CN101453988A - 高血糖素样肽1（glp-1）药物制剂 - Google Patents

高血糖素样肽1（glp-1）药物制剂 Download PDF

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Publication number
CN101453988A
CN101453988A CNA200780013424XA CN200780013424A CN101453988A CN 101453988 A CN101453988 A CN 101453988A CN A200780013424X A CNA200780013424X A CN A200780013424XA CN 200780013424 A CN200780013424 A CN 200780013424A CN 101453988 A CN101453988 A CN 101453988A
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China
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glp
fdkp
diketopiperazine
molecule
solution
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Pending
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CNA200780013424XA
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Chinese (zh)
Inventor
斯蒂芬尼·戈恩
大卫·布兰特
柯哈瓦·盖尔伯
马克·金
韦曼·温蒂尔·师特汉姆
凯斯·奥伯格
安德里亚·勒龙-贝
马克·J·豪肯森
玛丽·法瑞斯
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Mannkind Corp
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Mannkind Corp
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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CNA200780013424XA 2006-04-14 2007-04-16 高血糖素样肽1（glp-1）药物制剂 Pending CN101453988A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74488206P 2006-04-14 2006-04-14
US60/744,882 2006-04-14

Related Child Applications (1)

Application Number Title Priority Date Filing Date
CN201410514033.8A Division CN104288756A (zh) 2006-04-14 2007-04-16 高血糖素样肽1(glp-1)药物制剂

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Publication Number Publication Date
CN101453988A true CN101453988A (zh) 2009-06-10

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CNA200780013424XA Pending CN101453988A (zh) 2006-04-14 2007-04-16 高血糖素样肽1（glp-1）药物制剂
CN201410514033.8A Pending CN104288756A (zh) 2006-04-14 2007-04-16 高血糖素样肽1(glp-1)药物制剂

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EP (1) EP2010155A2 (https=)
JP (3) JP5415938B2 (https=)
KR (3) KR101438839B1 (https=)
CN (2) CN101453988A (https=)
AU (1) AU2007238000B2 (https=)
BR (1) BRPI0709964A2 (https=)
CA (1) CA2646400A1 (https=)
HK (1) HK1206241A1 (https=)
MX (1) MX2008013216A (https=)
RU (3) RU2542500C2 (https=)
WO (1) WO2007121411A2 (https=)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN106456707A (zh) * 2014-03-18 2017-02-22 阿佩普蒂科研究和开发有限责任公司 干粉肽药剂
CN115192554A (zh) * 2022-08-08 2022-10-18 浙江仙琚萃泽医药科技有限公司 无抛射剂的含肽吸入溶液剂及其制备方法

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