CN101687789A - C型肝炎病毒复制的新颖抑制剂 - Google Patents

C型肝炎病毒复制的新颖抑制剂 Download PDF

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CN101687789A
CN101687789A CN200880010161A CN200880010161A CN101687789A CN 101687789 A CN101687789 A CN 101687789A CN 200880010161 A CN200880010161 A CN 200880010161A CN 200880010161 A CN200880010161 A CN 200880010161A CN 101687789 A CN101687789 A CN 101687789A
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solution
ifn
group
optionally substituted
dose
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Chinese (zh)
Inventor
利奥尼德·拜格尔曼
布拉德·巴克曼
王光义
亚森卡·马图利克-阿达米克
安蒂察·迪米特罗娃·斯托伊切夫瓦
史蒂文·W·安德鲁斯
肖恩·莫里斯·米夏莱克
P.T.·拉维·拉贾格帕兰
安德鲁·M·弗赖尔
因德拉尼·古纳瓦德纳
朱莉娅·哈斯
莉莉·黄
马钱德·R·马杜鲁
张干
卡尔·科森
弗拉基米尔·谢列布里亚内
斯科特·塞韦特
劳伦斯·M·布拉特
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Array Biopharma Inc
Intermune Inc
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Array Biopharma Inc
Intermune Inc
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Publication of CN101687789A publication Critical patent/CN101687789A/zh
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  • Communicable Diseases (AREA)
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  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
CN200880010161A 2007-02-12 2008-02-11 C型肝炎病毒复制的新颖抑制剂 Pending CN101687789A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US88943307P 2007-02-12 2007-02-12
US60/889,433 2007-02-12
PCT/US2008/053617 WO2008100867A2 (en) 2007-02-12 2008-02-11 Novel inhibitors hepatitis c virus replication

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CN101687789A true CN101687789A (zh) 2010-03-31

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US (1) US20090047246A1 (https=)
EP (1) EP2134683A2 (https=)
JP (1) JP2010518125A (https=)
CN (1) CN101687789A (https=)
AU (1) AU2008216382A1 (https=)
CA (1) CA2676906A1 (https=)
MX (1) MX2009008439A (https=)
WO (1) WO2008100867A2 (https=)

Cited By (5)

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CN105348181A (zh) * 2015-12-16 2016-02-24 辽宁工程技术大学 一种2-氨基-5-甲基-6-溴吡啶的制备方法
CN107805244A (zh) * 2017-11-14 2018-03-16 牡丹江医学院 一种用于治疗乙型肝炎的药物及其制备方法
CN110526848A (zh) * 2019-09-04 2019-12-03 青岛农业大学 分子间氢迁移引发环胺β-C(sp3)–H官能化合成β-取代的吡咯烷类化合物的方法
CN110753683A (zh) * 2017-04-11 2020-02-04 赛吉制药有限责任公司 咔唑化合物及其使用方法
TWI784074B (zh) * 2017-10-25 2022-11-21 德商拜耳製藥公司 用於製備苯并噻吩-2-基硼酸酯之方法

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US8198449B2 (en) * 2008-09-11 2012-06-12 Bristol-Myers Squibb Company Compounds for the treatment of hepatitis C
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MX2011010058A (es) * 2009-03-25 2011-10-11 Abbott Lab Compuestos antivirales y usos de los mismos.
GB0906026D0 (en) * 2009-04-07 2009-05-20 Angeletti P Ist Richerche Bio Therapeutic compounds
CN104945420A (zh) 2009-06-29 2015-09-30 因塞特公司 作为pi3k抑制剂的嘧啶酮类
CN102574787B (zh) * 2009-07-30 2014-12-31 新加坡国立大学 具有潜在的抗癌活性的小分子异戊二烯基半胱氨酸羧基甲基转移酶抑制剂
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EP2491033A4 (en) * 2009-10-20 2013-03-13 Eiger Biopharmaceuticals Inc AZAINDAZOLES FOR THE TREATMENT OF FLAVIVIRIDAE VIRUS INFECTION
WO2011075643A1 (en) 2009-12-18 2011-06-23 Incyte Corporation Substituted heteroaryl fused derivatives as pi3k inhibitors
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CN103601683B (zh) * 2010-04-16 2016-03-30 中国科学院上海药物研究所 苯并杂环类化合物及其制备方法和用途
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AR081402A1 (es) 2010-05-17 2012-08-29 Envivo Pharmaceuticals Inc Una forma cristalina de clorhidrato de (r)-7-cloro-n-(quinuclidin-3-il) benzo(b)tiofeno-2-carboxamida monohidrato
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