CN101233132A - 调节trpv3功能的化合物 - Google Patents

调节trpv3功能的化合物 Download PDF

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Publication number
CN101233132A
CN101233132A CNA2006800251060A CN200680025106A CN101233132A CN 101233132 A CN101233132 A CN 101233132A CN A2006800251060 A CNA2006800251060 A CN A2006800251060A CN 200680025106 A CN200680025106 A CN 200680025106A CN 101233132 A CN101233132 A CN 101233132A
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China
Prior art keywords
trpv3
group
sulfonamido
low alkyl
represent
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Pending
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CNA2006800251060A
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Chinese (zh)
Inventor
介弘·A·崇
克里斯托弗·范格
马格达雷那·M·莫兰
丹尼斯·约翰·昂德伍德
甄晓广
艾米·里普卡
曼弗雷德·魏格勒
小威廉·C·卢马
格伦·R·拉森
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Hydra Biosciences LLC
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Hydra Biosciences LLC
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Publication of CN101233132A publication Critical patent/CN101233132A/zh
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CNA2006800251060A 2005-05-09 2006-05-09 调节trpv3功能的化合物 Pending CN101233132A (zh)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US67943805P 2005-05-09 2005-05-09
US67943605P 2005-05-09 2005-05-09
US60/679,438 2005-05-09
US60/679,436 2005-05-09
US70258405P 2005-07-25 2005-07-25
US60/702,584 2005-07-25
PCT/US2006/017995 WO2006122156A2 (en) 2005-05-09 2006-05-09 Compounds for modulating trpv3 function

Publications (1)

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CN101233132A true CN101233132A (zh) 2008-07-30

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CNA2006800251060A Pending CN101233132A (zh) 2005-05-09 2006-05-09 调节trpv3功能的化合物

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US (3) US7803790B2 (https=)
EP (2) EP2392328A1 (https=)
JP (2) JP2008540549A (https=)
CN (1) CN101233132A (https=)
AU (1) AU2006244074B2 (https=)
CA (1) CA2608194A1 (https=)
TW (1) TWI401254B (https=)
WO (1) WO2006122156A2 (https=)

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102747128A (zh) * 2012-05-24 2012-10-24 北京海威磐石生物医药科技有限公司 Trpv3通道蛋白在筛选用于皮肤病治疗或皮肤护理的药物中的应用
CN102802730A (zh) * 2009-06-10 2012-11-28 詹森药业有限公司 可用作trpm8通道调节剂的苯并咪唑衍生物
CN103140476A (zh) * 2010-08-10 2013-06-05 Abbvie公司 新颖的trpv3调节剂
CN103349786A (zh) * 2013-06-04 2013-10-16 北京大学第一医院 一种以trpv3通道蛋白为靶点的用于治疗皮肤瘙痒药物的筛选方法
WO2019192239A1 (zh) * 2018-04-02 2019-10-10 中国药科大学 瞬时受体电位阳离子通道trpv3在研制预防或治疗银屑病药物中的应用
CN116157130A (zh) * 2020-06-29 2023-05-23 勃林格殷格翰国际有限公司 作为trpa1抑制剂的四唑衍生物
CN119930563A (zh) * 2023-12-20 2025-05-06 苏中药业集团股份有限公司 一种瞬时受体电位阳离子通道trpv3抑制剂及其用途
CN120398870A (zh) * 2024-01-31 2025-08-01 深圳晶蛋生物医药科技有限公司 一种苯并吗啉类化合物及其应用

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