CN102725302B - 2＇-氟-6＇-亚甲基碳环核苷和治疗病毒感染的方法 - Google Patents

2＇-氟-6＇-亚甲基碳环核苷和治疗病毒感染的方法 Download PDF

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CN102725302B
CN102725302B CN201080062516.9A CN201080062516A CN102725302B CN 102725302 B CN102725302 B CN 102725302B CN 201080062516 A CN201080062516 A CN 201080062516A CN 102725302 B CN102725302 B CN 102725302B
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functional group
compound
hbv
virus
infection
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CN102725302A (zh
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钟凯楚
王佳宁
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University of Georgia Research Foundation Inc
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    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
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    • C07D473/00—Heterocyclic compounds containing purine ring systems
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    • A61P31/18—Antivirals for RNA viruses for HIV
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
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    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
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    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
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    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
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CN201080062516.9A 2009-11-16 2010-11-16 2＇-氟-6＇-亚甲基碳环核苷和治疗病毒感染的方法 Expired - Fee Related CN102725302B (zh)

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US28134209P 2009-11-16 2009-11-16
US61/281,342 2009-11-16
PCT/US2010/056808 WO2011060408A2 (en) 2009-11-16 2010-11-16 2'-fluoro-6'-methylene carbocyclic nucleosides and methods of treating viral infections

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CN102725302B true CN102725302B (zh) 2016-04-06

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US (1) US8946244B2 (https=)
EP (1) EP2501709A4 (https=)
JP (1) JP5779799B2 (https=)
KR (2) KR101961601B1 (https=)
CN (1) CN102725302B (https=)
AP (1) AP2012006310A0 (https=)
AU (1) AU2010319999B2 (https=)
CA (1) CA2781054A1 (https=)
EA (1) EA201270632A1 (https=)
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MX (1) MX2012005601A (https=)
PH (1) PH12012500963B1 (https=)
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ZA201204356B (en) 2013-02-27
AP2012006310A0 (en) 2012-06-30
CA2781054A1 (en) 2011-05-19
KR101961601B1 (ko) 2019-03-25
KR101840479B1 (ko) 2018-03-20
KR20180014179A (ko) 2018-02-07
EP2501709A4 (en) 2013-11-13
EA201270632A1 (ru) 2013-01-30
IL219748A0 (en) 2012-07-31
JP5779799B2 (ja) 2015-09-16
PH12012500963A1 (en) 2018-05-15
EP2501709A2 (en) 2012-09-26
US8946244B2 (en) 2015-02-03
US20130005677A1 (en) 2013-01-03
AU2010319999B2 (en) 2014-01-16
WO2011060408A3 (en) 2011-10-13
WO2011060408A2 (en) 2011-05-19
PH12012500963B1 (en) 2018-08-10
AU2010319999A1 (en) 2012-06-21
HK1172628A1 (zh) 2013-04-26
JP2013510904A (ja) 2013-03-28
MX2012005601A (es) 2012-08-01
CN102725302A (zh) 2012-10-10
KR20120092153A (ko) 2012-08-20

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