CA2089955A1 - Arylcarbonylaminoalkyl-dihydro-oxo-pyridines, their production and their use - Google Patents
Arylcarbonylaminoalkyl-dihydro-oxo-pyridines, their production and their useInfo
- Publication number
- CA2089955A1 CA2089955A1 CA002089955A CA2089955A CA2089955A1 CA 2089955 A1 CA2089955 A1 CA 2089955A1 CA 002089955 A CA002089955 A CA 002089955A CA 2089955 A CA2089955 A CA 2089955A CA 2089955 A1 CA2089955 A1 CA 2089955A1
- Authority
- CA
- Canada
- Prior art keywords
- oxo
- dihydro
- methyl ester
- loweralkyl
- aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/80—Acids; Esters in position 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP92102828 | 1992-02-20 | ||
| EP92102828.8 | 1992-02-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2089955A1 true CA2089955A1 (en) | 1993-08-21 |
Family
ID=8209352
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002089955A Abandoned CA2089955A1 (en) | 1992-02-20 | 1993-02-19 | Arylcarbonylaminoalkyl-dihydro-oxo-pyridines, their production and their use |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US5360808A (en10) |
| EP (1) | EP0556738B1 (en10) |
| JP (1) | JPH069560A (en10) |
| KR (1) | KR930017895A (en10) |
| CN (1) | CN1075480A (en10) |
| AT (1) | ATE122659T1 (en10) |
| AU (1) | AU3375993A (en10) |
| CA (1) | CA2089955A1 (en10) |
| CZ (1) | CZ403592A3 (en10) |
| DE (1) | DE69300152D1 (en10) |
| FI (1) | FI930716A (en10) |
| HU (1) | HU9300463D0 (en10) |
| IL (1) | IL104781A0 (en10) |
| MA (1) | MA22806A1 (en10) |
| MX (1) | MX9300915A (en10) |
| NO (1) | NO930594L (en10) |
| ZA (1) | ZA931185B (en10) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020052295A1 (en) * | 1999-12-21 | 2002-05-02 | Hegde Shridhar G. | Diacyl derivatives of propylene diamine having herbicidal activity |
| DE10205219A1 (de) * | 2002-02-08 | 2003-08-21 | Bayer Ag | Chinoxalinone und ihre Verwendung |
| US6869966B2 (en) * | 2002-09-30 | 2005-03-22 | Banyu Pharmaceutical Co., Ltd. | N-substituted-2-oxodihydropyridine derivatives |
| US20040127129A1 (en) * | 2002-12-31 | 2004-07-01 | Shuiyuan Luo | Grooved-shape monofilaments and the fabrics made thereof |
| WO2007008963A1 (en) * | 2005-07-13 | 2007-01-18 | Jenrin Discovery | Mao-b inhibitors useful for treating obesity |
| EP2114898A2 (en) * | 2007-02-16 | 2009-11-11 | Amgen Inc. | Nitrogen-containing heterocyclyl ketones and their use as c-met inhibitors |
| US8153808B2 (en) | 2008-12-23 | 2012-04-10 | Roche Palo Alto Llc | Dihydropyridone amides as P2X7 modulators |
| WO2010072599A1 (en) | 2008-12-23 | 2010-07-01 | F. Hoffmann-La Roche Ag | Dihydropyridone ureas as p2x7 modulators |
| CA2745952A1 (en) | 2008-12-23 | 2010-07-01 | F.Hoffmann-La Roche Ag | Dihydropyridone amides as p2x7 modulators |
| KR101381074B1 (ko) | 2008-12-23 | 2014-04-11 | 에프. 호프만-라 로슈 아게 | Ｐ2ｘ7 조절제로서의 디히드로피리돈 아미드 |
| SG172785A1 (en) | 2008-12-23 | 2011-08-29 | Hoffmann La Roche | Dihydropyridone amides as p2x7 modulators |
| WO2011023696A1 (en) | 2009-08-26 | 2011-03-03 | Nycomed Gmbh | Methylpyrrolopyridinecarboxamides |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2637477A1 (de) * | 1976-08-20 | 1978-02-23 | Hoechst Ag | Dihydro-oxo-nicotinsaeuren und verfahren zu ihrer herstellung |
| US4297360A (en) * | 1980-03-28 | 1981-10-27 | Sterling Drug Inc. | 5-(Pyridinyl)pyridine-2,3-diamines, preparation thereof and their cardiotonic use |
| NZ195564A (en) * | 1979-11-26 | 1983-09-30 | Sterling Drug Inc | 5-pyridinyl-2(1h)-pyridinones pharmaceutical compositions intermediate pyridine compounds |
| IT8367883A0 (it) * | 1982-08-23 | 1983-08-22 | Rorer Int Overseas | Composti cardiotonici del 2 piridone 5 biciclico eteroaril sostituito e relative composizioni farmaceutiche |
| GB8809481D0 (en) * | 1988-04-21 | 1988-05-25 | Smith Kline French Lab | Chemical compounds |
-
1992
- 1992-12-31 CZ CS924035A patent/CZ403592A3/cs unknown
-
1993
- 1993-02-12 EP EP93102220A patent/EP0556738B1/en not_active Expired - Lifetime
- 1993-02-12 DE DE69300152T patent/DE69300152D1/de not_active Expired - Lifetime
- 1993-02-12 AT AT93102220T patent/ATE122659T1/de not_active IP Right Cessation
- 1993-02-18 US US08/019,296 patent/US5360808A/en not_active Expired - Fee Related
- 1993-02-18 FI FI930716A patent/FI930716A/fi not_active Application Discontinuation
- 1993-02-18 KR KR1019930002218A patent/KR930017895A/ko not_active Application Discontinuation
- 1993-02-18 IL IL104781A patent/IL104781A0/xx unknown
- 1993-02-19 ZA ZA931185A patent/ZA931185B/xx unknown
- 1993-02-19 NO NO93930594A patent/NO930594L/no unknown
- 1993-02-19 MA MA23099A patent/MA22806A1/fr unknown
- 1993-02-19 CN CN93101816A patent/CN1075480A/zh active Pending
- 1993-02-19 AU AU33759/93A patent/AU3375993A/en not_active Abandoned
- 1993-02-19 JP JP5029515A patent/JPH069560A/ja active Pending
- 1993-02-19 MX MX9300915A patent/MX9300915A/es unknown
- 1993-02-19 CA CA002089955A patent/CA2089955A1/en not_active Abandoned
- 1993-02-19 HU HU9300463A patent/HU9300463D0/hu unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE69300152D1 (de) | 1995-06-22 |
| EP0556738B1 (en) | 1995-05-17 |
| EP0556738A1 (en) | 1993-08-25 |
| MX9300915A (es) | 1993-09-01 |
| ZA931185B (en) | 1993-09-16 |
| NO930594D0 (no) | 1993-02-19 |
| CZ403592A3 (en) | 1993-12-15 |
| AU3375993A (en) | 1993-08-26 |
| US5360808A (en) | 1994-11-01 |
| IL104781A0 (en) | 1993-06-10 |
| KR930017895A (ko) | 1993-09-20 |
| FI930716A (fi) | 1993-08-21 |
| NO930594L (no) | 1993-08-23 |
| JPH069560A (ja) | 1994-01-18 |
| ATE122659T1 (de) | 1995-06-15 |
| FI930716A0 (fi) | 1993-02-18 |
| HU9300463D0 (en) | 1993-05-28 |
| CN1075480A (zh) | 1993-08-25 |
| MA22806A1 (fr) | 1993-10-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |