CL2018000151A1 - Procesos mejorados para la preparación de compuestos de 1-aril-5-alquil pirazol (divisional de solicitud 201402825) - Google Patents
Procesos mejorados para la preparación de compuestos de 1-aril-5-alquil pirazol (divisional de solicitud 201402825)Info
- Publication number
- CL2018000151A1 CL2018000151A1 CL2018000151A CL2018000151A CL2018000151A1 CL 2018000151 A1 CL2018000151 A1 CL 2018000151A1 CL 2018000151 A CL2018000151 A CL 2018000151A CL 2018000151 A CL2018000151 A CL 2018000151A CL 2018000151 A1 CL2018000151 A1 CL 2018000151A1
- Authority
- CL
- Chile
- Prior art keywords
- preparation
- aryl
- pyrazole compounds
- improved processes
- alkyl pyrazole
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
Abstract
<p>PROCESO MEJORADO PARA LA PREPARACIÓN DE COMPUESTOS DE 1-ARIL PIRAZOL DE FÓRMULA (1) Y (IB), QUE ESTÁN SUSTITUIDOS EN LA POSICIÓN 5 DEL ANILLO PIRAZOL CON UN GRUPO FUNCIONAL UNIDO A CARBONO. EL PROCESO DESCRITO ES EFICAZ Y CON CAPACIDAD DE ESCALADO Y NO UTILIZA REACTIVOS DE HALURO DE SULFENILO PELIGROSOS.</p>
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261635969P | 2012-04-20 | 2012-04-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2018000151A1 true CL2018000151A1 (es) | 2018-05-18 |
Family
ID=48237288
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2014002825A CL2014002825A1 (es) | 2012-04-20 | 2014-10-20 | Procesos para la preparación de un compuesto de 1-aril-5-alquil pirazol |
CL2018000151A CL2018000151A1 (es) | 2012-04-20 | 2018-01-18 | Procesos mejorados para la preparación de compuestos de 1-aril-5-alquil pirazol (divisional de solicitud 201402825) |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2014002825A CL2014002825A1 (es) | 2012-04-20 | 2014-10-20 | Procesos para la preparación de un compuesto de 1-aril-5-alquil pirazol |
Country Status (23)
Country | Link |
---|---|
US (2) | US8937185B2 (es) |
EP (2) | EP2852577B1 (es) |
JP (2) | JP6197192B2 (es) |
KR (2) | KR102099547B1 (es) |
CN (2) | CN104334534B (es) |
AR (2) | AR090773A1 (es) |
AU (2) | AU2013248984B2 (es) |
BR (1) | BR112014026052A8 (es) |
CA (2) | CA3045419A1 (es) |
CL (2) | CL2014002825A1 (es) |
CO (1) | CO7141468A2 (es) |
EA (2) | EA028539B9 (es) |
ES (1) | ES2626167T3 (es) |
IL (3) | IL235108A (es) |
MX (1) | MX344802B (es) |
MY (2) | MY177999A (es) |
NZ (2) | NZ701406A (es) |
PH (1) | PH12014502346A1 (es) |
SG (2) | SG11201406734TA (es) |
TW (1) | TWI579274B (es) |
UA (1) | UA116629C2 (es) |
WO (1) | WO2013159094A2 (es) |
ZA (1) | ZA201407603B (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2019021059A1 (en) | 2017-07-28 | 2019-01-31 | Novartis Ag | INDOLE DERIVATIVES AND USES THEREOF |
CN111094278B (zh) | 2017-09-13 | 2023-07-14 | 诺华股份有限公司 | 二苯基衍生物及其用途 |
CN115124471B (zh) * | 2021-03-24 | 2024-02-13 | 中国工程物理研究院化工材料研究所 | 一类具有高能和低熔点特性的吡唑环类炸药及其合成方法 |
CN115353490A (zh) * | 2022-09-26 | 2022-11-18 | 安徽美诺华药物化学有限公司 | 一种氟虫腈的纯化工艺 |
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GB2136427B (en) | 1983-03-09 | 1986-07-09 | May & Baker Ltd | Herbicidal n-pyridylpyrazole derivatives |
DE3402308A1 (de) | 1984-01-24 | 1985-08-01 | Bayer Ag, 5090 Leverkusen | Herbizide mittel auf basis von pyrazolderivaten |
DE3602728A1 (de) | 1985-05-17 | 1986-11-20 | Bayer Ag, 51373 Leverkusen | Schaedlingsbekaempfungsmittel auf basis von pyrazolderivaten |
DE3520330A1 (de) | 1985-06-07 | 1986-12-11 | Bayer Ag, 5090 Leverkusen | 5-amino-1-pyridyl-pyrazole |
DE3617977A1 (de) | 1985-12-05 | 1987-06-11 | Bayer Ag | 5-dichloracetamido-4-nitro-1-aryl-pyrazole |
GB8531485D0 (en) | 1985-12-20 | 1986-02-05 | May & Baker Ltd | Compositions of matter |
US6372774B1 (en) | 1985-12-20 | 2002-04-16 | Rhone-Poulenc Agriculture Ltd. | Derivatives of N-phenylpyrazoles |
GB8713768D0 (en) | 1987-06-12 | 1987-07-15 | May & Baker Ltd | Compositions of matter |
US5232940A (en) | 1985-12-20 | 1993-08-03 | Hatton Leslie R | Derivatives of N-phenylpyrazoles |
US5547974A (en) | 1985-12-20 | 1996-08-20 | Rhone-Poulenc Agriculture Ltd. | Derivatives of N-phenylpyrazoles |
DE3600287A1 (de) | 1986-01-08 | 1987-07-16 | Bayer Ag | 1-arylpyrazole |
DE3628892A1 (de) * | 1986-08-26 | 1988-03-10 | Bayer Ag | Substituierte 1-aryl-3-tert.-butyl-pyrazole |
SE8802173D0 (sv) | 1988-06-10 | 1988-06-10 | Astra Ab | Pyrimidine derivatives |
GB8816915D0 (en) | 1988-07-15 | 1988-08-17 | May & Baker Ltd | New compositions of matter |
CA2004776C (fr) | 1988-12-13 | 2000-04-25 | Claude Wakselman | Procede de preparation de perfluoroalkylthioethers |
US4918085A (en) | 1989-03-02 | 1990-04-17 | Rhone-Poulenc Ag Company | Pesticidal 3-cyano-5-alkoxy-1-arylpyrazoles, compositions and use |
DE4003371A1 (de) | 1990-02-05 | 1991-08-08 | Richard Herbst | Verfahren zum entformen eines formteils sowie vorrichtung zur durchfuehrung des verfahrens |
CA2036147A1 (en) | 1990-06-29 | 1991-12-30 | Hiroki Tomioka | A 1-pyridylimidazole derivative and its production and use |
NO179282C (no) | 1991-01-18 | 1996-09-11 | Rhone Poulenc Agrochimie | Nye 1-(2-pyridyl)pyrazolforbindelser til kontroll av skadeinsekter |
US5246255A (en) | 1991-06-24 | 1993-09-21 | Forbes Christopher B | Repair flange |
GB9120641D0 (en) | 1991-09-27 | 1991-11-06 | Ici Plc | Heterocyclic compounds |
DE4343832A1 (de) * | 1993-12-22 | 1995-06-29 | Bayer Ag | Substituierte 1-Arylpyrazole |
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US20040220170A1 (en) | 2003-05-01 | 2004-11-04 | Atkinson Robert N. | Pyrazole-amides and sulfonamides as sodium channel modulators |
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2013
- 2013-04-19 TW TW102114082A patent/TWI579274B/zh not_active IP Right Cessation
- 2013-04-22 EA EA201500483A patent/EA028539B9/ru unknown
- 2013-04-22 EA EA201401159A patent/EA025905B9/ru not_active IP Right Cessation
- 2013-04-22 ES ES13720198.4T patent/ES2626167T3/es active Active
- 2013-04-22 UA UAA201412417A patent/UA116629C2/uk unknown
- 2013-04-22 JP JP2015507247A patent/JP6197192B2/ja not_active Expired - Fee Related
- 2013-04-22 CA CA3045419A patent/CA3045419A1/en not_active Abandoned
- 2013-04-22 NZ NZ701406A patent/NZ701406A/en not_active IP Right Cessation
- 2013-04-22 SG SG11201406734TA patent/SG11201406734TA/en unknown
- 2013-04-22 BR BR112014026052A patent/BR112014026052A8/pt not_active IP Right Cessation
- 2013-04-22 MX MX2014012647A patent/MX344802B/es active IP Right Grant
- 2013-04-22 KR KR1020197014640A patent/KR102099547B1/ko active IP Right Grant
- 2013-04-22 NZ NZ709054A patent/NZ709054A/en not_active IP Right Cessation
- 2013-04-22 CA CA2870909A patent/CA2870909C/en not_active Expired - Fee Related
- 2013-04-22 AU AU2013248984A patent/AU2013248984B2/en not_active Ceased
- 2013-04-22 WO PCT/US2013/037596 patent/WO2013159094A2/en active Application Filing
- 2013-04-22 CN CN201380027759.2A patent/CN104334534B/zh not_active Expired - Fee Related
- 2013-04-22 EP EP13720198.4A patent/EP2852577B1/en active Active
- 2013-04-22 CN CN201910845886.2A patent/CN110452174A/zh active Pending
- 2013-04-22 AR ARP130101318A patent/AR090773A1/es active IP Right Grant
- 2013-04-22 MY MYPI2017000575A patent/MY177999A/en unknown
- 2013-04-22 MY MYPI2014002968A patent/MY166795A/en unknown
- 2013-04-22 US US13/867,699 patent/US8937185B2/en active Active
- 2013-04-22 KR KR1020147031914A patent/KR102027755B1/ko active IP Right Grant
- 2013-04-22 EP EP16199220.1A patent/EP3184510B1/en active Active
- 2013-04-22 SG SG10201610736YA patent/SG10201610736YA/en unknown
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2014
- 2014-10-19 IL IL235108A patent/IL235108A/en active IP Right Grant
- 2014-10-20 PH PH12014502346A patent/PH12014502346A1/en unknown
- 2014-10-20 ZA ZA2014/07603A patent/ZA201407603B/en unknown
- 2014-10-20 CL CL2014002825A patent/CL2014002825A1/es unknown
- 2014-11-17 US US14/543,341 patent/US9273007B2/en active Active
- 2014-11-20 CO CO14255092A patent/CO7141468A2/es unknown
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2016
- 2016-12-06 AU AU2016269435A patent/AU2016269435B2/en not_active Ceased
- 2016-12-20 IL IL249668A patent/IL249668A0/en active IP Right Grant
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2017
- 2017-02-20 IL IL250684A patent/IL250684B/en active IP Right Grant
- 2017-07-26 JP JP2017144256A patent/JP6494700B2/ja not_active Expired - Fee Related
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2018
- 2018-01-18 CL CL2018000151A patent/CL2018000151A1/es unknown
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2019
- 2019-10-17 AR ARP190102946A patent/AR116733A2/es unknown
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