CN101048387B - 苯基2-嘧啶酮及其新的中间体的制备方法 - Google Patents

苯基2-嘧啶酮及其新的中间体的制备方法 Download PDF

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Publication number
CN101048387B
CN101048387B CN2005800373256A CN200580037325A CN101048387B CN 101048387 B CN101048387 B CN 101048387B CN 2005800373256 A CN2005800373256 A CN 2005800373256A CN 200580037325 A CN200580037325 A CN 200580037325A CN 101048387 B CN101048387 B CN 101048387B
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CN
China
Prior art keywords
compound
formula
hydrogen peroxide
salt
preparation
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Expired - Lifetime
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CN2005800373256A
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English (en)
Chinese (zh)
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CN101048387A (zh
Inventor
荒木恒一
佐藤美孝
M·J·福特
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Bayer CropScience AG
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Bayer CropScience AG
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CN2005800373256A 2004-10-29 2005-10-28 苯基2-嘧啶酮及其新的中间体的制备方法 Expired - Lifetime CN101048387B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP317222/2004 2004-10-29
JP2004317222A JP2006124347A (ja) 2004-10-29 2004-10-29 フェニル２−ピリミジニルケトン類の新規製造方法及びその新規中間体
PCT/EP2005/011531 WO2006045612A1 (en) 2004-10-29 2005-10-28 Process for the preparation of phenyl 2-pyrimidinyl ketones and their novel intermediates

Publications (2)

Publication Number Publication Date
CN101048387A CN101048387A (zh) 2007-10-03
CN101048387B true CN101048387B (zh) 2010-05-05

Family

ID=35447955

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CN2005800373256A Expired - Lifetime CN101048387B (zh) 2004-10-29 2005-10-28 苯基2-嘧啶酮及其新的中间体的制备方法

Country Status (12)

Country Link
US (1) US7772395B2 (enExample)
EP (1) EP1807401B1 (enExample)
JP (2) JP2006124347A (enExample)
KR (1) KR101318092B1 (enExample)
CN (1) CN101048387B (enExample)
AT (1) ATE473213T1 (enExample)
BR (1) BRPI0517388B1 (enExample)
DE (1) DE602005022213D1 (enExample)
DK (1) DK1807401T3 (enExample)
IL (1) IL182557A0 (enExample)
MX (1) MX2007005171A (enExample)
WO (1) WO2006045612A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7700076B2 (en) * 2002-10-25 2010-04-20 Foamix, Ltd. Penetrating pharmaceutical foam
AT515384B1 (de) * 2014-02-05 2016-04-15 Dietmar Dr Sonnleitner Vorverbundene mehrschichtige Folie zur Abdeckung einer Knochendefektstelle
AT515117B1 (de) * 2014-04-15 2015-06-15 Dietmar Dr Sonnleitner Zahnimplantatsystem

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040034251A1 (en) * 2000-10-17 2004-02-19 Hidetaka Hiyoshi Process for production of substituted aniline compound

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19521355A1 (de) * 1995-06-12 1996-12-19 Hoechst Schering Agrevo Gmbh Sulfonamide, Verfahren zu deren Herstellung und ihre Verwendung als Herbizide und Pflanzenwachstumsregulatoren
JP3632947B2 (ja) * 1998-07-29 2005-03-30 クミアイ化学工業株式会社 ジフルオロメタンスルホニルアニリド誘導体、その製造方法及びそれを有効成分とする除草剤
ES2209466T3 (es) * 1998-07-29 2004-06-16 Ihara Chemical Industry Co., Ltd. Derivados de difluormetanosulfonilanilida, procedimiento para su preparacion y herbicidas que contienen tales derivados como ingrediente activo.

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040034251A1 (en) * 2000-10-17 2004-02-19 Hidetaka Hiyoshi Process for production of substituted aniline compound

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
BONESI,TORRIANI,MELLA,ALBINI.The photooxygenation of Benzyl,Heteroarylmethyl, and allylsulfides.EUR.J.ORG.CHEM.7.1999,71723-1728. *
mondal, ejabul et al.a useful and environmentally begin synthetic protocol fordethiolization by employing vanadium pentoxide catalyzedoxidation of ammonium bromide by hydrogen peroxide.chemistry letters11.1999,111158-1159. *

Also Published As

Publication number Publication date
ATE473213T1 (de) 2010-07-15
KR101318092B1 (ko) 2013-10-14
DE602005022213D1 (de) 2010-08-19
WO2006045612A1 (en) 2006-05-04
IL182557A0 (en) 2007-09-20
DK1807401T3 (da) 2010-10-18
JP4879907B2 (ja) 2012-02-22
BRPI0517388A (pt) 2008-10-07
US20080004444A1 (en) 2008-01-03
CN101048387A (zh) 2007-10-03
US7772395B2 (en) 2010-08-10
MX2007005171A (es) 2007-06-22
BRPI0517388B1 (pt) 2013-12-24
EP1807401B1 (en) 2010-07-07
KR20070070200A (ko) 2007-07-03
JP2006124347A (ja) 2006-05-18
JP2008517967A (ja) 2008-05-29
EP1807401A1 (en) 2007-07-18

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