CN103402994B - 作为α7 NACHR调节剂的杂芳基衍生物 - Google Patents

作为α7 NACHR调节剂的杂芳基衍生物 Download PDF

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Publication number
CN103402994B
CN103402994B CN201280010409.0A CN201280010409A CN103402994B CN 103402994 B CN103402994 B CN 103402994B CN 201280010409 A CN201280010409 A CN 201280010409A CN 103402994 B CN103402994 B CN 103402994B
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methyl
benzenesulfonamide
compound
chlorophenyl
propionylthiophen
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CN201280010409.0A
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Chinese (zh)
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CN103402994A (zh
Inventor
N·辛哈
G·贾纳
S·萨科奇达南德
S·P·库哈德
N·P·卡彻
A·K·哈贾尔
A·R·泰尔卡
V·P·帕勒
R·K·坎伯吉
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Lupin Ltd
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Lupin Ltd
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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CN201280010409.0A 2011-02-23 2012-02-22 作为α7 NACHR调节剂的杂芳基衍生物 Expired - Fee Related CN103402994B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
IN242KO2011 2011-02-23
IN242/KOL/2011 2011-02-23
IN1184/KOL/2011 2011-09-09
IN1184KO2011 2011-09-09
PCT/IB2012/050806 WO2012114285A1 (en) 2011-02-23 2012-02-22 Heteroaryl derivatives as alpha7 nachr modulators

Publications (2)

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