CH636340A5 - Process for preparing novel N-(2-aminocyclopentyl)-N-alkanoyl anilides and 2-N-oxides thereof - Google Patents

Process for preparing novel N-(2-aminocyclopentyl)-N-alkanoyl anilides and 2-N-oxides thereof Download PDF

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Publication number
CH636340A5
CH636340A5 CH1461277A CH1461277A CH636340A5 CH 636340 A5 CH636340 A5 CH 636340A5 CH 1461277 A CH1461277 A CH 1461277A CH 1461277 A CH1461277 A CH 1461277A CH 636340 A5 CH636340 A5 CH 636340A5
Authority
CH
Switzerland
Prior art keywords
radical
formula
compounds
dimethylamino
cyclopentyl
Prior art date
Application number
CH1461277A
Other languages
German (de)
English (en)
Inventor
Jacob Szmuszkovicz
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of CH636340A5 publication Critical patent/CH636340A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/135—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/02—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH1461277A 1976-11-30 1977-11-29 Process for preparing novel N-(2-aminocyclopentyl)-N-alkanoyl anilides and 2-N-oxides thereof CH636340A5 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74619176A 1976-11-30 1976-11-30
US77759977A 1977-03-15 1977-03-15

Publications (1)

Publication Number Publication Date
CH636340A5 true CH636340A5 (en) 1983-05-31

Family

ID=27114572

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1461277A CH636340A5 (en) 1976-11-30 1977-11-29 Process for preparing novel N-(2-aminocyclopentyl)-N-alkanoyl anilides and 2-N-oxides thereof

Country Status (8)

Country Link
JP (1) JPS5368748A (it)
AU (1) AU511200B2 (it)
CH (1) CH636340A5 (it)
DE (1) DE2749214A1 (it)
FR (1) FR2384495A1 (it)
GB (2) GB1560218A (it)
NL (1) NL7712899A (it)
SE (1) SE441444B (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7803442A (nl) * 1978-02-09 1979-08-13 Upjohn Co Werkwijzen voor het bereiden en toepassen van amino-cycloalifatische amiden.
AU593562B2 (en) * 1985-07-22 1990-02-15 Lipha N-oxide of NN-dimethyl ethylamine, a process for its production and the pharmaceutical compositions containing it

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3510492A (en) * 1968-05-13 1970-05-05 Upjohn Co 2-anilino and 2-anilinomethyl cycloalkylamines

Also Published As

Publication number Publication date
FR2384495B1 (it) 1980-07-25
NL7712899A (nl) 1978-06-01
FR2384495A1 (fr) 1978-10-20
SE7713439L (sv) 1978-05-31
GB1560219A (en) 1980-01-30
AU511200B2 (en) 1980-07-31
JPS5368748A (en) 1978-06-19
SE441444B (sv) 1985-10-07
DE2749214A1 (de) 1978-06-01
AU3048977A (en) 1979-05-17
GB1560218A (en) 1980-01-30
DE2749214C2 (it) 1987-11-05

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Legal Events

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PL Patent ceased