CN103328434A - 制备2-氨基苯甲酰胺衍生物的方法 - Google Patents
制备2-氨基苯甲酰胺衍生物的方法 Download PDFInfo
- Publication number
- CN103328434A CN103328434A CN2012800057831A CN201280005783A CN103328434A CN 103328434 A CN103328434 A CN 103328434A CN 2012800057831 A CN2012800057831 A CN 2012800057831A CN 201280005783 A CN201280005783 A CN 201280005783A CN 103328434 A CN103328434 A CN 103328434A
- Authority
- CN
- China
- Prior art keywords
- formula
- compound
- palladium
- ligand
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 *c(cc1C(O*)=O)cc(*)c1N Chemical compound *c(cc1C(O*)=O)cc(*)c1N 0.000 description 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/10—Preparation of carboxylic acid amides from compounds not provided for in groups C07C231/02 - C07C231/08
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
- Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161437280P | 2011-01-28 | 2011-01-28 | |
| US61/437,280 | 2011-01-28 | ||
| PCT/US2012/022899 WO2012103436A1 (en) | 2011-01-28 | 2012-01-27 | Method for preparing 2-aminobenzamide derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN103328434A true CN103328434A (zh) | 2013-09-25 |
Family
ID=45582051
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN2012800057831A Pending CN103328434A (zh) | 2011-01-28 | 2012-01-27 | 制备2-氨基苯甲酰胺衍生物的方法 |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US8871939B2 (enExample) |
| EP (1) | EP2668153B1 (enExample) |
| JP (1) | JP2014511367A (enExample) |
| KR (1) | KR20140006007A (enExample) |
| CN (1) | CN103328434A (enExample) |
| AU (1) | AU2012211165A1 (enExample) |
| BR (1) | BR112013018228A2 (enExample) |
| HU (1) | HUE025309T2 (enExample) |
| IL (1) | IL226892A (enExample) |
| MX (1) | MX2013008560A (enExample) |
| TW (1) | TW201235338A (enExample) |
| WO (1) | WO2012103436A1 (enExample) |
| ZA (1) | ZA201304330B (enExample) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017219768A1 (zh) * | 2016-06-21 | 2017-12-28 | 华东理工大学 | 氯虫苯甲酰胺的多晶型及其制备方法 |
| CN113166095A (zh) * | 2018-12-24 | 2021-07-23 | Upl有限公司 | 用于制备邻氨基苯甲酰胺的方法 |
| CN115417781A (zh) * | 2022-09-30 | 2022-12-02 | 西安凯立新材料股份有限公司 | 一种制备氯虫苯甲酰胺中间体k胺的方法 |
| WO2024251227A1 (zh) * | 2023-06-08 | 2024-12-12 | 上海森辉医药有限公司 | 一种甲酰胺类化合物的制备方法 |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2648308T3 (es) * | 2011-07-08 | 2017-12-29 | Bayer Intellectual Property Gmbh | Procedimiento para la preparación de 2-amino-5-ciano-N,3-dimetilbenzamida |
| EP2812310A1 (de) * | 2012-02-07 | 2014-12-17 | Bayer Intellectual Property GmbH | Verfahren zur herstellung von substituierten anthranilsäure-derivaten |
| TWI678354B (zh) * | 2014-05-29 | 2019-12-01 | 新加坡商艾佛艾姆希農業新加坡有限公司 | 藉空氣氧化製備3-甲基-2-硝基苯甲酸之製程 |
| WO2020117493A1 (en) * | 2018-12-03 | 2020-06-11 | Fmc Corporation | Method for preparing n-phenylpyrazole-1-carboxamides |
| CA3129876A1 (en) | 2019-02-18 | 2020-08-27 | Pi Industries Ltd. | A process for preparing anthranilic diamides and intermediates thereof |
| KR102841700B1 (ko) | 2019-02-22 | 2025-08-01 | 피아이 인더스트리스 엘티디. | 안트라닐산 디아미드 화합물 및 그의 중간체의 합성 방법 |
| EP4143159B1 (en) * | 2020-04-29 | 2024-04-10 | Basf Se | Preparation of aromatic carboxyamides by a palladium-catalyzed carbonylation reaction |
| TW202219046A (zh) * | 2020-07-23 | 2022-05-16 | 美商富曼西公司 | 藉由使用一結晶中間體改善剋安勃製程 |
| CN116670115A (zh) | 2020-09-17 | 2023-08-29 | 皮埃企业有限公司 | 制备邻胺苯甲酸/邻胺苯甲酰胺化合物及其中间产物的方法 |
| AR123593A1 (es) | 2020-09-26 | 2022-12-21 | Pi Industries Ltd | Un proceso para la síntesis de compuestos antranílicos de ácido / amida e intermedios de los mismos |
| WO2024116197A1 (en) * | 2022-11-30 | 2024-06-06 | Natco Pharma Limited | An improved process for the preparation of intermediate of cyantraniliprole |
| WO2025134143A1 (en) | 2023-12-19 | 2025-06-26 | Pi Industries Ltd. | A method for the synthesis of substituted anthranilic amide compounds, intermediates and salts thereof |
| WO2025188963A1 (en) | 2024-03-06 | 2025-09-12 | Fmc Corporation | Metal catalyzed synthesis of 2-aminobenzamide derivatives |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1703417A (zh) * | 2002-10-04 | 2005-11-30 | 纳幕尔杜邦公司 | 邻氨基苯甲酰胺杀虫剂 |
| CN101072767A (zh) * | 2004-12-07 | 2007-11-14 | 杜邦公司 | 制备n-苯基吡唑-1-甲酰胺的方法 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR036872A1 (es) | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| TWI327566B (en) | 2001-08-13 | 2010-07-21 | Du Pont | Novel substituted ihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use |
| CA2454298A1 (en) | 2001-08-13 | 2003-02-27 | Gary David Annis | Substituted 1h-dihydropyrazoles, their preparation and use |
| EP1417176B1 (en) * | 2001-08-16 | 2008-12-17 | E.I. Du Pont De Nemours And Company | Substituted anthranilamides for controlling invertebrate pests |
| JP2004043474A (ja) | 2002-07-05 | 2004-02-12 | Nippon Nohyaku Co Ltd | 2−アミノ安息香酸誘導体及びその製造方法 |
| TWI343376B (en) | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
| SE526014C2 (sv) | 2002-09-11 | 2005-06-14 | Anmedic Ab | En apparat för att försörja en patient med en blandning av bärgas och ett gasformigt anestesimedel |
| TWI367882B (en) | 2003-03-26 | 2012-07-11 | Du Pont | Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates |
| WO2005095327A1 (ja) * | 2004-03-31 | 2005-10-13 | Ajinomoto Co., Inc. | アニリン誘導体 |
| GB0426894D0 (en) | 2004-12-08 | 2005-01-12 | Stylacats Ltd | Process |
| WO2008051533A2 (en) | 2006-10-25 | 2008-05-02 | Takeda Pharmaceutical Company Limited | Benzimidazole compounds |
| TWI431000B (zh) * | 2008-03-05 | 2014-03-21 | Du Pont | 製備2-胺基-5-氰基苯甲酸衍生物之方法 |
| JP5619730B2 (ja) * | 2008-05-27 | 2014-11-05 | ビーエーエスエフ ソシエタス・ヨーロピアBasf Se | 芳香族およびヘテロ芳香族カルボン酸、カルボン酸エステルおよびカルボン酸アミドの製造方法 |
| KR20100092909A (ko) | 2009-02-13 | 2010-08-23 | 주식회사 엘지생명과학 | 잔틴 옥시다제 저해제로서 효과적인 신규 화합물, 그 제조방법 및 그를 함유하는 약제학적 조성물 |
| CN101717395A (zh) * | 2009-12-04 | 2010-06-02 | 南开大学 | 一种氯虫苯甲酰胺农药的合成方法 |
-
2012
- 2012-01-27 AU AU2012211165A patent/AU2012211165A1/en not_active Abandoned
- 2012-01-27 JP JP2013551371A patent/JP2014511367A/ja active Pending
- 2012-01-27 CN CN2012800057831A patent/CN103328434A/zh active Pending
- 2012-01-27 US US13/981,919 patent/US8871939B2/en active Active - Reinstated
- 2012-01-27 BR BR112013018228A patent/BR112013018228A2/pt not_active IP Right Cessation
- 2012-01-27 WO PCT/US2012/022899 patent/WO2012103436A1/en not_active Ceased
- 2012-01-27 HU HUE12703656A patent/HUE025309T2/en unknown
- 2012-01-27 EP EP12703656.4A patent/EP2668153B1/en not_active Not-in-force
- 2012-01-27 KR KR1020137022651A patent/KR20140006007A/ko not_active Withdrawn
- 2012-01-27 MX MX2013008560A patent/MX2013008560A/es not_active Application Discontinuation
- 2012-01-30 TW TW101102830A patent/TW201235338A/zh unknown
-
2013
- 2013-06-12 IL IL226892A patent/IL226892A/en not_active IP Right Cessation
- 2013-06-12 ZA ZA2013/04330A patent/ZA201304330B/en unknown
-
2014
- 2014-09-16 US US14/487,600 patent/US9162973B2/en active Active
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1703417A (zh) * | 2002-10-04 | 2005-11-30 | 纳幕尔杜邦公司 | 邻氨基苯甲酰胺杀虫剂 |
| CN101072767A (zh) * | 2004-12-07 | 2007-11-14 | 杜邦公司 | 制备n-苯基吡唑-1-甲酰胺的方法 |
Non-Patent Citations (3)
| Title |
|---|
| A. SCHOENBERG, ET AL.: "Palladium-Catalyzed Amidation of Aryl, Heterocyclic, and Vinylic Halides", 《J. ORG. CHEM.》, vol. 39, no. 23, 1 November 1974 (1974-11-01), pages 3327 - 3331, XP000673766, DOI: doi:10.1021/jo00937a004 * |
| JENNIFER ALBANEZE-WALKER, ET AL.: "Improved Carbonylation of Heterocyclic Chlorides and Electronically Challenging Aryl Bromides", 《ORG. LETT.》, vol. 6, no. 13, 26 May 2004 (2004-05-26), pages 2097 - 2100 * |
| JOSEPH R. MARTINELLI, ET AL.: "Convenient Method for the Preparation of Weinreb Amides via Pd-Catalyzed Aminocarbonylation of Aryl Bromides at Atmospheric Pressure", 《ORG. LETT.》, vol. 8, no. 21, 21 September 2006 (2006-09-21), pages 4843 - 4846 * |
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017219768A1 (zh) * | 2016-06-21 | 2017-12-28 | 华东理工大学 | 氯虫苯甲酰胺的多晶型及其制备方法 |
| CN107522689A (zh) * | 2016-06-21 | 2017-12-29 | 华东理工大学 | 氯虫苯甲酰胺的多晶型及其制备方法 |
| CN113166095A (zh) * | 2018-12-24 | 2021-07-23 | Upl有限公司 | 用于制备邻氨基苯甲酰胺的方法 |
| CN115417781A (zh) * | 2022-09-30 | 2022-12-02 | 西安凯立新材料股份有限公司 | 一种制备氯虫苯甲酰胺中间体k胺的方法 |
| CN115417781B (zh) * | 2022-09-30 | 2023-08-29 | 西安凯立新材料股份有限公司 | 一种制备氯虫苯甲酰胺中间体k胺的方法 |
| WO2024251227A1 (zh) * | 2023-06-08 | 2024-12-12 | 上海森辉医药有限公司 | 一种甲酰胺类化合物的制备方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2668153B1 (en) | 2015-03-04 |
| BR112013018228A2 (pt) | 2016-11-08 |
| JP2014511367A (ja) | 2014-05-15 |
| US9162973B2 (en) | 2015-10-20 |
| WO2012103436A1 (en) | 2012-08-02 |
| ZA201304330B (en) | 2014-08-27 |
| US8871939B2 (en) | 2014-10-28 |
| US20150005503A1 (en) | 2015-01-01 |
| HUE025309T2 (en) | 2016-01-28 |
| IL226892A (en) | 2015-11-30 |
| EP2668153A1 (en) | 2013-12-04 |
| TW201235338A (en) | 2012-09-01 |
| KR20140006007A (ko) | 2014-01-15 |
| AU2012211165A1 (en) | 2013-07-04 |
| US20130310567A1 (en) | 2013-11-21 |
| MX2013008560A (es) | 2013-08-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C06 | Publication | ||
| PB01 | Publication | ||
| SE01 | Entry into force of request for substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C02 | Deemed withdrawal of patent application after publication (patent law 2001) | ||
| WD01 | Invention patent application deemed withdrawn after publication |
Application publication date: 20130925 |