CA2382405C - Nouveaux procedes de synthese de la (3as)-5,5-dioxo-2,3,3a,4-tetrahydro-1h-pyrrolo[2,1-c][1,2,4]benzothiadiazine - Google Patents
Nouveaux procedes de synthese de la (3as)-5,5-dioxo-2,3,3a,4-tetrahydro-1h-pyrrolo[2,1-c][1,2,4]benzothiadiazine Download PDFInfo
- Publication number
- CA2382405C CA2382405C CA002382405A CA2382405A CA2382405C CA 2382405 C CA2382405 C CA 2382405C CA 002382405 A CA002382405 A CA 002382405A CA 2382405 A CA2382405 A CA 2382405A CA 2382405 C CA2382405 C CA 2382405C
- Authority
- CA
- Canada
- Prior art keywords
- formula
- compound
- pyrrolo
- benzothiadiazine
- dioxo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR01.05226 | 2001-04-18 | ||
| FR0105226A FR2823753B1 (fr) | 2001-04-18 | 2001-04-18 | Nouveau procede de synthese de la (3as)-5,5-dioxo-2,3,3a, 4-tetrahydro-1h-pyrrolo [2,1-c] [1,2,4] benzothiadiazine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2382405A1 CA2382405A1 (fr) | 2002-10-18 |
| CA2382405C true CA2382405C (fr) | 2007-03-06 |
Family
ID=8862416
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002382405A Expired - Fee Related CA2382405C (fr) | 2001-04-18 | 2002-04-18 | Nouveaux procedes de synthese de la (3as)-5,5-dioxo-2,3,3a,4-tetrahydro-1h-pyrrolo[2,1-c][1,2,4]benzothiadiazine |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US6518422B2 (show.php) |
| EP (1) | EP1251132B1 (show.php) |
| JP (1) | JP4011956B2 (show.php) |
| KR (1) | KR100468066B1 (show.php) |
| CN (1) | CN1169811C (show.php) |
| AR (1) | AR036871A1 (show.php) |
| AT (1) | ATE269339T1 (show.php) |
| AU (1) | AU782080B2 (show.php) |
| BR (1) | BR0201307A (show.php) |
| CA (1) | CA2382405C (show.php) |
| DE (1) | DE60200627T2 (show.php) |
| DK (1) | DK1251132T3 (show.php) |
| EA (1) | EA004927B1 (show.php) |
| ES (1) | ES2223031T3 (show.php) |
| FR (1) | FR2823753B1 (show.php) |
| HU (1) | HUP0201256A3 (show.php) |
| MX (1) | MXPA02003639A (show.php) |
| NO (1) | NO20021768L (show.php) |
| NZ (1) | NZ518422A (show.php) |
| PL (1) | PL353512A1 (show.php) |
| PT (1) | PT1251132E (show.php) |
| SI (1) | SI1251132T1 (show.php) |
| ZA (1) | ZA200203085B (show.php) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2856065B1 (fr) * | 2003-06-13 | 2005-08-19 | Servier Lab | Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| US20060014887A1 (en) * | 2004-07-19 | 2006-01-19 | 3M Innovative Properties Company | Method of hydrolyzing a dispersion of ionic fluoropolymer |
| FR2879201B1 (fr) * | 2004-12-10 | 2007-02-16 | Servier Lab | Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| DK2230094T3 (en) | 2009-03-20 | 2014-03-03 | Kremstal Tuerenwerk Gmbh | Process for coating of panels |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3294791A (en) * | 1966-03-14 | 1966-12-27 | American Home Prod | Tetrahydro-2, 5-methano-1, 2, 5-benzothiadiazepine 1, 1-dioxide |
| US3471483A (en) * | 1967-11-09 | 1969-10-07 | American Home Prod | 1 - substituted - 2,3,3a - 4 - tetrahydro - 1h-pyrrolo(2,1 - c)(1,2,4)benzothiadiazine,5,5-dioxide |
| JPH06192272A (ja) * | 1992-12-24 | 1994-07-12 | Japan Tobacco Inc | 新規なトリアゾロベンゾチアジアジン及びトリアゾロベンゾチアジアゼピン誘導体 |
| FR2722502B1 (fr) * | 1994-07-12 | 1996-08-23 | Adir | Nouveau derive de benzothiadiazine, son procede depreparation et les compositions pharmaceutiques qui le contiennent |
| FR2812291B1 (fr) * | 2000-07-28 | 2002-12-13 | Adir | Nouveaux derives de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
-
2001
- 2001-04-18 FR FR0105226A patent/FR2823753B1/fr not_active Expired - Fee Related
-
2002
- 2002-04-10 MX MXPA02003639A patent/MXPA02003639A/es active IP Right Grant
- 2002-04-15 NO NO20021768A patent/NO20021768L/no not_active Application Discontinuation
- 2002-04-16 DE DE60200627T patent/DE60200627T2/de not_active Expired - Fee Related
- 2002-04-16 ES ES02290946T patent/ES2223031T3/es not_active Expired - Lifetime
- 2002-04-16 DK DK02290946T patent/DK1251132T3/da active
- 2002-04-16 JP JP2002113278A patent/JP4011956B2/ja not_active Expired - Fee Related
- 2002-04-16 EP EP02290946A patent/EP1251132B1/fr not_active Expired - Lifetime
- 2002-04-16 PT PT02290946T patent/PT1251132E/pt unknown
- 2002-04-16 SI SI200230015T patent/SI1251132T1/xx unknown
- 2002-04-16 AT AT02290946T patent/ATE269339T1/de not_active IP Right Cessation
- 2002-04-17 NZ NZ518422A patent/NZ518422A/xx unknown
- 2002-04-17 HU HU0201256A patent/HUP0201256A3/hu unknown
- 2002-04-17 AR ARP020101386A patent/AR036871A1/es not_active Application Discontinuation
- 2002-04-17 BR BR0201307-0A patent/BR0201307A/pt not_active IP Right Cessation
- 2002-04-17 EA EA200200378A patent/EA004927B1/ru not_active IP Right Cessation
- 2002-04-18 PL PL02353512A patent/PL353512A1/xx unknown
- 2002-04-18 AU AU34405/02A patent/AU782080B2/en not_active Ceased
- 2002-04-18 CA CA002382405A patent/CA2382405C/fr not_active Expired - Fee Related
- 2002-04-18 CN CNB021057907A patent/CN1169811C/zh not_active Expired - Fee Related
- 2002-04-18 KR KR10-2002-0021237A patent/KR100468066B1/ko not_active Expired - Fee Related
- 2002-04-18 US US10/125,192 patent/US6518422B2/en not_active Expired - Fee Related
- 2002-04-18 ZA ZA200203085A patent/ZA200203085B/xx unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| MKLA | Lapsed |