CN102459235B - 吡嗪基吡唑 - Google Patents

吡嗪基吡唑 Download PDF

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Publication number
CN102459235B
CN102459235B CN201080033587.6A CN201080033587A CN102459235B CN 102459235 B CN102459235 B CN 102459235B CN 201080033587 A CN201080033587 A CN 201080033587A CN 102459235 B CN102459235 B CN 102459235B
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CN
China
Prior art keywords
group
alkyl
spp
amino
base
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CN201080033587.6A
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English (en)
Chinese (zh)
Other versions
CN102459235A (zh
Inventor
H-G·施瓦茨
J·弗拉肯波尔
A·亨赛
S·米其林
S·施奈特尔
R·维尔坦
S·沃纳
A·贝克尔
O·马赛姆
E-M·弗兰肯
A·沃斯特
U·高根斯
P·拉默恩
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer CropScience AG
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Bayer CropScience AG
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Filing date
Publication date
Application filed by Bayer CropScience AG filed Critical Bayer CropScience AG
Publication of CN102459235A publication Critical patent/CN102459235A/zh
Application granted granted Critical
Publication of CN102459235B publication Critical patent/CN102459235B/zh
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
CN201080033587.6A 2009-05-29 2010-05-19 吡嗪基吡唑 Expired - Fee Related CN102459235B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09161568A EP2266973A1 (de) 2009-05-29 2009-05-29 Pyrazinylpyrazole
EP09161568.2 2009-05-29
PCT/EP2010/003060 WO2010136145A1 (de) 2009-05-29 2010-05-19 Pyrazinylpyrazole

Publications (2)

Publication Number Publication Date
CN102459235A CN102459235A (zh) 2012-05-16
CN102459235B true CN102459235B (zh) 2015-03-11

Family

ID=40897591

Family Applications (1)

Application Number Title Priority Date Filing Date
CN201080033587.6A Expired - Fee Related CN102459235B (zh) 2009-05-29 2010-05-19 吡嗪基吡唑

Country Status (21)

Country Link
US (2) US20120190687A1 (es)
EP (2) EP2266973A1 (es)
KR (1) KR101758935B1 (es)
CN (1) CN102459235B (es)
AR (1) AR076798A1 (es)
AU (1) AU2010252346B2 (es)
BR (1) BRPI1012771A2 (es)
CA (1) CA2763498A1 (es)
CO (1) CO6470821A2 (es)
DO (1) DOP2011000366A (es)
EC (1) ECSP11011487A (es)
ES (1) ES2409891T3 (es)
IL (1) IL216337A (es)
MX (1) MX2011012504A (es)
NI (1) NI201100208A (es)
NZ (1) NZ596681A (es)
PE (1) PE20120320A1 (es)
TW (1) TW201107310A (es)
UY (1) UY32659A (es)
WO (1) WO2010136145A1 (es)
ZA (1) ZA201108637B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5823398B2 (ja) * 2009-10-12 2015-11-25 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ 農薬としての新規なアミド類およびチオアミド類
CN103947645B (zh) * 2009-10-12 2016-07-06 拜尔农作物科学股份公司 作为杀虫剂的1-(吡啶-3-基)-吡唑和1-(嘧啶-5-基)-吡唑
WO2011057984A1 (de) 2009-11-11 2011-05-19 Bayer Cropscience Ag Neue diazinyl-pyrazolylverbindungen
KR20130088138A (ko) 2010-06-28 2013-08-07 바이엘 인텔렉쳐 프로퍼티 게엠베하 농약으로서 사용하기 위한 헤테로아릴-치환된 피리딘 화합물
DE102010063691A1 (de) * 2010-12-21 2012-06-21 Bayer Animal Health Gmbh Ektoparasitizide Wirkstoffkombinationen
WO2013076092A1 (en) 2011-11-21 2013-05-30 Basf Se Process for preparing n-substituted 1h-pyrazole-5-carboxylate compounds and derivatives thereof
EA201401213A1 (ru) 2012-05-04 2015-04-30 Басф Се Замещенные пиразолсодержащие соединения и их применение в качестве пестицидов
AU2013326600B2 (en) * 2012-10-02 2017-03-30 Bayer Cropscience Ag Heterocyclic compounds as pesticides
US20150284380A1 (en) * 2012-10-31 2015-10-08 Bayer Cropscience Ag Novel heterocyclic compounds as pest control agents
WO2016174049A1 (en) 2015-04-30 2016-11-03 Bayer Animal Health Gmbh Anti-parasitic combinations including halogen-substituted compounds
US10548316B2 (en) 2015-06-18 2020-02-04 Nippon Soda Co., Ltd. Diarylazole compound and harmful organism control agent
WO2017094790A1 (ja) * 2015-11-30 2017-06-08 北興化学工業株式会社 １，２，３－トリアゾール誘導体および当該誘導体を有効成分とする殺虫・殺ダニ剤
KR102352912B1 (ko) 2015-12-16 2022-01-18 닛뽕소다 가부시키가이샤 아릴아졸 화합물 및 유해 생물 방제제
TWI766916B (zh) 2016-12-19 2022-06-11 日商日本曹達股份有限公司 二芳基吡唑化合物及有害生物防治劑
CN110305115A (zh) * 2019-08-19 2019-10-08 南通大学 一种含1-(6-氯吡嗪-2-基)-3-甲氧基吡唑单元的吡唑肟衍生物的制备和应用
CN115943143A (zh) * 2020-04-29 2023-04-07 拜耳公司 1-吡嗪基吡唑基-3-氧基烷基酸和其衍生物及其用于控制不需要的植物生长的用途

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19544799A1 (de) * 1995-12-01 1997-06-05 Bayer Ag Substituierte 5-Aminopyrazole

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL253320A (es) 1959-07-03
US4101540A (en) * 1975-09-30 1978-07-18 Produits Chimiques Ugine Kuhlmann 3-Trifluoromethyl-4-phenyl-pyrazolium azo dyestuffs
FR2326421A1 (fr) 1975-09-30 1977-04-29 Ugine Kuhlmann Nouveaux trifluoromethyl-3-aryl-4 amino-5 pyrazoles et leur application comme bases diazotables pour la synthese de matieres colorantes
JPH08208620A (ja) 1995-02-03 1996-08-13 Takeda Chem Ind Ltd アミノピラゾール誘導体、その製造法および用途
US6169086B1 (en) * 1997-01-27 2001-01-02 Daiichi Pharmaceutical Co., Ltd. Pyrazole derivatives
EA002101B1 (ru) 1997-01-27 2001-12-24 Дайити Фармасьютикал Ко., Лтд. Производные пиразола
CA2297780A1 (en) 1998-06-10 1999-12-16 Boulder Scientific Company Synthesis of aryl boronic acids
US6518266B1 (en) * 1999-07-22 2003-02-11 3-Dimensional Pharmaceuticals 1- Aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides
US7514464B2 (en) 2003-12-18 2009-04-07 Pfizer Limited Substituted arylpyrazoles
EP1928455A1 (en) 2005-08-31 2008-06-11 Bayer Healthcare, LLC Anilinopyrazole derivatives useful for the treatment of diabetes
WO2007048733A1 (de) 2005-10-28 2007-05-03 Basf Se Verwendung von 5-amino-pyrazolen zur bekämpfung pflanzenpathogener schadpilze, neue 5-amino-pyrazole, verfahren zu ihrer herstellung und sie enthaltende mittel
DE102007003036A1 (de) 2006-12-20 2008-06-26 Bayer Cropscience Ag Pyrimidinylpyrazole
WO2009156090A2 (de) * 2008-06-26 2009-12-30 Bayer Cropscience Aktiengesellschaft Insektizide schwefel-derivatisierte 1-azinylpyrazole
WO2011057984A1 (de) * 2009-11-11 2011-05-19 Bayer Cropscience Ag Neue diazinyl-pyrazolylverbindungen

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19544799A1 (de) * 1995-12-01 1997-06-05 Bayer Ag Substituierte 5-Aminopyrazole

Also Published As

Publication number Publication date
AU2010252346B2 (en) 2015-11-19
MX2011012504A (es) 2011-12-12
EP2435420A1 (de) 2012-04-04
US20110021539A1 (en) 2011-01-27
BRPI1012771A2 (pt) 2016-03-29
AU2010252346A1 (en) 2011-12-22
WO2010136145A1 (de) 2010-12-02
TW201107310A (en) 2011-03-01
ES2409891T3 (es) 2013-06-28
PE20120320A1 (es) 2012-03-30
US20120190687A1 (en) 2012-07-26
UY32659A (es) 2010-12-31
NZ596681A (en) 2015-09-25
IL216337A0 (en) 2012-01-31
ZA201108637B (en) 2013-01-30
KR101758935B1 (ko) 2017-07-17
KR20120061779A (ko) 2012-06-13
EP2266973A1 (de) 2010-12-29
CA2763498A1 (en) 2010-12-02
NI201100208A (es) 2012-08-17
CO6470821A2 (es) 2012-06-29
US8513260B2 (en) 2013-08-20
EP2435420B1 (de) 2013-04-03
ECSP11011487A (es) 2011-12-30
DOP2011000366A (es) 2011-12-15
IL216337A (en) 2015-09-24
AR076798A1 (es) 2011-07-06
CN102459235A (zh) 2012-05-16

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PB01 Publication
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
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GR01 Patent grant
CF01 Termination of patent right due to non-payment of annual fee
CF01 Termination of patent right due to non-payment of annual fee

Granted publication date: 20150311

Termination date: 20180519