CA2719457C - Arylsulfonamide-based matrix metalloprotease inhibitors - Google Patents

Arylsulfonamide-based matrix metalloprotease inhibitors Download PDF

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Publication number
CA2719457C
CA2719457C CA2719457A CA2719457A CA2719457C CA 2719457 C CA2719457 C CA 2719457C CA 2719457 A CA2719457 A CA 2719457A CA 2719457 A CA2719457 A CA 2719457A CA 2719457 C CA2719457 C CA 2719457C
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chloro
benzenesulfonamide
alkyl
aryl
mmol
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CA2719457A
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English (en)
French (fr)
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CA2719457A1 (en
Inventor
Claus Ehrhardt
Leslie Wighton Mcquire
Pascal Rigollier
Olivier Rogel
Michael Shultz
Ruben Alberto Tommasi
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Novartis AG
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Novartis AG
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    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
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US9822092B2 (en) 2017-11-21
US20130096105A1 (en) 2013-04-18
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US8222424B2 (en) 2012-07-17
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