh) |
CO (1) | CO6801772A2 (zh) |
DK (1) | DK2697219T3 (zh) |
EA (1) | EA023638B1 (zh) |
EC (1) | ECSP13012983A (zh) |
ES (1) | ES2544616T3 (zh) |
HU (1) | HUE025443T2 (zh) |
IL (1) | IL228844A (zh) |
MA (1) | MA35305B1 (zh) |
MX (1) | MX342926B (zh) |
PL (1) | PL2697219T3 (zh) |
PT (1) | PT2697219E (zh) |
SG (1) | SG194183A1 (zh) |
TN (1) | TN2013000425A1 (zh) |
UA (1) | UA110822C2 (zh) |
WO (1) | WO2012140020A1 (zh) |
ZA (1) | ZA201307820B (zh) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
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US10662181B2 (en) | 2016-07-13 | 2020-05-26 | Leo Pharma A/S | Heteroaromatic modulators of the retinoid-related orphan receptor gamma |
CN111807954B (zh) * | 2019-04-10 | 2024-04-05 | 广东东阳光药业股份有限公司 | 一种辛波莫德中间体的制备方法 |
CN113332435B (zh) * | 2021-06-18 | 2022-10-18 | 广州中医药大学(广州中医药研究院) | 鞘氨醇-1-磷酸4受体激动剂及其与真武汤联合在制备治疗慢性肾小球肾炎药物中的应用 |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2003105771A2 (en) * | 2002-06-17 | 2003-12-24 | Merck & Co., Inc. | 1-((5-aryl-1,2,4-oxadiazol-3-yl)benzyl)azetidine-3-carboxylates and 1-((5-aryl-1,2,4-oxadiazol-3-yl)benzyl)pyrrolidine-3-carboxylates as edg receptor agonists |
WO2009080730A1 (en) * | 2007-12-21 | 2009-07-02 | Glaxo Group Limited | 1, 2, 4 -oxadiazole compounds for the treatment of autoimmune diseases |
CN101784535A (zh) * | 2007-06-15 | 2010-07-21 | 生物计划公司 | 作为s1p1受体激动剂的新的二羧酸衍生物 |
CN101970420A (zh) * | 2007-10-04 | 2011-02-09 | 默克雪兰诺有限公司 | 噁二唑衍生物 |
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- 2012-04-10 KR KR1020137030008A patent/KR101854152B1/ko active IP Right Grant
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- 2012-04-10 EP EP12714674.4A patent/EP2697219B1/en active Active
- 2012-04-10 ES ES12714674.4T patent/ES2544616T3/es active Active
- 2012-04-10 WO PCT/EP2012/056470 patent/WO2012140020A1/en active Application Filing
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- 2012-04-10 HU HUE12714674A patent/HUE025443T2/en unknown
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