CN102666545B - 作为jak抑制剂的杂环吡唑并嘧啶类似物 - Google Patents

作为jak抑制剂的杂环吡唑并嘧啶类似物 Download PDF

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Publication number
CN102666545B
CN102666545B CN201080058290.5A CN201080058290A CN102666545B CN 102666545 B CN102666545 B CN 102666545B CN 201080058290 A CN201080058290 A CN 201080058290A CN 102666545 B CN102666545 B CN 102666545B
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pyrazolo
methyl
pyrazol
pyrimidin
amine
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CN102666545A (zh
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N·拉姆斯登
R·J·哈里森
S·奥克森福德
K·贝尔
N·皮顿
C·达戈斯廷
C·布萨尔
A·拉特克利夫
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Cellzome Ltd
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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CN201080058290.5A 2009-10-20 2010-10-19 作为jak抑制剂的杂环吡唑并嘧啶类似物 Expired - Fee Related CN102666545B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP09173535 2009-10-20
EP09173535.7 2009-10-20
US37535810P 2010-08-20 2010-08-20
US61/375,358 2010-08-20
PCT/EP2010/065700 WO2011048082A1 (en) 2009-10-20 2010-10-19 Heterocyclyl pyrazolopyrimidine analogues as jak inhibitors

Publications (2)

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CN102666545A CN102666545A (zh) 2012-09-12
CN102666545B true CN102666545B (zh) 2016-04-06

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US (1) US9242987B2 (https=)
EP (1) EP2491039A1 (https=)
JP (1) JP5744887B2 (https=)
KR (1) KR20120102601A (https=)
CN (1) CN102666545B (https=)
AR (1) AR078675A1 (https=)
AU (1) AU2010309882B2 (https=)
BR (1) BR112012009327A2 (https=)
CA (1) CA2775009A1 (https=)
EA (1) EA022120B1 (https=)
IL (1) IL218751A0 (https=)
MX (1) MX2012004020A (https=)
NZ (1) NZ598907A (https=)
TW (1) TW201125867A (https=)
WO (1) WO2011048082A1 (https=)

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