ZA200203085B - Process for the synthesis of (3AS)-5,5-DIOXO-2,3,3A,4-tetrahydro-1H-pyrrolo [2,1-C][1,2,4]benzothiadiazine. - Google Patents

Process for the synthesis of (3AS)-5,5-DIOXO-2,3,3A,4-tetrahydro-1H-pyrrolo [2,1-C][1,2,4]benzothiadiazine.

Info

Publication number
ZA200203085B
ZA200203085B ZA200203085A ZA200203085A ZA200203085B ZA 200203085 B ZA200203085 B ZA 200203085B ZA 200203085 A ZA200203085 A ZA 200203085A ZA 200203085 A ZA200203085 A ZA 200203085A ZA 200203085 B ZA200203085 B ZA 200203085B
Authority
ZA
South Africa
Prior art keywords
benzothiadiazine
pyrrolo
dioxo
tetrahydro
synthesis
Prior art date
Application number
ZA200203085A
Other languages
English (en)
Inventor
Elsa Foucher
Gilles Thominot
Jean-Pierre Lecouve
James Andrew Ramsden
Christopher James Cobley
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of ZA200203085B publication Critical patent/ZA200203085B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
ZA200203085A 2001-04-18 2002-04-18 Process for the synthesis of (3AS)-5,5-DIOXO-2,3,3A,4-tetrahydro-1H-pyrrolo [2,1-C][1,2,4]benzothiadiazine. ZA200203085B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0105226A FR2823753B1 (fr) 2001-04-18 2001-04-18 Nouveau procede de synthese de la (3as)-5,5-dioxo-2,3,3a, 4-tetrahydro-1h-pyrrolo [2,1-c] [1,2,4] benzothiadiazine

Publications (1)

Publication Number Publication Date
ZA200203085B true ZA200203085B (en) 2002-11-25

Family

ID=8862416

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200203085A ZA200203085B (en) 2001-04-18 2002-04-18 Process for the synthesis of (3AS)-5,5-DIOXO-2,3,3A,4-tetrahydro-1H-pyrrolo [2,1-C][1,2,4]benzothiadiazine.

Country Status (24)

Country Link
US (1) US6518422B2 (es)
EP (1) EP1251132B1 (es)
JP (1) JP4011956B2 (es)
KR (1) KR100468066B1 (es)
CN (1) CN1169811C (es)
AR (1) AR036871A1 (es)
AT (1) ATE269339T1 (es)
AU (1) AU782080B2 (es)
BR (1) BR0201307A (es)
CA (1) CA2382405C (es)
DE (1) DE60200627T2 (es)
DK (1) DK1251132T3 (es)
EA (1) EA004927B1 (es)
ES (1) ES2223031T3 (es)
FR (1) FR2823753B1 (es)
HK (1) HK1049668A1 (es)
HU (1) HUP0201256A3 (es)
MX (1) MXPA02003639A (es)
NO (1) NO20021768L (es)
NZ (1) NZ518422A (es)
PL (1) PL353512A1 (es)
PT (1) PT1251132E (es)
SI (1) SI1251132T1 (es)
ZA (1) ZA200203085B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2856065B1 (fr) * 2003-06-13 2005-08-19 Servier Lab Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US20060014887A1 (en) * 2004-07-19 2006-01-19 3M Innovative Properties Company Method of hydrolyzing a dispersion of ionic fluoropolymer
FR2879201B1 (fr) * 2004-12-10 2007-02-16 Servier Lab Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
EP2230094B1 (de) 2009-03-20 2013-12-11 Kremstal Türenwerk GmbH Verfahren für das Beschichten von Plattenwerkstoffen

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3294791A (en) * 1966-03-14 1966-12-27 American Home Prod Tetrahydro-2, 5-methano-1, 2, 5-benzothiadiazepine 1, 1-dioxide
US3471483A (en) * 1967-11-09 1969-10-07 American Home Prod 1 - substituted - 2,3,3a - 4 - tetrahydro - 1h-pyrrolo(2,1 - c)(1,2,4)benzothiadiazine,5,5-dioxide
JPH06192272A (ja) * 1992-12-24 1994-07-12 Japan Tobacco Inc 新規なトリアゾロベンゾチアジアジン及びトリアゾロベンゾチアジアゼピン誘導体
FR2722502B1 (fr) * 1994-07-12 1996-08-23 Adir Nouveau derive de benzothiadiazine, son procede depreparation et les compositions pharmaceutiques qui le contiennent
FR2812291B1 (fr) * 2000-07-28 2002-12-13 Adir Nouveaux derives de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
CN1169811C (zh) 2004-10-06
HU0201256D0 (es) 2002-06-29
AU3440502A (en) 2002-10-24
PT1251132E (pt) 2004-09-30
NZ518422A (en) 2002-12-20
HUP0201256A2 (hu) 2002-12-28
MXPA02003639A (es) 2004-11-12
US6518422B2 (en) 2003-02-11
KR100468066B1 (ko) 2005-01-24
DE60200627T2 (de) 2005-07-14
DE60200627D1 (de) 2004-07-22
EA200200378A3 (ru) 2002-12-26
FR2823753B1 (fr) 2004-07-16
EA200200378A2 (ru) 2002-10-31
CN1381455A (zh) 2002-11-27
US20020161222A1 (en) 2002-10-31
PL353512A1 (en) 2002-10-21
CA2382405C (fr) 2007-03-06
AR036871A1 (es) 2004-10-13
AU782080B2 (en) 2005-06-30
NO20021768L (no) 2002-10-21
FR2823753A1 (fr) 2002-10-25
EA004927B1 (ru) 2004-10-28
CA2382405A1 (fr) 2002-10-18
HUP0201256A3 (en) 2004-11-29
BR0201307A (pt) 2003-06-10
NO20021768D0 (no) 2002-04-15
HK1049668A1 (en) 2003-05-23
KR20020081148A (ko) 2002-10-26
JP2003012674A (ja) 2003-01-15
ES2223031T3 (es) 2005-02-16
JP4011956B2 (ja) 2007-11-21
SI1251132T1 (en) 2004-10-31
EP1251132B1 (fr) 2004-06-16
EP1251132A1 (fr) 2002-10-23
DK1251132T3 (da) 2004-10-25
ATE269339T1 (de) 2004-07-15

Similar Documents

Publication Publication Date Title
AU2001259707A1 (en) 6,5-fused bicyclic heterocycles
ZA200203581B (en) Bicyclic imidazo-3-yl-amine derivatives.
ZA200110254B (en) Process for the preparation of herbicidal derivatives.
MXPA03010020A (es) PROCEDIMIETO PARA LA PREPARACIoN DE UREA.
AU4607301A (en) Ring oscillator
AU5426500A (en) Benzazepine derivatives, process for the preparation of the same and uses thereof
ZA200108392B (en) Process for the preparation of substituted pyrimidines.
IL139023A0 (en) Process for the preparation of 2,3,5-trimethyl-p- benzoquinone
MXPA02006102A (es) Metodo para preparar compuestos bormodifluoroaceticos.
ZA200203085B (en) Process for the synthesis of (3AS)-5,5-DIOXO-2,3,3A,4-tetrahydro-1H-pyrrolo [2,1-C][1,2,4]benzothiadiazine.
GB2343892B (en) Process for the preparation of d,l-menthol
AU5585700A (en) Process for making 2,4,6, 8,10,12- hexanitro- 2,4,6,8,10, 12- hexa azatetracyclo(5.5.0. 05,9.03,11} -dodecane
AU2002330042A1 (en) Process for the preparation of 1,5-diarylpyrazoles
HUP0402475A3 (en) Process for the preparation of [1,4,5]-oxadiazepine derivatives
MXPA03002926A (es) Proceso para la sintesis de 2,2,6,6,-tetrametil-4--oxipiperidina.
AU2001286188A1 (en) Tricyclic heterocyclic compound, process for producing the same, and use thereof
AU6870500A (en) Process for the preparation of 2,3-dihydroazepine derivatives
AU6870600A (en) Process for the preparation of 2,3-dihydroazepine compounds
AU2002359412A1 (en) Process for the preparation of 3,7-disubstituted-2,3,4,5- tetrahydro-1h-1,4-benzodiazepine compounds
AU2001262240A1 (en) Process for the production of 2,2,6-trimethylcyclohexane-1,4-dione
AU2001282403A1 (en) An improved process for the preparation of 3,4-dihydro-1,4-benzothiazine
MXPA03006508A (es) Proceso para preparacion de derivado de pirazolo (4,3-d) pirimidina.
MXPA01001471A (es) Nuevo proceso para la sintesis de exoquelinas.
AU4777500A (en) Processes for the preparation of 2,3-dihydrothiepine derivatives
HK1041606A1 (en) Process for the preparation of n,n'-carbonylbislactams.