CA1323032C - Process for preparing 2-guanidinothiazole derivatives - Google Patents

Process for preparing 2-guanidinothiazole derivatives

Info

Publication number
CA1323032C
CA1323032C CA000549936A CA549936A CA1323032C CA 1323032 C CA1323032 C CA 1323032C CA 000549936 A CA000549936 A CA 000549936A CA 549936 A CA549936 A CA 549936A CA 1323032 C CA1323032 C CA 1323032C
Authority
CA
Canada
Prior art keywords
formula
group
compound
iii
solvent
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CA000549936A
Other languages
English (en)
French (fr)
Inventor
Erik Bogsch
Ferenc Trischler
Peter Bod
Kalman Harsanyi
Eva Againe Csongor
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Richter Gedeon Vegyeszeti Gyar Nyrt
Original Assignee
Richter Gedeon Vegyeszeti Gyar RT
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszeti Gyar RT filed Critical Richter Gedeon Vegyeszeti Gyar RT
Application granted granted Critical
Publication of CA1323032C publication Critical patent/CA1323032C/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/28—Radicals substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/50—Nitrogen atoms bound to hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
CA000549936A 1986-11-12 1987-10-21 Process for preparing 2-guanidinothiazole derivatives Expired - Fee Related CA1323032C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU4658/86 1986-11-12
HU864658A HU195959B (en) 1986-11-12 1986-11-12 Process for producing 2-guanidino-thiazole derivatives

Publications (1)

Publication Number Publication Date
CA1323032C true CA1323032C (en) 1993-10-12

Family

ID=10968597

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000549936A Expired - Fee Related CA1323032C (en) 1986-11-12 1987-10-21 Process for preparing 2-guanidinothiazole derivatives

Country Status (14)

Country Link
KR (1) KR900006556B1 (hu)
AR (1) AR243874A1 (hu)
AT (1) AT389510B (hu)
CA (1) CA1323032C (hu)
CS (1) CS268693B2 (hu)
DK (1) DK169966B1 (hu)
ES (1) ES2005441A6 (hu)
FI (1) FI84912C (hu)
GR (1) GR871696B (hu)
HU (1) HU195959B (hu)
NO (1) NO167387C (hu)
PT (1) PT86113B (hu)
SU (1) SU1678205A3 (hu)
YU (1) YU46086B (hu)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5856500A (en) * 1997-03-11 1999-01-05 Albemarle Corporation Synthesis of thiazole derivatives
US5731442A (en) * 1997-03-11 1998-03-24 Albemarle Corporation Synthesis of thiazole derivatives

Also Published As

Publication number Publication date
GR871696B (en) 1987-12-08
SU1678205A3 (ru) 1991-09-15
KR900006556B1 (ko) 1990-09-13
AT389510B (de) 1989-12-27
FI875003A (fi) 1988-06-13
PT86113B (pt) 1990-08-31
YU46086B (sh) 1992-12-21
YU204987A (en) 1988-10-31
FI875003A0 (fi) 1987-11-12
NO874698D0 (no) 1987-11-11
AR243874A1 (es) 1993-09-30
FI84912B (fi) 1991-10-31
NO167387C (no) 1991-10-30
CS268693B2 (en) 1990-04-11
DK587287D0 (da) 1987-11-10
DK587287A (da) 1988-05-13
HU195959B (en) 1988-08-29
ES2005441A6 (es) 1989-03-01
FI84912C (fi) 1992-02-10
CS810187A2 (en) 1989-07-12
DK169966B1 (da) 1995-04-18
ATA277087A (de) 1989-05-15
PT86113A (en) 1987-12-01
KR890008120A (ko) 1989-07-08
NO167387B (no) 1991-07-22
NO874698L (no) 1988-05-13

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Legal Events

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