MXPA02003639A - Proceso nuevo para la sintesis de (3as)-5, 5-dioxo-2, 3, 3a-4- tetrahidro-1h-pirrolo[2, 1c][1, 2, 4] benzotiadiazina. - Google Patents
Proceso nuevo para la sintesis de (3as)-5, 5-dioxo-2, 3, 3a-4- tetrahidro-1h-pirrolo[2, 1c][1, 2, 4] benzotiadiazina.Info
- Publication number
- MXPA02003639A MXPA02003639A MXPA02003639A MXPA02003639A MXPA02003639A MX PA02003639 A MXPA02003639 A MX PA02003639A MX PA02003639 A MXPA02003639 A MX PA02003639A MX PA02003639 A MXPA02003639 A MX PA02003639A MX PA02003639 A MXPA02003639 A MX PA02003639A
- Authority
- MX
- Mexico
- Prior art keywords
- pyrrolo
- dioxo
- synthesis
- benothiadiazine
- new process
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Se describe un procedimiento para la sintesis industrial de (3aS)-5,5-dioxo-2,3,3a,4-tetrahidro-lH- pirrolo [2,1-c] [ 1,2,4]benzotiadiazina de formula (1) : por hidrogenacion catalitica enantioselectiva de 5,5-dioxo- 2,3-dihidro-1H-pirrolo[2,1-c] [1,2,4]benzotiadiazina.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0105226A FR2823753B1 (fr) | 2001-04-18 | 2001-04-18 | Nouveau procede de synthese de la (3as)-5,5-dioxo-2,3,3a, 4-tetrahydro-1h-pyrrolo [2,1-c] [1,2,4] benzothiadiazine |
Publications (1)
Publication Number | Publication Date |
---|---|
MXPA02003639A true MXPA02003639A (es) | 2004-11-12 |
Family
ID=8862416
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MXPA02003639A MXPA02003639A (es) | 2001-04-18 | 2002-04-10 | Proceso nuevo para la sintesis de (3as)-5, 5-dioxo-2, 3, 3a-4- tetrahidro-1h-pirrolo[2, 1c][1, 2, 4] benzotiadiazina. |
Country Status (24)
Country | Link |
---|---|
US (1) | US6518422B2 (es) |
EP (1) | EP1251132B1 (es) |
JP (1) | JP4011956B2 (es) |
KR (1) | KR100468066B1 (es) |
CN (1) | CN1169811C (es) |
AR (1) | AR036871A1 (es) |
AT (1) | ATE269339T1 (es) |
AU (1) | AU782080B2 (es) |
BR (1) | BR0201307A (es) |
CA (1) | CA2382405C (es) |
DE (1) | DE60200627T2 (es) |
DK (1) | DK1251132T3 (es) |
EA (1) | EA004927B1 (es) |
ES (1) | ES2223031T3 (es) |
FR (1) | FR2823753B1 (es) |
HK (1) | HK1049668A1 (es) |
HU (1) | HUP0201256A3 (es) |
MX (1) | MXPA02003639A (es) |
NO (1) | NO20021768L (es) |
NZ (1) | NZ518422A (es) |
PL (1) | PL353512A1 (es) |
PT (1) | PT1251132E (es) |
SI (1) | SI1251132T1 (es) |
ZA (1) | ZA200203085B (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2856065B1 (fr) * | 2003-06-13 | 2005-08-19 | Servier Lab | Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
US20060014887A1 (en) * | 2004-07-19 | 2006-01-19 | 3M Innovative Properties Company | Method of hydrolyzing a dispersion of ionic fluoropolymer |
FR2879201B1 (fr) * | 2004-12-10 | 2007-02-16 | Servier Lab | Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
EP2230094B1 (de) | 2009-03-20 | 2013-12-11 | Kremstal Türenwerk GmbH | Verfahren für das Beschichten von Plattenwerkstoffen |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3294791A (en) * | 1966-03-14 | 1966-12-27 | American Home Prod | Tetrahydro-2, 5-methano-1, 2, 5-benzothiadiazepine 1, 1-dioxide |
US3471483A (en) * | 1967-11-09 | 1969-10-07 | American Home Prod | 1 - substituted - 2,3,3a - 4 - tetrahydro - 1h-pyrrolo(2,1 - c)(1,2,4)benzothiadiazine,5,5-dioxide |
JPH06192272A (ja) * | 1992-12-24 | 1994-07-12 | Japan Tobacco Inc | 新規なトリアゾロベンゾチアジアジン及びトリアゾロベンゾチアジアゼピン誘導体 |
FR2722502B1 (fr) * | 1994-07-12 | 1996-08-23 | Adir | Nouveau derive de benzothiadiazine, son procede depreparation et les compositions pharmaceutiques qui le contiennent |
FR2812291B1 (fr) * | 2000-07-28 | 2002-12-13 | Adir | Nouveaux derives de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
-
2001
- 2001-04-18 FR FR0105226A patent/FR2823753B1/fr not_active Expired - Fee Related
-
2002
- 2002-04-10 MX MXPA02003639A patent/MXPA02003639A/es active IP Right Grant
- 2002-04-15 NO NO20021768A patent/NO20021768L/no not_active Application Discontinuation
- 2002-04-16 EP EP02290946A patent/EP1251132B1/fr not_active Expired - Lifetime
- 2002-04-16 DK DK02290946T patent/DK1251132T3/da active
- 2002-04-16 PT PT02290946T patent/PT1251132E/pt unknown
- 2002-04-16 DE DE60200627T patent/DE60200627T2/de not_active Expired - Fee Related
- 2002-04-16 JP JP2002113278A patent/JP4011956B2/ja not_active Expired - Fee Related
- 2002-04-16 AT AT02290946T patent/ATE269339T1/de not_active IP Right Cessation
- 2002-04-16 ES ES02290946T patent/ES2223031T3/es not_active Expired - Lifetime
- 2002-04-16 SI SI200230015T patent/SI1251132T1/xx unknown
- 2002-04-17 AR ARP020101386A patent/AR036871A1/es not_active Application Discontinuation
- 2002-04-17 NZ NZ518422A patent/NZ518422A/xx unknown
- 2002-04-17 BR BR0201307-0A patent/BR0201307A/pt not_active IP Right Cessation
- 2002-04-17 EA EA200200378A patent/EA004927B1/ru not_active IP Right Cessation
- 2002-04-17 HU HU0201256A patent/HUP0201256A3/hu unknown
- 2002-04-18 AU AU34405/02A patent/AU782080B2/en not_active Ceased
- 2002-04-18 CA CA002382405A patent/CA2382405C/fr not_active Expired - Fee Related
- 2002-04-18 CN CNB021057907A patent/CN1169811C/zh not_active Expired - Fee Related
- 2002-04-18 US US10/125,192 patent/US6518422B2/en not_active Expired - Fee Related
- 2002-04-18 ZA ZA200203085A patent/ZA200203085B/xx unknown
- 2002-04-18 KR KR10-2002-0021237A patent/KR100468066B1/ko not_active IP Right Cessation
- 2002-04-18 PL PL02353512A patent/PL353512A1/xx unknown
-
2003
- 2003-03-14 HK HK03101848A patent/HK1049668A1/xx not_active IP Right Cessation
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