CN101945875B - 氮杂吲嗪及其使用方法 - Google Patents

氮杂吲嗪及其使用方法 Download PDF

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Publication number
CN101945875B
CN101945875B CN2008801273742A CN200880127374A CN101945875B CN 101945875 B CN101945875 B CN 101945875B CN 2008801273742 A CN2008801273742 A CN 2008801273742A CN 200880127374 A CN200880127374 A CN 200880127374A CN 101945875 B CN101945875 B CN 101945875B
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China
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alkyl
acid
formula
compound
compounds
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Expired - Fee Related
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CN2008801273742A
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English (en)
Chinese (zh)
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CN101945875A (zh
Inventor
斯蒂芬·普莱斯
罗伯特·希尔德
彼得·赫维特
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Genentech Inc
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Genentech Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CN2008801273742A 2007-12-21 2008-12-19 氮杂吲嗪及其使用方法 Expired - Fee Related CN101945875B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US1594207P 2007-12-21 2007-12-21
US61/015,942 2007-12-21
PCT/US2008/087626 WO2009082687A1 (en) 2007-12-21 2008-12-19 Azaindolizines and methods of use

Publications (2)

Publication Number Publication Date
CN101945875A CN101945875A (zh) 2011-01-12
CN101945875B true CN101945875B (zh) 2013-04-24

Family

ID=40352017

Family Applications (1)

Application Number Title Priority Date Filing Date
CN2008801273742A Expired - Fee Related CN101945875B (zh) 2007-12-21 2008-12-19 氮杂吲嗪及其使用方法

Country Status (12)

Country Link
US (1) US8486963B2 (enExample)
EP (1) EP2220092B1 (enExample)
JP (1) JP5710269B2 (enExample)
KR (1) KR20100099185A (enExample)
CN (1) CN101945875B (enExample)
AU (1) AU2008340247B2 (enExample)
BR (1) BRPI0819505A2 (enExample)
CA (1) CA2708176A1 (enExample)
ES (1) ES2387707T3 (enExample)
IL (1) IL206125A (enExample)
NZ (1) NZ586575A (enExample)
WO (1) WO2009082687A1 (enExample)

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KR20130118612A (ko) * 2012-04-20 2013-10-30 (주)네오믹스 신규한 아미노피리딘 유도체 및 이의 용도
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WO2020106305A1 (en) 2018-11-20 2020-05-28 Nflection Therapeutics, Inc. Thienyl-aniline compounds for treatment of dermal disorders
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Also Published As

Publication number Publication date
KR20100099185A (ko) 2010-09-10
IL206125A0 (en) 2010-11-30
EP2220092B1 (en) 2012-06-06
AU2008340247A1 (en) 2009-07-02
WO2009082687A1 (en) 2009-07-02
JP5710269B2 (ja) 2015-04-30
EP2220092A1 (en) 2010-08-25
ES2387707T3 (es) 2012-09-28
BRPI0819505A2 (pt) 2017-04-04
AU2008340247B2 (en) 2012-11-15
CA2708176A1 (en) 2009-07-02
RU2010130315A (ru) 2012-01-27
CN101945875A (zh) 2011-01-12
US8486963B2 (en) 2013-07-16
US20110142826A1 (en) 2011-06-16
IL206125A (en) 2015-08-31
NZ586575A (en) 2012-03-30
JP2011507896A (ja) 2011-03-10

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Granted publication date: 20130424

Termination date: 20161219