CN1032690C - 咪唑的制备 - Google Patents
咪唑的制备 Download PDFInfo
- Publication number
- CN1032690C CN1032690C CN93118117A CN93118117A CN1032690C CN 1032690 C CN1032690 C CN 1032690C CN 93118117 A CN93118117 A CN 93118117A CN 93118117 A CN93118117 A CN 93118117A CN 1032690 C CN1032690 C CN 1032690C
- Authority
- CN
- China
- Prior art keywords
- group
- alkyl
- formula
- imidazoles
- integer
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/68—Halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
- Radar Systems Or Details Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP219078/92 | 1992-08-18 | ||
| JP21907892 | 1992-08-18 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN1091130A CN1091130A (zh) | 1994-08-24 |
| CN1032690C true CN1032690C (zh) | 1996-09-04 |
Family
ID=16729919
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN93118117A Expired - Fee Related CN1032690C (zh) | 1992-08-18 | 1993-08-18 | 咪唑的制备 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US5312927A (enExample) |
| EP (1) | EP0585014B1 (enExample) |
| JP (1) | JP3393891B2 (enExample) |
| KR (1) | KR100244831B1 (enExample) |
| CN (1) | CN1032690C (enExample) |
| AT (1) | ATE189890T1 (enExample) |
| CA (1) | CA2104268C (enExample) |
| DE (1) | DE69327890T2 (enExample) |
| DK (1) | DK0585014T3 (enExample) |
| ES (1) | ES2145033T3 (enExample) |
| GR (1) | GR3032807T3 (enExample) |
| HU (1) | HU216973B (enExample) |
| PT (1) | PT585014E (enExample) |
| TW (1) | TW240223B (enExample) |
| ZA (1) | ZA936054B (enExample) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5681956A (en) * | 1990-12-28 | 1997-10-28 | Neurogen Corporation | 4-aryl substituted piperazinylmethyl phenylimidazole derivatives; a new class of dopamine receptor subtype specific ligands |
| US5656762A (en) * | 1990-12-28 | 1997-08-12 | Neurogen Corporation | 4-piperidino-and piperazinomethyl-2-phenylimidazole derivatives, dopamine receptor subtype specific ligands |
| US5633376A (en) * | 1990-12-28 | 1997-05-27 | Neurogen Corporation | Certain aminomethyl phenylimidazole derivatives; and 4-aryl substituted piperazinyl and piperidinylmethyl phenylimidazole derivatives; a new class of dopamine receptor subtype ligands |
| US5646279A (en) * | 1990-12-28 | 1997-07-08 | Neurogen Corporation | Substituted 4-piperazinylmethyl 2-phenylimidazoles; dopamine receptor subtype specific ligands |
| US5362334A (en) * | 1993-12-23 | 1994-11-08 | Macdermid, Incorporated | Composition and process for treatment of metallic surfaces |
| FR2717474B1 (fr) * | 1994-03-15 | 1996-06-21 | Hoechst France | Procédé de préparation d'acétals du formyl-2 imidazole. |
| CA2232467A1 (en) * | 1997-03-20 | 1998-09-20 | Richard A. Glennon | Imidazoles with serotonin receptor binding activity |
| US6503935B1 (en) | 1998-08-07 | 2003-01-07 | Abbott Laboratories | Imidazoles and related compounds as α1A agonists |
| US6166205A (en) * | 1998-09-02 | 2000-12-26 | Neurogen Corporation | 2-Aryl-4-(1-[4-heteroaryl]piperazin-1-yl)methylimidazoles: dopamine . D.sub4 receptor subtype ligands |
| US7108834B2 (en) | 2004-10-14 | 2006-09-19 | Chuan Pan Huang | Device for producing negative ion fragrance |
| HUE060249T2 (hu) | 2008-06-16 | 2023-02-28 | Univ Tennessee Res Found | Vegyületek rák kezelésére |
| US9029408B2 (en) | 2008-06-16 | 2015-05-12 | Gtx, Inc. | Compounds for treatment of cancer |
| US9447049B2 (en) | 2010-03-01 | 2016-09-20 | University Of Tennessee Research Foundation | Compounds for treatment of cancer |
| AU2010347233B2 (en) * | 2010-03-01 | 2015-06-18 | Oncternal Therapeutics, Inc. | Compounds for treatment of cancer |
| CN102199126B (zh) * | 2010-03-25 | 2013-06-05 | 中国石油化工股份有限公司 | 一种二烷基咪唑的制备方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL7017486A (enExample) * | 1969-12-15 | 1971-06-17 | ||
| GB2068362B (en) * | 1980-01-25 | 1983-11-16 | Kodak Ltd | Preparation of imidazoles |
| DE3018458A1 (de) * | 1980-05-14 | 1982-01-21 | Basf Ag, 6700 Ludwigshafen | Verfahren zur herstellung von 4-methylimidazolen |
| YU47834B (sr) * | 1989-08-10 | 1996-01-09 | Schering Agrochemical Limited | Azolni pesticid |
| AU1191292A (en) * | 1991-02-11 | 1992-09-07 | Schering Agrochemicals Limited | Imidazole pesticides |
-
1993
- 1993-08-12 JP JP20052393A patent/JP3393891B2/ja not_active Expired - Fee Related
- 1993-08-13 DK DK93306405T patent/DK0585014T3/da active
- 1993-08-13 EP EP93306405A patent/EP0585014B1/en not_active Expired - Lifetime
- 1993-08-13 AT AT93306405T patent/ATE189890T1/de not_active IP Right Cessation
- 1993-08-13 ES ES93306405T patent/ES2145033T3/es not_active Expired - Lifetime
- 1993-08-13 DE DE69327890T patent/DE69327890T2/de not_active Expired - Fee Related
- 1993-08-13 PT PT93306405T patent/PT585014E/pt unknown
- 1993-08-16 US US08/106,550 patent/US5312927A/en not_active Expired - Fee Related
- 1993-08-17 CA CA002104268A patent/CA2104268C/en not_active Expired - Fee Related
- 1993-08-17 KR KR1019930015913A patent/KR100244831B1/ko not_active Expired - Fee Related
- 1993-08-17 HU HU9302360A patent/HU216973B/hu not_active IP Right Cessation
- 1993-08-18 ZA ZA936054A patent/ZA936054B/xx unknown
- 1993-08-18 TW TW082106649A patent/TW240223B/zh active
- 1993-08-18 CN CN93118117A patent/CN1032690C/zh not_active Expired - Fee Related
-
2000
- 2000-02-29 GR GR20000400512T patent/GR3032807T3/el not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| JP3393891B2 (ja) | 2003-04-07 |
| GR3032807T3 (en) | 2000-06-30 |
| ES2145033T3 (es) | 2000-07-01 |
| HUT65121A (en) | 1994-04-28 |
| ZA936054B (en) | 1995-02-03 |
| EP0585014A3 (en) | 1994-12-14 |
| HU9302360D0 (en) | 1993-11-29 |
| HU216973B (hu) | 1999-10-28 |
| DE69327890T2 (de) | 2000-07-20 |
| US5312927A (en) | 1994-05-17 |
| EP0585014A2 (en) | 1994-03-02 |
| DK0585014T3 (da) | 2000-06-05 |
| PT585014E (pt) | 2000-06-30 |
| KR940003938A (ko) | 1994-03-14 |
| CN1091130A (zh) | 1994-08-24 |
| ATE189890T1 (de) | 2000-03-15 |
| JPH06116242A (ja) | 1994-04-26 |
| TW240223B (enExample) | 1995-02-11 |
| EP0585014B1 (en) | 2000-02-23 |
| CA2104268A1 (en) | 1994-02-19 |
| CA2104268C (en) | 2003-10-28 |
| KR100244831B1 (ko) | 2000-03-02 |
| DE69327890D1 (de) | 2000-03-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C06 | Publication | ||
| PB01 | Publication | ||
| C10 | Entry into substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C14 | Grant of patent or utility model | ||
| GR01 | Patent grant | ||
| C19 | Lapse of patent right due to non-payment of the annual fee | ||
| CF01 | Termination of patent right due to non-payment of annual fee |