FR2707639B1 - Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B. - Google Patents

Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B.

Info

Publication number
FR2707639B1
FR2707639B1 FR9307982A FR9307982A FR2707639B1 FR 2707639 B1 FR2707639 B1 FR 2707639B1 FR 9307982 A FR9307982 A FR 9307982A FR 9307982 A FR9307982 A FR 9307982A FR 2707639 B1 FR2707639 B1 FR 2707639B1
Authority
FR
France
Prior art keywords
5ht1d
arylamines
compounds derived
indole compounds
selective ligands
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9307982A
Other languages
English (en)
Other versions
FR2707639A1 (fr
Inventor
Halazy Serge
Perez Michel
Briley Michael
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pierre Fabre Medicament SA
Original Assignee
Pierre Fabre Medicament SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pierre Fabre Medicament SA filed Critical Pierre Fabre Medicament SA
Priority to FR9307982A priority Critical patent/FR2707639B1/fr
Priority to PCT/FR1994/000788 priority patent/WO1995001334A1/fr
Priority to AU71883/94A priority patent/AU7188394A/en
Publication of FR2707639A1 publication Critical patent/FR2707639A1/fr
Application granted granted Critical
Publication of FR2707639B1 publication Critical patent/FR2707639B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16Tryptamines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR9307982A 1993-06-30 1993-06-30 Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B. Expired - Fee Related FR2707639B1 (fr)

Priority Applications (3)

Application Number Priority Date Filing Date Title
FR9307982A FR2707639B1 (fr) 1993-06-30 1993-06-30 Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B.
PCT/FR1994/000788 WO1995001334A1 (fr) 1993-06-30 1994-06-29 Composes indoliques derives d'arylamines comme ligands selectifs des recepteurs 5ht1d et 5ht¿1b?
AU71883/94A AU7188394A (en) 1993-06-30 1994-06-29 Arylamine-derived indole compounds as selective 5ht1d and 5ht1b receptor ligands

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9307982A FR2707639B1 (fr) 1993-06-30 1993-06-30 Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B.

Publications (2)

Publication Number Publication Date
FR2707639A1 FR2707639A1 (fr) 1995-01-20
FR2707639B1 true FR2707639B1 (fr) 1995-10-13

Family

ID=9448735

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9307982A Expired - Fee Related FR2707639B1 (fr) 1993-06-30 1993-06-30 Nouveaux composés indoliques dérivés d'arylamines comme ligands sélectifs des récepteurs 5HT1D et 5HT1B.

Country Status (3)

Country Link
AU (1) AU7188394A (fr)
FR (1) FR2707639B1 (fr)
WO (1) WO1995001334A1 (fr)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2724933A1 (fr) * 1994-09-22 1996-03-29 Pf Medicament Nouveaux ethers aromatiques derives d'indoles utiles comme medicaments
FR2731223A1 (fr) * 1995-03-02 1996-09-06 Pf Medicament Nouveaux derives bi-tryptaminiques, leur procede de preparation et leur utilisation a titre de medicaments
US5654431A (en) * 1996-05-30 1997-08-05 Meng; Qingchang 5-alkoxy tryptamine derivatives
FR2763243A1 (fr) * 1997-05-14 1998-11-20 Pf Medicament Utilisation d'amines indoliques comme medicaments antithrombotiques
ATE406371T1 (de) 2000-11-02 2008-09-15 Us Gov Health & Human Serv Wirkstoffe für die verminderung von amyloid precursor protein und die behandlung von schwachsinn, und deren verfahren der verwendung
AU2006244074B2 (en) 2005-05-09 2012-12-13 Hydra Biosciences, Inc. Compounds for modulating TRPV3 function
US8916550B2 (en) 2005-05-09 2014-12-23 Hydra Biosciences, Inc. Compounds for modulating TRPV3 function
US7998980B2 (en) 2006-09-15 2011-08-16 Hydra Biosciences, Inc. Compounds for modulating TRPV3 function
WO2020045982A1 (fr) * 2018-08-29 2020-03-05 숙명여자대학교산학협력단 DÉRIVÉ D'INDOLE SUBSTITUÉ, SON PROCÉDÉ DE PRÉPARATION, ET COMPOSITION PHARMACEUTIQUE LE COMPRENANT EN TANT QUE COMPOSANT ACTIF POUR PRÉVENIR OU TRAITER DES MALADIES ASSOCIÉES À PPARα, PPARγ ET PPARδ
EP4096661A4 (fr) 2020-01-29 2024-03-06 Kamari Pharma Ltd. Composés et compositions pour leur utilisation dans le traitement de troubles cutanés
US20230219889A1 (en) 2020-05-19 2023-07-13 Cybin Irl Limited Deuterated tryptamine derivatives and methods of use

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8431426D0 (en) * 1984-12-13 1985-01-23 Glaxo Group Ltd Chemical compounds
GB8600397D0 (en) * 1986-01-08 1986-02-12 Glaxo Group Ltd Chemical compounds
GB8614287D0 (en) * 1986-06-12 1986-07-16 Glaxo Group Ltd Chemical compounds
GB9103770D0 (en) * 1991-02-22 1991-04-10 Glaxo Group Ltd Chemical compounds

Also Published As

Publication number Publication date
AU7188394A (en) 1995-01-24
FR2707639A1 (fr) 1995-01-20
WO1995001334A1 (fr) 1995-01-12

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