CN102665718B - 可用作pdk1抑制剂的杂环化合物 - Google Patents

可用作pdk1抑制剂的杂环化合物 Download PDF

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Publication number
CN102665718B
CN102665718B CN201080055337.2A CN201080055337A CN102665718B CN 102665718 B CN102665718 B CN 102665718B CN 201080055337 A CN201080055337 A CN 201080055337A CN 102665718 B CN102665718 B CN 102665718B
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ring
nitrogen
optionally substituted
sulfur
oxygen
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Chinese (zh)
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CN102665718A (zh
Inventor
J.阿尔恩特
T.钱
K.古基安
G.库马拉维尔
李文成
林盈翔
D.斯科特
L.孙
J.托马斯
K.范弗洛坦
D.王
L.张
D.厄兰森
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Millennium Pharmaceuticals Inc
Viracta Therapeutics Inc
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Millennium Pharmaceuticals Inc
Sunesis Pharmaceuticals Inc
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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