CN102869664A - 吡唑并嘧啶类激酶抑制剂 - Google Patents

吡唑并嘧啶类激酶抑制剂 Download PDF

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Publication number
CN102869664A
CN102869664A CN2011800104452A CN201180010445A CN102869664A CN 102869664 A CN102869664 A CN 102869664A CN 2011800104452 A CN2011800104452 A CN 2011800104452A CN 201180010445 A CN201180010445 A CN 201180010445A CN 102869664 A CN102869664 A CN 102869664A
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Chinese (zh)
Inventor
J-M·吉米内斯
L·塞迪默
D·弗雷斯
G·布兰克雷
J·C·戴维斯
A·W·米勒
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Vertex Pharmaceuticals Inc
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Vertex Pharmaceuticals Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P31/04—Antibacterial agents
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    • A61P35/00—Antineoplastic agents
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Psychology (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
CN2011800104452A 2010-01-27 2011-01-26 吡唑并嘧啶类激酶抑制剂 Pending CN102869664A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29866810P 2010-01-27 2010-01-27
US61/298,668 2010-01-27
PCT/US2011/022547 WO2011094290A1 (en) 2010-01-27 2011-01-26 Pyrazolopyrimidine kinase inhibitors

Publications (1)

Publication Number Publication Date
CN102869664A true CN102869664A (zh) 2013-01-09

Family

ID=43661996

Family Applications (1)

Application Number Title Priority Date Filing Date
CN2011800104452A Pending CN102869664A (zh) 2010-01-27 2011-01-26 吡唑并嘧啶类激酶抑制剂

Country Status (8)

Country Link
US (1) US8809335B2 (https=)
EP (1) EP2582702A1 (https=)
JP (1) JP2013518114A (https=)
CN (1) CN102869664A (https=)
AU (1) AU2011209651A1 (https=)
CA (1) CA2787363A1 (https=)
MX (1) MX2012008643A (https=)
WO (1) WO2011094290A1 (https=)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105837574A (zh) * 2015-02-02 2016-08-10 四川大学 N-(3-哌啶基)-芳香胺衍生物及其制备方法和用途
CN113544130A (zh) * 2019-05-31 2021-10-22 四川海思科制药有限公司 一种btk抑制剂环衍生物及其制备方法和药学上的应用

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