CA1175415A - Procede de preparation de nouveaux derives steroides 3-amino substitue - Google Patents

Procede de preparation de nouveaux derives steroides 3-amino substitue

Info

Publication number
CA1175415A
CA1175415A CA000390559A CA390559A CA1175415A CA 1175415 A CA1175415 A CA 1175415A CA 000390559 A CA000390559 A CA 000390559A CA 390559 A CA390559 A CA 390559A CA 1175415 A CA1175415 A CA 1175415A
Authority
CA
Canada
Prior art keywords
radical
alpha
amino
methyl
carbon atoms
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000390559A
Other languages
English (en)
French (fr)
Inventor
Roger Deraedt
Vesperto Torelli
Josette Benzoni
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Application granted granted Critical
Publication of CA1175415A publication Critical patent/CA1175415A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
    • C07J13/007—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 17 (20)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0027—Azides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA000390559A 1980-11-21 1981-11-20 Procede de preparation de nouveaux derives steroides 3-amino substitue Expired CA1175415A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8024750A FR2494698A1 (fr) 1980-11-21 1980-11-21 Nouveaux derives steroides 3-amino substitues, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant
FR80-24750 1980-11-21

Publications (1)

Publication Number Publication Date
CA1175415A true CA1175415A (fr) 1984-10-02

Family

ID=9248226

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000390559A Expired CA1175415A (fr) 1980-11-21 1981-11-20 Procede de preparation de nouveaux derives steroides 3-amino substitue

Country Status (23)

Country Link
JP (1) JPS57116099A (nl)
KR (1) KR880001239B1 (nl)
AT (1) AT389703B (nl)
AU (1) AU546100B2 (nl)
BE (1) BE891201A (nl)
CA (1) CA1175415A (nl)
CH (1) CH651056A5 (nl)
DE (1) DE3146117A1 (nl)
DK (1) DK161093C (nl)
ES (1) ES8207195A1 (nl)
FI (1) FI77871C (nl)
FR (1) FR2494698A1 (nl)
GB (1) GB2087894B (nl)
HU (1) HU184896B (nl)
IE (1) IE52188B1 (nl)
IL (1) IL64224A0 (nl)
IT (1) IT1172086B (nl)
LU (1) LU83781A1 (nl)
NL (1) NL8105260A (nl)
PT (1) PT74015B (nl)
SE (1) SE451456B (nl)
SU (1) SU1327789A3 (nl)
ZA (1) ZA817806B (nl)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9084800B2 (en) * 2011-11-07 2015-07-21 Natreon, Inc. Indolealkylamino-withasteroid conjugates and method of use

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2430467A (en) * 1944-02-11 1947-11-11 Glidden Co 3-amino-derivatives of steroids and method of making same
US2781342A (en) * 1952-05-17 1957-02-12 Upjohn Co Steroid enamines
GB962324A (en) * 1959-09-12 1964-07-01 Clin Byla Ets Steroid compounds and production thereof
FR1311761A (fr) * 1959-09-12 1962-12-14 Clin Byla Ets Composés aminés de la série des stéroïdes et procédé de préparation de tels composés
NL103735C (nl) * 1961-02-17
US3503959A (en) * 1962-03-30 1970-03-31 Sterling Drug Inc 3-amino steroids
US3196168A (en) * 1964-02-18 1965-07-20 American Home Prod Aminoaroyl aminosteroids
BE647858A (nl) * 1964-05-13
US3196169A (en) * 1964-11-03 1965-07-20 American Home Prod Aminoacyl aminosteroids
BE672238A (nl) * 1965-11-12 1966-03-01
BE811304R (fr) * 1973-10-24 1974-06-17 Pr0cede de preparation du (20 s) 3 beta -n-dimethylamino
FR2463777A1 (fr) * 1979-08-17 1981-02-27 Roussel Uclaf Nouveaux derives du 5a-pregnan-20-ol, leur procede de preparation et leur application comme medicaments

Also Published As

Publication number Publication date
DK161093C (da) 1991-11-18
IT8149746A0 (it) 1981-11-20
AU7772381A (en) 1982-05-27
ATA497081A (de) 1989-06-15
SU1327789A3 (ru) 1987-07-30
AU546100B2 (en) 1985-08-15
DK514981A (da) 1982-05-22
FR2494698A1 (fr) 1982-05-28
HU184896B (en) 1984-10-29
BE891201A (fr) 1982-05-21
AT389703B (de) 1990-01-25
PT74015A (fr) 1981-12-01
FR2494698B1 (nl) 1983-06-24
GB2087894B (en) 1984-09-26
IE812732L (en) 1982-05-21
FI77871C (fi) 1989-05-10
NL8105260A (nl) 1982-06-16
KR830007716A (ko) 1983-11-04
ES507309A0 (es) 1982-09-01
SE8105995L (sv) 1982-05-22
FI77871B (fi) 1989-01-31
SE451456B (sv) 1987-10-12
IE52188B1 (en) 1987-08-05
CH651056A5 (fr) 1985-08-30
FI813677L (fi) 1982-05-22
DK161093B (da) 1991-05-27
PT74015B (fr) 1983-11-30
LU83781A1 (fr) 1982-06-30
GB2087894A (en) 1982-06-03
JPS57116099A (en) 1982-07-19
IT1172086B (it) 1987-06-18
ES8207195A1 (es) 1982-09-01
KR880001239B1 (ko) 1988-07-12
IL64224A0 (en) 1982-02-28
JPH0247479B2 (nl) 1990-10-19
DE3146117A1 (de) 1982-06-16
ZA817806B (en) 1982-10-27

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Legal Events

Date Code Title Description
MKEC Expiry (correction)
MKEX Expiry