CL2017001459A1 - Biarilo compuestos útiles para el tratamiento de enfermedades humanas en oncología, neurología e inmunología - Google Patents

Biarilo compuestos útiles para el tratamiento de enfermedades humanas en oncología, neurología e inmunología

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Publication number
CL2017001459A1
CL2017001459A1 CL2017001459A CL2017001459A CL2017001459A1 CL 2017001459 A1 CL2017001459 A1 CL 2017001459A1 CL 2017001459 A CL2017001459 A CL 2017001459A CL 2017001459 A CL2017001459 A CL 2017001459A CL 2017001459 A1 CL2017001459 A1 CL 2017001459A1
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CL
Chile
Prior art keywords
neurology
oncology
immunology
treatment
compounds useful
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CL2017001459A
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English (en)
Inventor
T Hopkins Brian
Ma Bin
Raymond Chan Timothy
Sun Lihong
Zhang Lei
Kumaravel Gnanasambandam
P Lyssikatos Joseph
Koch Kevin
Miao Hua
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Sunesis Pharmaceuticals Inc
Biogen Ma Inc
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Application filed by Sunesis Pharmaceuticals Inc, Biogen Ma Inc filed Critical Sunesis Pharmaceuticals Inc
Publication of CL2017001459A1 publication Critical patent/CL2017001459A1/es

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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P19/00Drugs for skeletal disorders
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P35/00Antineoplastic agents
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    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
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    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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Abstract

<p>La presente invención proporciona compuestos y composiciones de estos que son útiles como inhibidores de Ia tirosina cinasa de Bruton y que presentan caracterIsticas deseables para estos.</p>
CL2017001459A 2013-12-11 2017-06-08 Biarilo compuestos útiles para el tratamiento de enfermedades humanas en oncología, neurología e inmunología CL2017001459A1 (es)

Applications Claiming Priority (1)

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US201361914886P 2013-12-11 2013-12-11

Publications (1)

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CL2017001459A1 true CL2017001459A1 (es) 2018-03-23

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CL2016001435A CL2016001435A1 (es) 2013-12-11 2016-06-10 Biarilo compuestos útiles para el tratamiento de enfermedades humanas en oncologia, neurología e inmunología
CL2017001459A CL2017001459A1 (es) 2013-12-11 2017-06-08 Biarilo compuestos útiles para el tratamiento de enfermedades humanas en oncología, neurología e inmunología

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CL2016001435A CL2016001435A1 (es) 2013-12-11 2016-06-10 Biarilo compuestos útiles para el tratamiento de enfermedades humanas en oncologia, neurología e inmunología

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US (4) US9809577B2 (es)
EP (3) EP3357921A3 (es)
JP (4) JP6431914B2 (es)
KR (1) KR102413253B1 (es)
CN (3) CN108947913A (es)
AR (2) AR098721A1 (es)
AU (2) AU2014362231B2 (es)
BR (1) BR112016012860A2 (es)
CA (1) CA2932608C (es)
CL (2) CL2016001435A1 (es)
CY (1) CY1120517T1 (es)
DK (1) DK3080103T3 (es)
EA (2) EA030538B1 (es)
ES (1) ES2678021T3 (es)
HR (1) HRP20181109T1 (es)
HU (1) HUE040346T2 (es)
IL (2) IL246031B (es)
LT (1) LT3080103T (es)
MX (2) MX370103B (es)
MY (1) MY179781A (es)
NZ (1) NZ721217A (es)
PH (1) PH12016501107A1 (es)
PL (1) PL3080103T3 (es)
PT (1) PT3080103T (es)
RS (1) RS57662B1 (es)
SA (1) SA518391170B1 (es)
SG (2) SG10201908558WA (es)
SI (1) SI3080103T1 (es)
TW (3) TWI675833B (es)
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