CA2748181C - Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders - Google Patents

Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders Download PDF

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Publication number
CA2748181C
CA2748181C CA2748181A CA2748181A CA2748181C CA 2748181 C CA2748181 C CA 2748181C CA 2748181 A CA2748181 A CA 2748181A CA 2748181 A CA2748181 A CA 2748181A CA 2748181 C CA2748181 C CA 2748181C
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pyrimido
diazepin
benzo
methoxy
phenylamino
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French (fr)
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CA2748181A1 (en
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Nathanael S. Gray
Xianming Deng
Nicholas Paul Kwiatkowski
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Dana Farber Cancer Institute Inc
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Dana Farber Cancer Institute Inc
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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CA2748181A 2009-01-06 2010-01-06 Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders Active CA2748181C (en)

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US19390109P 2009-01-06 2009-01-06
US61/193,901 2009-01-06
PCT/US2010/000050 WO2010080712A2 (en) 2009-01-06 2010-01-06 Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders

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CA2748181C true CA2748181C (en) 2019-07-16

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US9273077B2 (en) 2008-05-21 2016-03-01 Ariad Pharmaceuticals, Inc. Phosphorus derivatives as kinase inhibitors
PT2300013T (pt) 2008-05-21 2017-10-31 Ariad Pharma Inc Derivados de fósforo como inibidores de cinases
EP2379559B1 (en) * 2009-01-06 2017-10-25 Dana-Farber Cancer Institute, Inc. Pyrimido-diazepinone kinase scaffold compounds and methods of treating disorders
JP5918693B2 (ja) 2009-05-05 2016-05-18 ダナ ファーバー キャンサー インスティテュート インコーポレイテッド Ｅｇｆｒ阻害剤及び疾患の治療方法
TWI711610B (zh) 2009-09-04 2020-12-01 美商百健Ｍａ公司 布魯頓氏酪胺酸激酶抑制劑
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