CA2323678A1 - Process for the preparation of a tetrapeptide - Google Patents

Process for the preparation of a tetrapeptide Download PDF

Info

Publication number
CA2323678A1
CA2323678A1 CA002323678A CA2323678A CA2323678A1 CA 2323678 A1 CA2323678 A1 CA 2323678A1 CA 002323678 A CA002323678 A CA 002323678A CA 2323678 A CA2323678 A CA 2323678A CA 2323678 A1 CA2323678 A1 CA 2323678A1
Authority
CA
Canada
Prior art keywords
phe
derivative
group
ester
process according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002323678A
Other languages
English (en)
French (fr)
Inventor
Henry Franzen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca AB
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2323678A1 publication Critical patent/CA2323678A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10Tetrapeptides
    • C07K5/1002Tetrapeptides with the first amino acid being neutral
    • C07K5/1016Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10Tetrapeptides
    • C07K5/1027Tetrapeptides containing heteroatoms different from O, S, or N

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CA002323678A 1998-03-16 1999-03-16 Process for the preparation of a tetrapeptide Abandoned CA2323678A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE9800865-9 1998-03-16
SE9800865A SE9800865D0 (sv) 1998-03-16 1998-03-16 New Process
PCT/SE1999/000414 WO1999047548A1 (en) 1998-03-16 1999-03-16 Process for the preparation of a tetrapeptide

Publications (1)

Publication Number Publication Date
CA2323678A1 true CA2323678A1 (en) 1999-09-23

Family

ID=20410566

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002323678A Abandoned CA2323678A1 (en) 1998-03-16 1999-03-16 Process for the preparation of a tetrapeptide

Country Status (19)

Country Link
EP (1) EP1062231A1 (ko)
JP (1) JP2002506880A (ko)
KR (1) KR20010041888A (ko)
CN (1) CN1300293A (ko)
AU (1) AU2968899A (ko)
BR (1) BR9908765A (ko)
CA (1) CA2323678A1 (ko)
EE (1) EE200000540A (ko)
HU (1) HUP0102877A3 (ko)
ID (1) ID26938A (ko)
IL (1) IL138244A0 (ko)
IS (1) IS5612A (ko)
NO (1) NO20004613L (ko)
PL (1) PL343277A1 (ko)
SE (1) SE9800865D0 (ko)
SK (1) SK13442000A3 (ko)
TR (1) TR200002652T2 (ko)
WO (1) WO1999047548A1 (ko)
ZA (1) ZA200004376B (ko)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9903291D0 (sv) * 1999-09-15 1999-09-15 Astra Ab New process
WO2009076672A1 (en) * 2007-12-13 2009-06-18 Cytogel, Llc Advantageous salts of mu-opiate receptor peptides
CN104371002B (zh) * 2013-06-20 2017-10-10 重庆理工大学 一种非蛋白氨基酸抗菌肽及其应用
CN104478993B (zh) * 2013-06-20 2017-10-10 重庆理工大学 一种非蛋白氨基酸抗菌肽及其应用
CN103319568B (zh) * 2013-06-20 2015-01-21 重庆理工大学 一种非蛋白氨基酸抗菌肽及其应用
CN104783298A (zh) * 2015-03-24 2015-07-22 湖州珍贝羊绒制品有限公司 一种生物灭菌组合物及其纳米乳的制备与应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9503924D0 (sv) * 1995-08-18 1995-11-07 Astra Ab Novel opioid peptides
GB9516994D0 (en) * 1995-08-18 1995-10-18 Iaf Biochem Int Solution synthesis of peripheral acting analgestic opioid tetrapeptides

Also Published As

Publication number Publication date
NO20004613L (no) 2000-10-30
NO20004613D0 (no) 2000-09-15
HUP0102877A3 (en) 2002-02-28
IL138244A0 (en) 2001-10-31
JP2002506880A (ja) 2002-03-05
TR200002652T2 (tr) 2000-11-21
PL343277A1 (en) 2001-08-13
KR20010041888A (ko) 2001-05-25
HUP0102877A2 (hu) 2002-01-28
WO1999047548A1 (en) 1999-09-23
BR9908765A (pt) 2000-11-07
IS5612A (is) 2000-08-30
SK13442000A3 (sk) 2001-04-09
ID26938A (id) 2001-02-22
SE9800865D0 (sv) 1998-03-16
CN1300293A (zh) 2001-06-20
ZA200004376B (en) 2001-10-31
EE200000540A (et) 2002-02-15
AU2968899A (en) 1999-10-11
EP1062231A1 (en) 2000-12-27

Similar Documents

Publication Publication Date Title
EP1212350A1 (en) A process for the preparation of h-tyr-d-ala-phe(f)-phe-nh 2?
GB2058079A (en) TRH analogues
KR100607556B1 (ko) (2S, 3aS,7aS)-1-[(S)-알라닐]-옥타히드로-1H-인돌-2-카르복실산유도체의 신규한 합성 방법 및 페린도프릴 합성에서의이의 용도
CA2323678A1 (en) Process for the preparation of a tetrapeptide
JP5445456B2 (ja) ジベンゾフルベンの除去方法
AU2002310004A1 (en) Uronium and immonium salts for peptide coupling
WO2002094822A1 (en) Uronium and immonium salts for peptide coupling
JP4331207B2 (ja) ペリンドプリルおよびその薬学的に許容され得る塩の、新規な合成方法
KR100825537B1 (ko) 페린도프릴 및 이의 약학적으로 허용되는 염의 합성 방법
JP4331206B2 (ja) ペリンドプリルおよびその薬学的に許容され得る塩の、新規な合成方法
HU221619B1 (hu) Eljárás peptidek előállítására és intermedierek
EP0410182A2 (en) A new technique for rapid peptide coupling
MXPA00008828A (en) Process for the preparation of a tetrapeptide
PL211506B1 (pl) Sposób otrzymywania związków kwasu (2S, 3aS, 7aS)-1-[(S)-alanilo]-oktahydro-1H-indolo-2-karboksylowego i ich zastosowanie w syntezie perindoprilu oraz związek przejściowy
CZ20003342A3 (cs) Způsob přípravy tetrapeptidu
JP4290844B2 (ja) テアニンの製造方法
DK149631B (da) Fremgangsmaade til fremstilling af h-sar-lys-sar-gln-nh2
RU2111972C1 (ru) СПОСОБ ПОЛУЧЕНИЯ ПЕПТИДА δ СНА
JP3554399B2 (ja) ペプチド誘導体
JP5982720B2 (ja) 高分子固体状支持体を用いたヒスチジル−プロリンアミド誘導体の製造方法
EP0564587A4 (en) Solution phase process for synthesis of peptide
JPH0786102B2 (ja) 光学活性な6−(4−イミダゾリルメチル)−3−置換−2,5−ピペラジンジオンの製造法
HU179926B (hu) Eljárás a gasztrin C-terminális tetrapeptid-szekvenciájának előállítására
JPH085812B2 (ja) 酸アミド化合物の製造方法
JPS63215697A (ja) 弛緩ペプチドおよびその製造方法

Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued