FR2707639B1 - Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B. - Google Patents
Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B.Info
- Publication number
- FR2707639B1 FR2707639B1 FR9307982A FR9307982A FR2707639B1 FR 2707639 B1 FR2707639 B1 FR 2707639B1 FR 9307982 A FR9307982 A FR 9307982A FR 9307982 A FR9307982 A FR 9307982A FR 2707639 B1 FR2707639 B1 FR 2707639B1
- Authority
- FR
- France
- Prior art keywords
- 5ht1d
- arylamines
- compounds derived
- indole compounds
- selective ligands
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9307982A FR2707639B1 (fr) | 1993-06-30 | 1993-06-30 | Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B. |
PCT/FR1994/000788 WO1995001334A1 (fr) | 1993-06-30 | 1994-06-29 | Composes indoliques derives d'arylamines comme ligands selectifs des recepteurs 5ht1d et 5ht¿1b? |
AU71883/94A AU7188394A (en) | 1993-06-30 | 1994-06-29 | Arylamine-derived indole compounds as selective 5ht1d and 5ht1b receptor ligands |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9307982A FR2707639B1 (fr) | 1993-06-30 | 1993-06-30 | Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B. |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2707639A1 FR2707639A1 (fr) | 1995-01-20 |
FR2707639B1 true FR2707639B1 (fr) | 1995-10-13 |
Family
ID=9448735
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR9307982A Expired - Fee Related FR2707639B1 (fr) | 1993-06-30 | 1993-06-30 | Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B. |
Country Status (3)
Country | Link |
---|---|
AU (1) | AU7188394A (fr) |
FR (1) | FR2707639B1 (fr) |
WO (1) | WO1995001334A1 (fr) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2724933A1 (fr) * | 1994-09-22 | 1996-03-29 | Pf Medicament | Nouveaux ethers aromatiques derives d'indoles utiles comme medicaments |
FR2731223A1 (fr) * | 1995-03-02 | 1996-09-06 | Pf Medicament | Nouveaux derives bi-tryptaminiques, leur procede de preparation et leur utilisation a titre de medicaments |
US5654431A (en) * | 1996-05-30 | 1997-08-05 | Meng; Qingchang | 5-alkoxy tryptamine derivatives |
FR2763243A1 (fr) * | 1997-05-14 | 1998-11-20 | Pf Medicament | Utilisation d'amines indoliques comme medicaments antithrombotiques |
ATE406371T1 (de) | 2000-11-02 | 2008-09-15 | Us Gov Health & Human Serv | Wirkstoffe für die verminderung von amyloid precursor protein und die behandlung von schwachsinn, und deren verfahren der verwendung |
AU2006244074B2 (en) | 2005-05-09 | 2012-12-13 | Hydra Biosciences, Inc. | Compounds for modulating TRPV3 function |
US8916550B2 (en) | 2005-05-09 | 2014-12-23 | Hydra Biosciences, Inc. | Compounds for modulating TRPV3 function |
US7998980B2 (en) | 2006-09-15 | 2011-08-16 | Hydra Biosciences, Inc. | Compounds for modulating TRPV3 function |
WO2020045982A1 (fr) * | 2018-08-29 | 2020-03-05 | 숙명여자대학교산학협력단 | DÉRIVÉ D'INDOLE SUBSTITUÉ, SON PROCÉDÉ DE PRÉPARATION, ET COMPOSITION PHARMACEUTIQUE LE COMPRENANT EN TANT QUE COMPOSANT ACTIF POUR PRÉVENIR OU TRAITER DES MALADIES ASSOCIÉES À PPARα, PPARγ ET PPARδ |
EP4096661A4 (fr) | 2020-01-29 | 2024-03-06 | Kamari Pharma Ltd. | Composés et compositions pour leur utilisation dans le traitement de troubles cutanés |
US20230219889A1 (en) | 2020-05-19 | 2023-07-13 | Cybin Irl Limited | Deuterated tryptamine derivatives and methods of use |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8431426D0 (en) * | 1984-12-13 | 1985-01-23 | Glaxo Group Ltd | Chemical compounds |
GB8600397D0 (en) * | 1986-01-08 | 1986-02-12 | Glaxo Group Ltd | Chemical compounds |
GB8614287D0 (en) * | 1986-06-12 | 1986-07-16 | Glaxo Group Ltd | Chemical compounds |
GB9103770D0 (en) * | 1991-02-22 | 1991-04-10 | Glaxo Group Ltd | Chemical compounds |
-
1993
- 1993-06-30 FR FR9307982A patent/FR2707639B1/fr not_active Expired - Fee Related
-
1994
- 1994-06-29 WO PCT/FR1994/000788 patent/WO1995001334A1/fr active Application Filing
- 1994-06-29 AU AU71883/94A patent/AU7188394A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
AU7188394A (en) | 1995-01-24 |
FR2707639A1 (fr) | 1995-01-20 |
WO1995001334A1 (fr) | 1995-01-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |