MXPA03010142A - Nuevos derivados de arilheteroalquilamina. - Google Patents

Nuevos derivados de arilheteroalquilamina.

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Publication number
MXPA03010142A
MXPA03010142A MXPA03010142A MXPA03010142A MXPA03010142A MX PA03010142 A MXPA03010142 A MX PA03010142A MX PA03010142 A MXPA03010142 A MX PA03010142A MX PA03010142 A MXPA03010142 A MX PA03010142A MX PA03010142 A MXPA03010142 A MX PA03010142A
Authority
MX
Mexico
Prior art keywords
arylheteroalkylamine
derivatives
novel
compounds
racemates
Prior art date
Application number
MXPA03010142A
Other languages
English (en)
Inventor
Tim Brikinshaw
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE0101617A external-priority patent/SE0101617D0/xx
Priority claimed from SE0103271A external-priority patent/SE0103271D0/xx
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of MXPA03010142A publication Critical patent/MXPA03010142A/es

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    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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Abstract

La presente invencion proporciona compuestos novedosos de la formula (I) (Ver Formula) en donde R1, R2, R3, R4, R5, R6, T, U, X, Y, V y W son como se definieron en la especificacion, y las sales de los mismos farmaceuticamente aceptables, y los enantiomeros y racematos de los mismos; junto con procesos para su preparacion, composiciones que los contienen y su uso en terapia. Los compuestos son inhibidores de la oxido nitrico sintasa y son por esto particularmente utiles en el tratamiento o profilaxis de la enfermedad inflamatoria y el dolor.
MXPA03010142A 2001-05-08 2002-05-06 Nuevos derivados de arilheteroalquilamina. MXPA03010142A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0101617A SE0101617D0 (sv) 2001-05-08 2001-05-08 Novel compounds
SE0103271A SE0103271D0 (sv) 2001-09-28 2001-09-28 Novel compounds
PCT/SE2002/000876 WO2002090332A2 (en) 2001-05-08 2002-05-06 Novel aeylheteroalkylaminε derivatives

Publications (1)

Publication Number Publication Date
MXPA03010142A true MXPA03010142A (es) 2004-03-10

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MXPA03010142A MXPA03010142A (es) 2001-05-08 2002-05-06 Nuevos derivados de arilheteroalquilamina.

Country Status (15)

Country Link
US (1) US20040242871A1 (es)
EP (1) EP1572655A2 (es)
JP (1) JP2005506308A (es)
KR (1) KR20030096361A (es)
CN (1) CN100340548C (es)
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IL158388A0 (en) 2004-05-12
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