CA3218491A1 - Crystalline forms of a bruton's tyrosine kinase inhibitor - Google Patents

Crystalline forms of a bruton's tyrosine kinase inhibitor

Info

Publication number
CA3218491A1
CA3218491A1 CA3218491A CA3218491A CA3218491A1 CA 3218491 A1 CA3218491 A1 CA 3218491A1 CA 3218491 A CA3218491 A CA 3218491A CA 3218491 A CA3218491 A CA 3218491A CA 3218491 A1 CA3218491 A1 CA 3218491A1
Authority
CA
Canada
Prior art keywords
sodium
pharmaceutical formulation
compound
lymphoma
theta
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CA3218491A
Other languages
English (en)
French (fr)
Inventor
Norbert Purro
Mark Smyth
Erick Goldman
David D. Wirth
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacyclics LLC
Original Assignee
Pharmacyclics LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49712527&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CA3218491(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics LLC filed Critical Pharmacyclics LLC
Publication of CA3218491A1 publication Critical patent/CA3218491A1/en
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
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  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Otolaryngology (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Mechanical Engineering (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Composite Materials (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Transplantation (AREA)
  • Heart & Thoracic Surgery (AREA)
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CA3218491A 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor Pending CA3218491A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261655381P 2012-06-04 2012-06-04
US61/655,381 2012-06-04
CA3015208A CA3015208C (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CA3015208A Division CA3015208C (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor

Publications (1)

Publication Number Publication Date
CA3218491A1 true CA3218491A1 (en) 2013-12-12

Family

ID=49712527

Family Applications (4)

Application Number Title Priority Date Filing Date
CA3015208A Active CA3015208C (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor
CA2991994A Active CA2991994C (en) 2012-06-04 2013-06-03 Pharmaceutical formulation for oral administration comprising ibrutinib
CA2875986A Active CA2875986C (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor
CA3218491A Pending CA3218491A1 (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor

Family Applications Before (3)

Application Number Title Priority Date Filing Date
CA3015208A Active CA3015208C (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor
CA2991994A Active CA2991994C (en) 2012-06-04 2013-06-03 Pharmaceutical formulation for oral administration comprising ibrutinib
CA2875986A Active CA2875986C (en) 2012-06-04 2013-06-03 Crystalline forms of a bruton's tyrosine kinase inhibitor

Country Status (32)

Country Link
US (26) US9296753B2 (enExample)
EP (1) EP2854859A4 (enExample)
JP (10) JP6236071B2 (enExample)
KR (8) KR20250151610A (enExample)
CN (2) CN104736178A (enExample)
AR (2) AR092844A1 (enExample)
AU (7) AU2013271918C1 (enExample)
BR (1) BR112014030424A8 (enExample)
CA (4) CA3015208C (enExample)
CL (3) CL2014003306A1 (enExample)
CO (1) CO7240408A2 (enExample)
CR (1) CR20140558A (enExample)
DO (3) DOP2014000274A (enExample)
EA (1) EA201492082A1 (enExample)
EC (2) ECSP14033163A (enExample)
GT (1) GT201400281A (enExample)
HK (1) HK1208803A1 (enExample)
IL (4) IL315394A (enExample)
JO (2) JO3754B1 (enExample)
MA (2) MA37711A1 (enExample)
MX (3) MX387669B (enExample)
MY (2) MY187999A (enExample)
NZ (4) NZ702548A (enExample)
PE (3) PE20150174A1 (enExample)
PH (3) PH12021552282A1 (enExample)
SG (2) SG11201408067YA (enExample)
TN (1) TN2014000492A1 (enExample)
TW (3) TWI653041B (enExample)
UA (2) UA114421C2 (enExample)
UY (2) UY34848A (enExample)
WO (1) WO2013184572A1 (enExample)
ZA (4) ZA202105175B (enExample)

Families Citing this family (126)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK2529622T3 (en) 2006-09-22 2018-05-07 Pharmacyclics Llc INHIBITORS OF BRUTON-TYROSINKINASE
US20120101114A1 (en) 2007-03-28 2012-04-26 Pharmacyclics, Inc. Inhibitors of bruton's tyrosine kinase
US20110224235A1 (en) 2008-07-16 2011-09-15 Pharmacyclics, Inc. Inhibitors of bruton's tyrosine kinase for the treatment of solid tumors
US8491927B2 (en) * 2009-12-02 2013-07-23 Nimble Epitech, Llc Pharmaceutical composition containing a hypomethylating agent and a histone deacetylase inhibitor
KR101580714B1 (ko) 2010-06-03 2016-01-04 파마싸이클릭스 엘엘씨 브루톤 티로신 인산화효소(ｂｔｋ)의 억제제의 용도
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