CN100340548C - 新型芳杂烷基胺衍生物 - Google Patents
新型芳杂烷基胺衍生物 Download PDFInfo
- Publication number
- CN100340548C CN100340548C CNB028096185A CN02809618A CN100340548C CN 100340548 C CN100340548 C CN 100340548C CN B028096185 A CNB028096185 A CN B028096185A CN 02809618 A CN02809618 A CN 02809618A CN 100340548 C CN100340548 C CN 100340548C
- Authority
- CN
- China
- Prior art keywords
- amino
- thio
- hydroxy
- pyridinecarbonitrile
- phenylbutyl
- Prior art date
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- C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
- C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
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- C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
- C07C217/54—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
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- C—CHEMISTRY; METALLURGY
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- Health & Medical Sciences (AREA)
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- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Rheumatology (AREA)
- Ophthalmology & Optometry (AREA)
- Psychiatry (AREA)
- Physical Education & Sports Medicine (AREA)
- Psychology (AREA)
- Oncology (AREA)
- Immunology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Addiction (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Communicable Diseases (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE01016179 | 2001-05-08 | ||
| SE0101617A SE0101617D0 (sv) | 2001-05-08 | 2001-05-08 | Novel compounds |
| SE0103271A SE0103271D0 (sv) | 2001-09-28 | 2001-09-28 | Novel compounds |
| SE01032713 | 2001-09-28 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN1630637A CN1630637A (zh) | 2005-06-22 |
| CN100340548C true CN100340548C (zh) | 2007-10-03 |
Family
ID=26655458
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB028096185A Expired - Fee Related CN100340548C (zh) | 2001-05-08 | 2002-05-06 | 新型芳杂烷基胺衍生物 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20040242871A1 (enExample) |
| EP (1) | EP1572655A2 (enExample) |
| JP (1) | JP2005506308A (enExample) |
| KR (1) | KR20030096361A (enExample) |
| CN (1) | CN100340548C (enExample) |
| AR (1) | AR035700A1 (enExample) |
| AU (1) | AU2002306039B2 (enExample) |
| BR (1) | BR0209518A (enExample) |
| CA (1) | CA2446120A1 (enExample) |
| IL (1) | IL158388A0 (enExample) |
| MX (1) | MXPA03010142A (enExample) |
| NO (1) | NO20034970D0 (enExample) |
| NZ (1) | NZ529107A (enExample) |
| TW (1) | TWI278450B (enExample) |
| WO (1) | WO2002090332A2 (enExample) |
Families Citing this family (29)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0004152D0 (en) | 2000-02-23 | 2000-04-12 | Astrazeneca Uk Ltd | Novel compounds |
| SE0102640D0 (sv) | 2001-07-31 | 2001-07-31 | Astrazeneca Ab | Novel compounds |
| SE0203304D0 (sv) * | 2002-11-07 | 2002-11-07 | Astrazeneca Ab | Novel Coumpounds |
| WO2005080320A1 (en) | 2004-02-13 | 2005-09-01 | Warner-Lambert Company Llc | Androgen receptor modulators |
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| EA024845B1 (ru) | 2011-07-26 | 2016-10-31 | Бёрингер Ингельхайм Интернациональ Гмбх | Замещенные хинолины и их применение в качестве лекарственных средств |
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2002
- 2002-04-30 AR ARP020101589A patent/AR035700A1/es not_active Application Discontinuation
- 2002-05-06 BR BR0209518-1A patent/BR0209518A/pt not_active IP Right Cessation
- 2002-05-06 TW TW091109347A patent/TWI278450B/zh not_active IP Right Cessation
- 2002-05-06 EP EP02733658A patent/EP1572655A2/en not_active Withdrawn
- 2002-05-06 MX MXPA03010142A patent/MXPA03010142A/es not_active Application Discontinuation
- 2002-05-06 NZ NZ529107A patent/NZ529107A/en unknown
- 2002-05-06 CN CNB028096185A patent/CN100340548C/zh not_active Expired - Fee Related
- 2002-05-06 WO PCT/SE2002/000876 patent/WO2002090332A2/en not_active Ceased
- 2002-05-06 IL IL15838802A patent/IL158388A0/xx unknown
- 2002-05-06 KR KR10-2003-7014492A patent/KR20030096361A/ko not_active Ceased
- 2002-05-06 CA CA002446120A patent/CA2446120A1/en not_active Abandoned
- 2002-05-06 JP JP2002587412A patent/JP2005506308A/ja active Pending
- 2002-05-06 US US10/476,958 patent/US20040242871A1/en not_active Abandoned
- 2002-05-06 AU AU2002306039A patent/AU2002306039B2/en not_active Expired - Fee Related
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2003
- 2003-11-07 NO NO20034970A patent/NO20034970D0/no not_active Application Discontinuation
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| WO1999018960A1 (en) * | 1997-10-10 | 1999-04-22 | Astrazeneca Uk Limited | Novel combination |
| WO2000027842A1 (en) * | 1998-11-05 | 2000-05-18 | Astrazeneca Ab | Compounds |
Also Published As
| Publication number | Publication date |
|---|---|
| KR20030096361A (ko) | 2003-12-24 |
| WO2002090332A3 (en) | 2007-11-01 |
| MXPA03010142A (es) | 2004-03-10 |
| AR035700A1 (es) | 2004-06-23 |
| WO2002090332A2 (en) | 2002-11-14 |
| BR0209518A (pt) | 2004-07-13 |
| NZ529107A (en) | 2006-10-27 |
| IL158388A0 (en) | 2004-05-12 |
| AU2002306039B2 (en) | 2008-05-29 |
| TWI278450B (en) | 2007-04-11 |
| CN1630637A (zh) | 2005-06-22 |
| EP1572655A2 (en) | 2005-09-14 |
| US20040242871A1 (en) | 2004-12-02 |
| JP2005506308A (ja) | 2005-03-03 |
| CA2446120A1 (en) | 2002-11-14 |
| NO20034970D0 (no) | 2003-11-07 |
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